KR20000029564A - 5HT2c길항제및D2길항제를함유하는약제학적조성물 - Google Patents

5HT2c길항제및D2길항제를함유하는약제학적조성물 Download PDF

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Publication number
KR20000029564A
KR20000029564A KR1019997000622A KR19997000622A KR20000029564A KR 20000029564 A KR20000029564 A KR 20000029564A KR 1019997000622 A KR1019997000622 A KR 1019997000622A KR 19997000622 A KR19997000622 A KR 19997000622A KR 20000029564 A KR20000029564 A KR 20000029564A
Authority
KR
South Korea
Prior art keywords
antagonist
5ht2c
pharmaceutically acceptable
pharmaceutical composition
compound
Prior art date
Application number
KR1019997000622A
Other languages
English (en)
Korean (ko)
Inventor
토마스 폴 블랙번
Original Assignee
피터 기딩스
스미스클라인비이참피이엘시이
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 피터 기딩스, 스미스클라인비이참피이엘시이 filed Critical 피터 기딩스
Publication of KR20000029564A publication Critical patent/KR20000029564A/ko

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1019997000622A 1996-07-26 1997-07-22 5HT2c길항제및D2길항제를함유하는약제학적조성물 KR20000029564A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9615767.2A GB9615767D0 (en) 1996-07-26 1996-07-26 Novel treatment
GB9615767.2 1996-07-26

Publications (1)

Publication Number Publication Date
KR20000029564A true KR20000029564A (ko) 2000-05-25

Family

ID=10797573

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019997000622A KR20000029564A (ko) 1996-07-26 1997-07-22 5HT2c길항제및D2길항제를함유하는약제학적조성물

Country Status (19)

Country Link
EP (1) EP0936924A2 (es)
JP (1) JP2000516924A (es)
KR (1) KR20000029564A (es)
CN (1) CN1230894A (es)
AR (1) AR008083A1 (es)
AU (1) AU725817B2 (es)
BR (1) BR9710568A (es)
CA (1) CA2261813A1 (es)
CO (1) CO5031292A1 (es)
CZ (1) CZ23799A3 (es)
GB (1) GB9615767D0 (es)
HU (1) HUP9903619A3 (es)
IL (1) IL128219A0 (es)
NO (1) NO990322L (es)
NZ (1) NZ333813A (es)
PL (1) PL331426A1 (es)
TR (1) TR199900140T2 (es)
WO (1) WO1998004289A2 (es)
ZA (1) ZA976593B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9612883D0 (en) * 1996-06-20 1996-08-21 Smithkline Beecham Plc Novel compounds
JP2002530341A (ja) 1998-11-23 2002-09-17 セプラコール, インク. デスメチルオランザピン組成物及び方法
JP2002530339A (ja) 1998-11-23 2002-09-17 セプラコール, インク. 2−ヒドロキシメチルオランザピン組成物及び方法
JP2002530340A (ja) * 1998-11-23 2002-09-17 セプラコール, インク. オランザピン−n−オキサイドを含む医薬組成物
EP1165090A2 (en) * 1999-03-18 2002-01-02 Children's Hospital Research Foundation A method of treating bulimia nervosa and related eating disorders by administration of atypical antipsychotic medications
WO2000071106A2 (en) * 1999-05-19 2000-11-30 Astrazeneca Ab Method of treating weight gain
WO2005013969A1 (en) * 2003-07-15 2005-02-17 Janssen Pharmaceutica N.V. Antipsychotic agent with socializing properties

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9500998D0 (sv) * 1995-03-19 1995-03-19 Haakan Wilhelm Wikstroem New sulfone ester analogues of iso-clozapine and related structures: atypical neuroleptics

Also Published As

Publication number Publication date
JP2000516924A (ja) 2000-12-19
PL331426A1 (en) 1999-07-19
AU4297297A (en) 1998-02-20
GB9615767D0 (en) 1996-09-04
CN1230894A (zh) 1999-10-06
AR008083A1 (es) 1999-12-09
HUP9903619A2 (hu) 2000-10-28
HUP9903619A3 (en) 2001-03-28
NZ333813A (en) 2000-07-28
EP0936924A2 (en) 1999-08-25
ZA976593B (en) 1999-01-25
CZ23799A3 (cs) 1999-06-16
CO5031292A1 (es) 2001-04-27
TR199900140T2 (xx) 1999-03-22
NO990322L (no) 1999-03-24
NO990322D0 (no) 1999-01-25
WO1998004289A2 (en) 1998-02-05
AU725817B2 (en) 2000-10-19
IL128219A0 (en) 1999-11-30
CA2261813A1 (en) 1998-02-05
WO1998004289A3 (en) 1998-03-19
BR9710568A (pt) 1999-08-17

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