KR20120042766A - 지방산 아마이드 가수분해효소 억제제로서의 이속사졸린 - Google Patents

지방산 아마이드 가수분해효소 억제제로서의 이속사졸린 Download PDF

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KR20120042766A
KR20120042766A KR1020117030377A KR20117030377A KR20120042766A KR 20120042766 A KR20120042766 A KR 20120042766A KR 1020117030377 A KR1020117030377 A KR 1020117030377A KR 20117030377 A KR20117030377 A KR 20117030377A KR 20120042766 A KR20120042766 A KR 20120042766A
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South Korea
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alkyl
certain embodiments
aryl
independently
alkenyl
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Korean (ko)
Inventor
마크 엘 벤크
알프레도 씨 카스트로
로렌스 케이 찬
캐서린 에이 에반스
루이스 그레니어
마이클 제이 그로간
이브스 르블랑
타오 리우
스테판 페루소
다니엘 에이 스나이더
토마스 티 티비츠
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인피니티 파마슈티칼스, 인코포레이티드
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Publication of KR20120042766A publication Critical patent/KR20120042766A/ko
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Anesthesiology (AREA)
  • Vascular Medicine (AREA)
KR1020117030377A 2009-05-18 2010-05-18 지방산 아마이드 가수분해효소 억제제로서의 이속사졸린 Withdrawn KR20120042766A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US17928509P 2009-05-18 2009-05-18
US17928309P 2009-05-18 2009-05-18
US17928009P 2009-05-18 2009-05-18
US61/179,285 2009-05-18
US61/179,283 2009-05-18
US61/179,280 2009-05-18

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KR20120042766A true KR20120042766A (ko) 2012-05-03

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EP (1) EP2432771A4 (enExample)
JP (1) JP2012527467A (enExample)
KR (1) KR20120042766A (enExample)
CN (1) CN102459202B (enExample)
AR (1) AR076687A1 (enExample)
AU (1) AU2010249674A1 (enExample)
BR (1) BRPI1011049A2 (enExample)
CA (1) CA2762527A1 (enExample)
IL (1) IL216420A0 (enExample)
MX (1) MX2011012263A (enExample)
NZ (2) NZ619076A (enExample)
RU (1) RU2539595C2 (enExample)
SG (2) SG176168A1 (enExample)
TW (1) TW201043620A (enExample)
WO (1) WO2010135360A1 (enExample)
ZA (1) ZA201108657B (enExample)

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US20130150346A1 (en) 2010-01-08 2013-06-13 Quest Ventures Ltd. Use of FAAH Inhibitors for Treating Parkinson's Disease and Restless Legs Syndrome
WO2011123719A2 (en) 2010-03-31 2011-10-06 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating abdominal, visceral and pelvic pain
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WO2018112843A1 (en) 2016-12-22 2018-06-28 Merck Sharp & Dohme Corp. Heteroaryl piperidine ether allosteric modulators of the m4 muscarinic acetylcholine receptor
JP7052798B2 (ja) 2017-08-10 2022-04-12 大正製薬株式会社 アゾールで置換されたピリジン化合物
US10485790B1 (en) 2018-09-13 2019-11-26 Syneurx International (Taiwan) Corp. Salts of cycloserine compounds and applications thereof
US12698259B2 (en) 2018-10-15 2026-08-04 Dana-Farber Cancer Institute, Inc. Transcriptional enhanced associate domain (TEAD) transcription factor inhibitors and uses thereof
CN110016142B (zh) * 2019-04-30 2021-08-03 合肥工业大学 一种含嘧啶硼酸结构的硅油及其制备方法
US11458149B1 (en) 2019-05-31 2022-10-04 Ikena Oncology, Inc. TEAD inhibitors and uses thereof
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US12595239B2 (en) 2021-02-11 2026-04-07 Basf Se Substituted isoxazoline derivatives
KR20240111312A (ko) 2021-10-25 2024-07-16 카이메라 쎄라퓨틱스 인코포레이티드 Tyk2 분해제 및 이의 용도
EP4238971A1 (en) 2022-03-02 2023-09-06 Basf Se Substituted isoxazoline derivatives
US20250163037A1 (en) 2022-03-02 2025-05-22 Basf Se Substituted isoxazoline derivatives
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WO2024061665A1 (en) 2022-09-20 2024-03-28 Basf Se N-(3-(aminomethyl)-phenyl)-5-(4-phenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-amine derivatives and similar compounds as pesticides
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CA2762527A1 (en) 2010-11-25
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