KR20110008263A - 치료제로서의 치환된 감마 락탐 - Google Patents
치료제로서의 치환된 감마 락탐 Download PDFInfo
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- KR20110008263A KR20110008263A KR1020107026219A KR20107026219A KR20110008263A KR 20110008263 A KR20110008263 A KR 20110008263A KR 1020107026219 A KR1020107026219 A KR 1020107026219A KR 20107026219 A KR20107026219 A KR 20107026219A KR 20110008263 A KR20110008263 A KR 20110008263A
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- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
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- A61P27/00—Drugs for disorders of the senses
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- A61P27/06—Antiglaucoma agents or miotics
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
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- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyrrole Compounds (AREA)
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| US9216183B2 (en) | 2002-02-04 | 2015-12-22 | Allergan, Inc. | Topical treatment for chemotherapy induced eyelash loss or hypotrichosis using prostamide F2 alpha agonists |
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| US8673341B2 (en) | 2004-04-30 | 2014-03-18 | Allergan, Inc. | Intraocular pressure reduction with intracameral bimatoprost implants |
| US7993634B2 (en) | 2004-04-30 | 2011-08-09 | Allergan, Inc. | Oil-in-oil emulsified polymeric implants containing a hypotensive lipid and related methods |
| US7799336B2 (en) | 2004-04-30 | 2010-09-21 | Allergan, Inc. | Hypotensive lipid-containing biodegradable intraocular implants and related methods |
| US9498457B2 (en) | 2004-04-30 | 2016-11-22 | Allergan, Inc. | Hypotensive prostamide-containing biodegradable intraocular implants and related implants |
| US8377984B2 (en) * | 2008-01-29 | 2013-02-19 | Allergan, Inc. | Substituted gamma lactams as therapeutic agents |
| US9192571B2 (en) * | 2008-03-03 | 2015-11-24 | Allergan, Inc. | Ketorolac tromethamine compositions for treating or preventing ocular pain |
| US7842714B2 (en) * | 2008-03-03 | 2010-11-30 | Allergan, Inc. | Ketorolac tromethamine compositions for treating ocular pain |
| CA2721749A1 (en) * | 2008-04-16 | 2009-10-22 | Allergan, Inc. | Combination therapy for glaucoma |
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| US6034413A (en) * | 1997-02-27 | 2000-03-07 | Texas Instruments Incorporated | High speed biCMOS gate power for power MOSFETs incorporating improved injection immunity |
| US6437146B1 (en) | 1998-09-25 | 2002-08-20 | Fujisawa Pharmaceutical Co., Ltd. | Oxazole compounds as prostaglandin e2 agonists or antagonists |
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2009
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- 2009-04-22 RU RU2010144637/04A patent/RU2543379C2/ru active
- 2009-04-22 WO PCT/US2009/041389 patent/WO2009132088A1/en not_active Ceased
- 2009-04-22 PL PL09734653T patent/PL2291368T3/pl unknown
- 2009-04-22 BR BRPI0911347A patent/BRPI0911347A2/pt not_active IP Right Cessation
- 2009-04-22 AU AU2009239372A patent/AU2009239372B2/en not_active Ceased
- 2009-04-22 MY MYPI20105007 patent/MY150518A/en unknown
- 2009-04-22 KR KR1020107026219A patent/KR20110008263A/ko not_active Ceased
- 2009-04-22 US US12/427,968 patent/US7820661B2/en active Active
- 2009-04-22 EP EP09734653A patent/EP2291368B1/en active Active
- 2009-04-22 CA CA2722529A patent/CA2722529A1/en not_active Abandoned
- 2009-04-22 DK DK09734653.0T patent/DK2291368T3/da active
- 2009-04-22 JP JP2011506415A patent/JP5524181B2/ja not_active Expired - Fee Related
- 2009-04-22 UA UAA201013802A patent/UA103616C2/ru unknown
- 2009-04-22 ES ES09734653T patent/ES2399314T3/es active Active
- 2009-04-22 MX MX2010011636A patent/MX2010011636A/es active IP Right Grant
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2010
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Also Published As
| Publication number | Publication date |
|---|---|
| IL208899A0 (en) | 2011-01-31 |
| JP2011518833A (ja) | 2011-06-30 |
| MY150518A (en) | 2014-01-30 |
| US7820661B2 (en) | 2010-10-26 |
| RU2010144637A (ru) | 2012-05-27 |
| US20090270392A1 (en) | 2009-10-29 |
| MX2010011636A (es) | 2010-11-25 |
| BRPI0911347A2 (pt) | 2018-03-20 |
| EP2291368B1 (en) | 2012-12-19 |
| CA2722529A1 (en) | 2009-10-29 |
| ES2399314T3 (es) | 2013-03-27 |
| UA103616C2 (ru) | 2013-11-11 |
| RU2543379C2 (ru) | 2015-02-27 |
| EP2291368A1 (en) | 2011-03-09 |
| AU2009239372B2 (en) | 2013-09-19 |
| DK2291368T3 (da) | 2013-03-18 |
| JP5524181B2 (ja) | 2014-06-18 |
| CO6321273A2 (es) | 2011-09-20 |
| ZA201007553B (en) | 2011-08-31 |
| WO2009132088A1 (en) | 2009-10-29 |
| AU2009239372A1 (en) | 2009-10-29 |
| CN102076681A (zh) | 2011-05-25 |
| PL2291368T3 (pl) | 2013-05-31 |
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