KR20070112775A - 선택적인 안드로겐 수용체 조절자로서의 아미노페닐 유도체 - Google Patents
선택적인 안드로겐 수용체 조절자로서의 아미노페닐 유도체 Download PDFInfo
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- KR20070112775A KR20070112775A KR1020077018305A KR20077018305A KR20070112775A KR 20070112775 A KR20070112775 A KR 20070112775A KR 1020077018305 A KR1020077018305 A KR 1020077018305A KR 20077018305 A KR20077018305 A KR 20077018305A KR 20070112775 A KR20070112775 A KR 20070112775A
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Classifications
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- C07D451/06—Oxygen atoms
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- Ophthalmology & Optometry (AREA)
- Child & Adolescent Psychology (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
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| US64284105P | 2005-01-10 | 2005-01-10 | |
| US60/642,841 | 2005-01-10 |
Publications (1)
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| KR20070112775A true KR20070112775A (ko) | 2007-11-27 |
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Family Applications (1)
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| US (2) | US7585877B2 (https=) |
| EP (1) | EP1836202B1 (https=) |
| JP (1) | JP5203712B2 (https=) |
| KR (1) | KR20070112775A (https=) |
| CN (1) | CN101119993B (https=) |
| AU (1) | AU2006205066B2 (https=) |
| CA (1) | CA2594340C (https=) |
| MX (1) | MX2007008334A (https=) |
| NZ (1) | NZ555974A (https=) |
| RU (1) | RU2007130558A (https=) |
| WO (1) | WO2006076317A2 (https=) |
| ZA (1) | ZA200705458B (https=) |
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| US20060173037A1 (en) * | 2005-01-10 | 2006-08-03 | Nathalie Schlienger | Aminophenyl derivatives as selective androgen receptor modulators |
| JP5070054B2 (ja) * | 2005-08-01 | 2012-11-07 | 武田薬品工業株式会社 | 環状アミン化合物 |
| PL2018380T3 (pl) | 2006-05-19 | 2012-05-31 | Abbvie Bahamas Ltd | Skondensowane azabicykliczne pochodne alkanowe podstawione bicykloheterocyklem o aktywności wobec OUN |
| JP5241507B2 (ja) | 2006-11-30 | 2013-07-17 | 武田薬品工業株式会社 | 環状アミン化合物 |
| ME01579B (me) | 2007-08-07 | 2014-09-20 | Takeda Pharmaceuticals Co | Derivati pirolidin-2-ona kao modulatori androgenskih receptora |
| CA2716320C (en) | 2008-02-22 | 2014-01-28 | Radius Health, Inc. | Selective androgen receptor modulators |
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| AU2011212813B2 (en) | 2010-02-04 | 2014-10-23 | Radius Health, Inc. | Selective androgen receptor modulators |
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| US8642632B2 (en) | 2010-07-02 | 2014-02-04 | Radius Health, Inc. | Selective androgen receptor modulators |
| US9133182B2 (en) | 2010-09-28 | 2015-09-15 | Radius Health, Inc. | Selective androgen receptor modulators |
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| WO2014149998A1 (en) * | 2013-03-15 | 2014-09-25 | Lin, Qing | Systemic administration of androgen in treating dry eye syndrome |
| ES3055185T3 (en) | 2014-03-28 | 2026-02-10 | Univ Duke | Treatment of an estrogen receptor positive breast cancer using a selective estrogen receptor modulator |
| US9421264B2 (en) | 2014-03-28 | 2016-08-23 | Duke University | Method of treating cancer using selective estrogen receptor modulators |
| CN106103434B (zh) * | 2014-05-29 | 2019-05-10 | 大鹏药品工业株式会社 | 四氢吡啶并嘧啶化合物或其盐 |
| US10441570B2 (en) | 2015-04-21 | 2019-10-15 | University Of Tennessee Research Foundation | Selective androgen receptor degrader (SARD) Ligands and methods of use thereof |
| US10865184B2 (en) | 2015-04-21 | 2020-12-15 | University Of Tennessee Research Foundation | Selective androgen receptor degrader (SARD) ligands and methods of use thereof |
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| US10806720B2 (en) | 2015-04-21 | 2020-10-20 | University Of Tennessee Research Foundation | Selective androgen receptor degrader (SARD) ligands and methods of use thereof |
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| JP7481115B2 (ja) | 2017-01-05 | 2024-05-10 | ラジウス ファーマシューティカルズ，インコーポレイテッド | Ｒａｄ１９０１－２ｈｃｌの多形性形態 |
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| WO2020051344A1 (en) | 2018-09-05 | 2020-03-12 | University Of Tennessee Research Foundation | Selective androgen receptor degrader (sard) ligands and methods of use thereof |
| EP3924328A1 (en) | 2019-02-12 | 2021-12-22 | Radius Pharmaceuticals, Inc. | Processes and compounds |
| CA3138197A1 (en) | 2019-05-14 | 2020-11-19 | Nuvation Bio Inc. | Anti-cancer nuclear hormone receptor-targeting compounds |
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| WO2022212631A1 (en) * | 2021-03-31 | 2022-10-06 | Taiho Pharmaceutical Co., Ltd. | Treatment of patients metastatic castration-resistant prostate cancer with an androgen receptor antagonist |
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| US20060173037A1 (en) * | 2005-01-10 | 2006-08-03 | Nathalie Schlienger | Aminophenyl derivatives as selective androgen receptor modulators |
-
2006
- 2006-01-09 CN CN200680002003.2A patent/CN101119993B/zh not_active Expired - Fee Related
- 2006-01-09 EP EP06733660.2A patent/EP1836202B1/en not_active Expired - Lifetime
- 2006-01-09 WO PCT/US2006/000733 patent/WO2006076317A2/en not_active Ceased
- 2006-01-09 JP JP2007550547A patent/JP5203712B2/ja not_active Expired - Fee Related
- 2006-01-09 CA CA2594340A patent/CA2594340C/en not_active Expired - Fee Related
- 2006-01-09 KR KR1020077018305A patent/KR20070112775A/ko not_active Withdrawn
- 2006-01-09 US US11/329,267 patent/US7585877B2/en not_active Expired - Fee Related
- 2006-01-09 ZA ZA200705458A patent/ZA200705458B/xx unknown
- 2006-01-09 RU RU2007130558/04A patent/RU2007130558A/ru not_active Application Discontinuation
- 2006-01-09 AU AU2006205066A patent/AU2006205066B2/en not_active Ceased
- 2006-01-09 MX MX2007008334A patent/MX2007008334A/es not_active Application Discontinuation
- 2006-01-09 NZ NZ555974A patent/NZ555974A/en not_active IP Right Cessation
-
2009
- 2009-06-30 US US12/495,514 patent/US20090270449A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2594340A1 (en) | 2006-07-20 |
| EP1836202A2 (en) | 2007-09-26 |
| AU2006205066B2 (en) | 2012-05-17 |
| ZA200705458B (en) | 2008-12-31 |
| WO2006076317A3 (en) | 2006-11-23 |
| US20090270449A1 (en) | 2009-10-29 |
| US20060160845A1 (en) | 2006-07-20 |
| MX2007008334A (es) | 2007-09-11 |
| CN101119993B (zh) | 2015-03-04 |
| CA2594340C (en) | 2015-11-10 |
| EP1836202B1 (en) | 2016-12-21 |
| RU2007130558A (ru) | 2009-02-20 |
| JP2008526888A (ja) | 2008-07-24 |
| WO2006076317A2 (en) | 2006-07-20 |
| US7585877B2 (en) | 2009-09-08 |
| JP5203712B2 (ja) | 2013-06-05 |
| AU2006205066A1 (en) | 2006-07-20 |
| CN101119993A (zh) | 2008-02-06 |
| NZ555974A (en) | 2010-11-26 |
| WO2006076317A9 (en) | 2007-09-27 |
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