KR20100086981A - 항당뇨 의약 조성물 - Google Patents
항당뇨 의약 조성물 Download PDFInfo
- Publication number
- KR20100086981A KR20100086981A KR1020107004947A KR20107004947A KR20100086981A KR 20100086981 A KR20100086981 A KR 20100086981A KR 1020107004947 A KR1020107004947 A KR 1020107004947A KR 20107004947 A KR20107004947 A KR 20107004947A KR 20100086981 A KR20100086981 A KR 20100086981A
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- KR
- South Korea
- Prior art keywords
- pharmaceutical composition
- methyl
- optionally substituted
- carbetoxy
- hydroxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Images
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/405—Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2007134267/15A RU2361581C2 (ru) | 2007-09-14 | 2007-09-14 | Фармацевтическая композиция, обладающая противодиабетической, гиполипидемической, гипогликемической и гипохолестеринемической активностью, способ ее получения и способы лечения указанных заболеваний |
| RU2007134267 | 2007-09-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20100086981A true KR20100086981A (ko) | 2010-08-02 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| KR1020107004947A Withdrawn KR20100086981A (ko) | 2007-09-14 | 2008-05-22 | 항당뇨 의약 조성물 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US8247407B2 (https=) |
| EP (1) | EP2204173B1 (https=) |
| JP (1) | JP2010539160A (https=) |
| KR (1) | KR20100086981A (https=) |
| CN (1) | CN101801373B (https=) |
| AU (1) | AU2008297608A1 (https=) |
| BR (1) | BRPI0815200A2 (https=) |
| CA (1) | CA2699403A1 (https=) |
| MX (1) | MX2010002754A (https=) |
| RU (1) | RU2361581C2 (https=) |
| WO (1) | WO2009035368A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2361581C2 (ru) | 2007-09-14 | 2009-07-20 | Закрытое Акционерное Общество "Мастерклон" | Фармацевтическая композиция, обладающая противодиабетической, гиполипидемической, гипогликемической и гипохолестеринемической активностью, способ ее получения и способы лечения указанных заболеваний |
| RU2421219C1 (ru) * | 2009-11-19 | 2011-06-20 | Закрытое Акционерное Общество "Мастерклон" | Ингибиторы протеинкиназы с |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US3510491A (en) * | 1967-02-02 | 1970-05-05 | Sterling Drug Inc | 4-(cyclicaminomethyl)-5-hydroxyindole-3-carboxylic acids and esters thereof |
| US4226829A (en) * | 1978-10-04 | 1980-10-07 | Andrew Mike | Renewable vaporizer for air treatment and the like |
| US4889286A (en) * | 1988-09-19 | 1989-12-26 | Donald Spector | Controllable air freshener unit |
| FR2674522B1 (fr) * | 1991-03-26 | 1993-07-16 | Lipha | Nouveaux derives de l'indole, procedes de preparation et medicaments les contenant. |
| DE19753956A1 (de) * | 1997-12-05 | 1999-06-17 | Draeger Sicherheitstech Gmbh | Duftpatrone |
| SE0104334D0 (sv) | 2001-12-19 | 2001-12-19 | Astrazeneca Ab | Therapeutic agents |
| CN100457730C (zh) * | 2002-08-29 | 2009-02-04 | 默克公司 | 具有抗糖尿病活性的吲哚化合物 |
| AR041481A1 (es) | 2002-10-07 | 2005-05-18 | Hoffmann La Roche | Derivados de acido arilpropionico-oxazol y su uso como agonistas de ppar |
| CA2502269C (en) | 2002-10-18 | 2009-12-22 | Merck & Co., Inc. | Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes |
| WO2005102320A1 (fr) | 2004-04-21 | 2005-11-03 | Zakrytoe Aktsionernoe Obschestvo 'masterklon' | Medicament pour traiter des infections virales |
| US20060233538A1 (en) * | 2005-04-14 | 2006-10-19 | Tollens Fernando R | Energized systems and devices for delivering volatile materials |
| WO2007075102A1 (en) | 2005-12-28 | 2007-07-05 | Zakrytoe Aktsionernoe Obschestvo 'masterklon' | Medicinal agent for treating viral infections |
| US20070176015A1 (en) * | 2006-01-30 | 2007-08-02 | The Procter & Gamble Company | System for delivering volatile materials |
| WO2007136302A2 (en) | 2006-05-23 | 2007-11-29 | Alla Chem, Llc | Active substances, pharmaceutical composition and a method for the production and use thereof |
| US8329689B2 (en) | 2006-05-23 | 2012-12-11 | Alexandre Vasilievich Ivachtchenko | Substituted indoles and a method for the production and use thereof |
| WO2008100977A2 (en) * | 2007-02-14 | 2008-08-21 | N.V. Organon | Carbamates therapeutic release agents as amidase inhibitors |
| RU2344817C1 (ru) | 2007-06-19 | 2009-01-27 | Андрей Александрович Иващенко | Замещенные эфиры 5-гидрокси-1н-индол-3-карбоновой кислоты, фармацевтическая композиция, способ их получения и применения |
| RU2361581C2 (ru) | 2007-09-14 | 2009-07-20 | Закрытое Акционерное Общество "Мастерклон" | Фармацевтическая композиция, обладающая противодиабетической, гиполипидемической, гипогликемической и гипохолестеринемической активностью, способ ее получения и способы лечения указанных заболеваний |
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2007
- 2007-09-14 RU RU2007134267/15A patent/RU2361581C2/ru not_active IP Right Cessation
-
2008
- 2008-05-22 AU AU2008297608A patent/AU2008297608A1/en not_active Abandoned
- 2008-05-22 US US12/673,243 patent/US8247407B2/en not_active Expired - Fee Related
- 2008-05-22 WO PCT/RU2008/000320 patent/WO2009035368A1/ru not_active Ceased
- 2008-05-22 MX MX2010002754A patent/MX2010002754A/es active IP Right Grant
- 2008-05-22 EP EP08779173.7A patent/EP2204173B1/en not_active Not-in-force
- 2008-05-22 KR KR1020107004947A patent/KR20100086981A/ko not_active Withdrawn
- 2008-05-22 CN CN2008801068127A patent/CN101801373B/zh not_active Expired - Fee Related
- 2008-05-22 BR BRPI0815200 patent/BRPI0815200A2/pt not_active IP Right Cessation
- 2008-05-22 CA CA2699403A patent/CA2699403A1/en not_active Abandoned
- 2008-05-22 JP JP2010524811A patent/JP2010539160A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP2204173A1 (en) | 2010-07-07 |
| CN101801373A (zh) | 2010-08-11 |
| AU2008297608A1 (en) | 2009-03-19 |
| BRPI0815200A2 (pt) | 2015-03-31 |
| RU2361581C2 (ru) | 2009-07-20 |
| EP2204173A4 (en) | 2010-12-29 |
| JP2010539160A (ja) | 2010-12-16 |
| US8247407B2 (en) | 2012-08-21 |
| CA2699403A1 (en) | 2009-03-19 |
| MX2010002754A (es) | 2010-03-30 |
| CN101801373B (zh) | 2013-03-27 |
| US20100168092A1 (en) | 2010-07-01 |
| EP2204173B1 (en) | 2013-07-03 |
| WO2009035368A1 (en) | 2009-03-19 |
| RU2007134267A (ru) | 2009-03-20 |
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| PC1203 | Withdrawal of no request for examination | ||
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |