KR20080067000A - 폐 고혈압을 치료하기 위한 디아릴 우레아 - Google Patents
폐 고혈압을 치료하기 위한 디아릴 우레아 Download PDFInfo
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- KR20080067000A KR20080067000A KR1020087013800A KR20087013800A KR20080067000A KR 20080067000 A KR20080067000 A KR 20080067000A KR 1020087013800 A KR1020087013800 A KR 1020087013800A KR 20087013800 A KR20087013800 A KR 20087013800A KR 20080067000 A KR20080067000 A KR 20080067000A
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- compound
- pulmonary hypertension
- inhibitor
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05024509.1 | 2005-11-10 | ||
| EP05024509 | 2005-11-10 | ||
| EP05027450.5 | 2005-12-15 | ||
| EP05027450 | 2005-12-15 | ||
| EP06012234.8 | 2006-06-14 | ||
| EP06012234 | 2006-06-14 |
Publications (1)
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| KR20080067000A true KR20080067000A (ko) | 2008-07-17 |
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| KR1020087013800A Withdrawn KR20080067000A (ko) | 2005-11-10 | 2006-10-30 | 폐 고혈압을 치료하기 위한 디아릴 우레아 |
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|---|---|
| US (1) | US20100035888A1 (https=) |
| EP (1) | EP1948170A1 (https=) |
| JP (1) | JP5084736B2 (https=) |
| KR (1) | KR20080067000A (https=) |
| AR (1) | AR057849A1 (https=) |
| AU (1) | AU2006312714A1 (https=) |
| BR (1) | BRPI0618522A2 (https=) |
| CA (1) | CA2628849A1 (https=) |
| CR (1) | CR9953A (https=) |
| EC (1) | ECSP088430A (https=) |
| GT (1) | GT200800058A (https=) |
| IL (1) | IL191178A0 (https=) |
| NO (1) | NO20082498L (https=) |
| PE (1) | PE20070806A1 (https=) |
| SV (1) | SV2009002900A (https=) |
| TW (1) | TW200733961A (https=) |
| UY (1) | UY29903A1 (https=) |
| WO (1) | WO2007054216A1 (https=) |
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| US8124630B2 (en) | 1999-01-13 | 2012-02-28 | Bayer Healthcare Llc | ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors |
| ATE538794T1 (de) * | 1999-01-13 | 2012-01-15 | Bayer Healthcare Llc | Gamma carboxyarylsubstituierte diphenylharnstoffverbindungen als p38 kinasehemmer |
| US7371763B2 (en) * | 2001-04-20 | 2008-05-13 | Bayer Pharmaceuticals Corporation | Inhibition of raf kinase using quinolyl, isoquinolyl or pyridyl ureas |
| US20080108672A1 (en) * | 2002-01-11 | 2008-05-08 | Bernd Riedl | Omega-Carboxyaryl Substituted Diphenyl Ureas As Raf Kinase Inhibitors |
| MXPA04007832A (es) | 2002-02-11 | 2005-09-08 | Bayer Pharmaceuticals Corp | Aril-ureas con actividad inhibitoria de angiogenesis. |
| DE202004021759U1 (de) * | 2003-02-21 | 2010-10-07 | ResMed Ltd., Bella Vista | Nasale Anordnung |
| US7557129B2 (en) * | 2003-02-28 | 2009-07-07 | Bayer Healthcare Llc | Cyanopyridine derivatives useful in the treatment of cancer and other disorders |
| WO2004113274A2 (en) * | 2003-05-20 | 2004-12-29 | Bayer Pharmaceuticals Corporation | Diaryl ureas with kinase inhibiting activity |
| EA010485B1 (ru) | 2003-07-23 | 2008-10-30 | Байер Фамэсьютиклс Копэрейшн | Производное n,n'-дифенилмочевины, фармацевтическая композиция (варианты) и способ лечения и предупреждения заболеваний и состояний с его использованием (варианты) |
| KR101381454B1 (ko) * | 2004-09-29 | 2014-04-04 | 바이엘 인텔렉쳐 프로퍼티 게엠베하 | 열역학적으로 안정한 형태의 ｂａｙ 43-9006 토실레이트 |
| AR062927A1 (es) * | 2006-10-11 | 2008-12-17 | Bayer Healthcare Ag | 4- [4-( [ [ 4- cloro-3-( trifluorometil) fenil) carbamoil] amino] -3- fluorofenoxi) -n- metilpiridin-2- carboxamida monohidratada |
| JP5885012B2 (ja) * | 2007-01-19 | 2016-03-15 | バイエル・ヘルスケア・エルエルシーＢａｙｅｒ ＨｅａｌｔｈＣａｒｅＬＬＣ | Ｋｉｔ阻害剤に対して獲得した抵抗性を有する癌の処置 |
| JP2011525503A (ja) * | 2008-06-25 | 2011-09-22 | バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト | 心不全を処置するためのジアリールウレア |
| CA2796744A1 (en) * | 2010-04-17 | 2011-10-20 | Bayer Healthcare Llc | Synthetic metabolites of fluoro substituted omega-carboxyaryl diphenyl urea for the treatment and prevention of diseases and conditions |
| MA34553B1 (fr) | 2010-10-01 | 2013-09-02 | Bayer Ip Gmbh | Combinaisons contenant du n-(2-arylamino)arylsulfonamide substitué |
| US20140127295A1 (en) * | 2011-03-14 | 2014-05-08 | Cellworks Group, Inc | Compositions, process of preparation of said compositions and method of treating inflammatory diseases |
| US20160317542A1 (en) | 2013-12-09 | 2016-11-03 | Respira Therapeutics, Inc. | Pde5 inhibitor powder formulations and methods relating thereto |
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| MXPA04007832A (es) * | 2002-02-11 | 2005-09-08 | Bayer Pharmaceuticals Corp | Aril-ureas con actividad inhibitoria de angiogenesis. |
| WO2003084543A1 (en) * | 2002-04-10 | 2003-10-16 | Virginia Commonwealth University | Combination of glivec(sti571) with a cyclin-dependent kinase inhibitor, especially flavopiridol in the treatment of cancer |
| WO2004113274A2 (en) * | 2003-05-20 | 2004-12-29 | Bayer Pharmaceuticals Corporation | Diaryl ureas with kinase inhibiting activity |
| EA010485B1 (ru) * | 2003-07-23 | 2008-10-30 | Байер Фамэсьютиклс Копэрейшн | Производное n,n'-дифенилмочевины, фармацевтическая композиция (варианты) и способ лечения и предупреждения заболеваний и состояний с его использованием (варианты) |
| WO2006091542A2 (en) * | 2005-02-22 | 2006-08-31 | Cedars-Sinai Medical Center | Use of sildenafil, vardenafil and other 5-phosphodiesterase inhibitors to enhance permeability of the abnormal blood-brain barrier |
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2006
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- 2006-10-30 EP EP06818314A patent/EP1948170A1/en not_active Withdrawn
- 2006-10-30 KR KR1020087013800A patent/KR20080067000A/ko not_active Withdrawn
- 2006-10-30 JP JP2008539299A patent/JP5084736B2/ja not_active Expired - Fee Related
- 2006-10-30 WO PCT/EP2006/010406 patent/WO2007054216A1/en not_active Ceased
- 2006-10-30 US US12/084,662 patent/US20100035888A1/en not_active Abandoned
- 2006-10-30 AU AU2006312714A patent/AU2006312714A1/en not_active Abandoned
- 2006-10-30 BR BRPI0618522-3A patent/BRPI0618522A2/pt not_active IP Right Cessation
- 2006-10-31 AR ARP060104767A patent/AR057849A1/es not_active Application Discontinuation
- 2006-11-07 UY UY29903A patent/UY29903A1/es not_active Application Discontinuation
- 2006-11-09 TW TW095141431A patent/TW200733961A/zh unknown
- 2006-11-09 PE PE2006001406A patent/PE20070806A1/es not_active Application Discontinuation
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2008
- 2008-05-01 IL IL191178A patent/IL191178A0/en unknown
- 2008-05-06 CR CR9953A patent/CR9953A/es not_active Application Discontinuation
- 2008-05-06 GT GT200800058A patent/GT200800058A/es unknown
- 2008-05-06 SV SV2008002900A patent/SV2009002900A/es not_active Application Discontinuation
- 2008-05-07 EC EC2008008430A patent/ECSP088430A/es unknown
- 2008-06-04 NO NO20082498A patent/NO20082498L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| GT200800058A (es) | 2010-02-23 |
| JP5084736B2 (ja) | 2012-11-28 |
| CR9953A (es) | 2008-10-08 |
| UY29903A1 (es) | 2007-06-29 |
| AU2006312714A1 (en) | 2007-05-18 |
| AR057849A1 (es) | 2007-12-19 |
| US20100035888A1 (en) | 2010-02-11 |
| NO20082498L (no) | 2008-08-07 |
| SV2009002900A (es) | 2009-04-28 |
| IL191178A0 (en) | 2009-08-03 |
| JP2009514910A (ja) | 2009-04-09 |
| ECSP088430A (es) | 2008-07-30 |
| CA2628849A1 (en) | 2007-05-18 |
| BRPI0618522A2 (pt) | 2011-09-06 |
| TW200733961A (en) | 2007-09-16 |
| WO2007054216A1 (en) | 2007-05-18 |
| PE20070806A1 (es) | 2007-09-29 |
| EP1948170A1 (en) | 2008-07-30 |
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