KR19990077165A - 신규한 치환 이미다졸 화합물 - Google Patents

신규한 치환 이미다졸 화합물 Download PDF

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Publication number
KR19990077165A
KR19990077165A KR1019980705303A KR19980705303A KR19990077165A KR 19990077165 A KR19990077165 A KR 19990077165A KR 1019980705303 A KR1019980705303 A KR 1019980705303A KR 19980705303 A KR19980705303 A KR 19980705303A KR 19990077165 A KR19990077165 A KR 19990077165A
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KR
South Korea
Prior art keywords
alkyl
formula
compound
imidazole
disease
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
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KR1019980705303A
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English (en)
Korean (ko)
Inventor
제리 엘. 아담스
제프리 시. 보엠
Original Assignee
스튜어트 알. 수터, 스티븐 베네티아너, 피터 존 기딩스
스미스클라인 비참 코포레이션
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Application filed by 스튜어트 알. 수터, 스티븐 베네티아너, 피터 존 기딩스, 스미스클라인 비참 코포레이션 filed Critical 스튜어트 알. 수터, 스티븐 베네티아너, 피터 존 기딩스
Publication of KR19990077165A publication Critical patent/KR19990077165A/ko
Ceased legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P31/12—Antivirals
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    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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    • A—HUMAN NECESSITIES
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    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Toxicology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Virology (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
KR1019980705303A 1996-01-11 1997-01-10 신규한 치환 이미다졸 화합물 Ceased KR19990077165A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US990996P 1996-01-11 1996-01-11
US60/009,909 1996-01-11

Publications (1)

Publication Number Publication Date
KR19990077165A true KR19990077165A (ko) 1999-10-25

Family

ID=21740430

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019980705303A Ceased KR19990077165A (ko) 1996-01-11 1997-01-10 신규한 치환 이미다졸 화합물

Country Status (26)

Country Link
US (3) US5716955A (https=)
EP (1) EP0935465B1 (https=)
JP (2) JP2000503303A (https=)
KR (1) KR19990077165A (https=)
CN (1) CN1213307A (https=)
AR (1) AR006307A1 (https=)
AT (1) ATE264105T1 (https=)
AU (1) AU726084C (https=)
BR (1) BR9706934A (https=)
DE (1) DE69728685T2 (https=)
DK (1) DK0935465T3 (https=)
EA (1) EA001430B1 (https=)
ES (1) ES2219750T3 (https=)
HU (1) HUP9900645A3 (https=)
IL (1) IL125282A (https=)
MX (1) MX9805634A (https=)
NO (1) NO316625B1 (https=)
NZ (1) NZ327052A (https=)
OA (1) OA11514A (https=)
PL (1) PL187616B1 (https=)
PT (1) PT935465E (https=)
SK (2) SK92898A3 (https=)
TR (1) TR199801360T2 (https=)
TW (1) TW523512B (https=)
WO (1) WO1997025046A1 (https=)
ZA (1) ZA97175B (https=)

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