KR102346913B1 - 갈렉틴과 관련된 질환의 예방 및 치료를 위한 셀레노갈락토시드 화합물 및 이의 용도 - Google Patents

갈렉틴과 관련된 질환의 예방 및 치료를 위한 셀레노갈락토시드 화합물 및 이의 용도 Download PDF

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KR102346913B1
KR102346913B1 KR1020187028691A KR20187028691A KR102346913B1 KR 102346913 B1 KR102346913 B1 KR 102346913B1 KR 1020187028691 A KR1020187028691 A KR 1020187028691A KR 20187028691 A KR20187028691 A KR 20187028691A KR 102346913 B1 KR102346913 B1 KR 102346913B1
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naphthyl
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샤론 쉐터
엘리제 조머
피터 쥐 트래버
라파엘 니어
조셉 엠 존슨
라이언 조지
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갈랙틴 사이언시즈, 엘엘씨
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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KR1020187028691A 2016-03-04 2017-03-03 갈렉틴과 관련된 질환의 예방 및 치료를 위한 셀레노갈락토시드 화합물 및 이의 용도 Active KR102346913B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662303872P 2016-03-04 2016-03-04
US62/303,872 2016-03-04
PCT/US2017/020658 WO2017152048A1 (en) 2016-03-04 2017-03-03 Selenogalactoside compounds for the prevention and treatment of diseases associated with galectin and the use thereof

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Publication Number Publication Date
KR20180128419A KR20180128419A (ko) 2018-12-03
KR102346913B1 true KR102346913B1 (ko) 2022-01-04

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KR1020187028691A Active KR102346913B1 (ko) 2016-03-04 2017-03-03 갈렉틴과 관련된 질환의 예방 및 치료를 위한 셀레노갈락토시드 화합물 및 이의 용도

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US (2) US20190367552A1 (https=)
EP (1) EP3423461A4 (https=)
JP (1) JP7086008B2 (https=)
KR (1) KR102346913B1 (https=)
CN (1) CN109071585B (https=)
AU (1) AU2017228365B2 (https=)
CA (1) CA3016343C (https=)
IL (2) IL261431B (https=)
MX (1) MX394409B (https=)
WO (1) WO2017152048A1 (https=)
ZA (1) ZA201805900B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3062648A1 (en) * 2017-05-12 2018-11-15 Galectin Sciences, Llc Compounds for the prevention and treatment of diseases and the use thereof
AU2018361991A1 (en) * 2017-10-31 2020-05-14 Galectin Sciences, Llc Selenogalactoside compounds for the treatment of systemic insulin resistance disorders and the use thereof
AU2020214796A1 (en) * 2019-01-30 2021-07-29 Truebinding, Inc. Anti-Gal3 antibodies and uses thereof
CN114206893A (zh) * 2019-08-09 2022-03-18 爱杜西亚药品有限公司 (杂)芳基-甲基-硫代-β-D-吡喃半乳糖苷衍生物
CN113476442A (zh) * 2021-07-28 2021-10-08 上海交通大学医学院附属第九人民医院 化合物gb-0139在治疗心肌梗死后心肌过度纤维化的药物中的应用
JP2025511354A (ja) 2022-04-06 2025-04-15 シャペロン インク． タウロデオキシコール酸又はその薬学的に許容される塩を有効成分として含有する肺線維症の予防又は治療用組成物

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014078655A1 (en) 2012-11-15 2014-05-22 Tufts University Methods, compositions and kits for treating, modulating, or preventing ocular angiogenesis or fibrosis in a subject using a galectin protein inhibitor
WO2015155207A1 (en) 2014-04-08 2015-10-15 Galecto Biotech Ab Galactoside inhibitors for the treatment of alpha-synucleinopthies

Family Cites Families (9)

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Publication number Priority date Publication date Assignee Title
SE0401301D0 (sv) * 2004-05-21 2004-05-21 Forskarpatent I Syd Ab Novel 3-triazolyl-galactoside inhibitors of galectins
CA2668693A1 (en) * 2006-11-15 2008-05-22 David E. Anderson Therapeutic uses of tim-3 modulators
CN102439021B (zh) * 2009-04-28 2015-09-02 格莱克特生物技术公司 半乳凝素的新型半乳糖苷抑制剂
CA2794066C (en) * 2012-10-31 2017-02-28 Neil Henderson Galactoside inhibitor of galectins
ES2869884T3 (es) * 2011-09-16 2021-10-26 Galectin Therapeutics Inc Composiciones de galacto-ramnogalacturonato para el tratamiento de la esteatohepatitis no alcohólica y la enfermedad de hígado graso no alcohólico
AU2012363033B2 (en) * 2011-12-28 2016-06-02 Galectin Therapeutics, Inc. Composition of novel carbohydrate drug for treatment of human diseases
EP2620443A1 (en) * 2012-01-25 2013-07-31 Galecto Biotech AB Novel galactoside inhibitors of galectins
JP2015535233A (ja) * 2012-10-31 2015-12-10 ガレクト・バイオテック・エイビイ ガレクチン−３のガラクトシド阻害剤及び肺線維症のためのその使用
JP2017512205A (ja) * 2014-03-10 2017-05-18 ラ ホヤ ファーマシューティカル カンパニーＬａ Ｊｏｌｌａ Ｐｈａｒｍａｃｅｕｔｉｃａｌ Ｃｏｍｐａｎｙ 腎臓障害を治療するための組成物及び方法

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014078655A1 (en) 2012-11-15 2014-05-22 Tufts University Methods, compositions and kits for treating, modulating, or preventing ocular angiogenesis or fibrosis in a subject using a galectin protein inhibitor
WO2015155207A1 (en) 2014-04-08 2015-10-15 Galecto Biotech Ab Galactoside inhibitors for the treatment of alpha-synucleinopthies

Non-Patent Citations (3)

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A.A.Kumar et al., Carbohydrate Research, Vol.360 (2012) pp.8-18*
B.M.Swarts et al., Adv. Carbohydra. Chem Biochem., Vol.67 (2012) pp.1-113
S.Andre et al., Bioorganic Medicinal Chem. Letters, Vol.25 (2015) pp.931-935*

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Publication number Publication date
MX394409B (es) 2025-03-24
IL281585B (en) 2022-04-01
CN109071585A (zh) 2018-12-21
IL261431A (en) 2018-10-31
US20230127345A1 (en) 2023-04-27
IL261431B (en) 2021-04-29
KR20180128419A (ko) 2018-12-03
CA3016343C (en) 2024-03-26
US20190367552A1 (en) 2019-12-05
ZA201805900B (en) 2019-07-31
JP7086008B2 (ja) 2022-06-17
CA3016343A1 (en) 2017-09-08
JP2019507194A (ja) 2019-03-14
AU2017228365B2 (en) 2021-05-27
MX2018010683A (es) 2019-05-27
AU2017228365A1 (en) 2018-09-27
IL281585A (en) 2021-05-31
BR112018067693A2 (pt) 2019-01-08
EP3423461A1 (en) 2019-01-09
CN109071585B (zh) 2022-08-16
EP3423461A4 (en) 2020-03-25
WO2017152048A1 (en) 2017-09-08

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