KR102006518B1 - 1-알킬-3-플루오로알킬-1h-피라졸-4-카르복실산 클로라이드의 제조 방법 - Google Patents
1-알킬-3-플루오로알킬-1h-피라졸-4-카르복실산 클로라이드의 제조 방법 Download PDFInfo
- Publication number
- KR102006518B1 KR102006518B1 KR1020147031605A KR20147031605A KR102006518B1 KR 102006518 B1 KR102006518 B1 KR 102006518B1 KR 1020147031605 A KR1020147031605 A KR 1020147031605A KR 20147031605 A KR20147031605 A KR 20147031605A KR 102006518 B1 KR102006518 B1 KR 102006518B1
- Authority
- KR
- South Korea
- Prior art keywords
- alkyl
- pyrazole
- formula
- fluoroalkyl
- carbaldehyde
- Prior art date
Links
- AYCXDJXKBPZTTR-UHFFFAOYSA-N CCOC(c1c(C(F)F)[n](C)nc1)=O Chemical compound CCOC(c1c(C(F)F)[n](C)nc1)=O AYCXDJXKBPZTTR-UHFFFAOYSA-N 0.000 description 1
- MRQQMVMIANXDKC-UHFFFAOYSA-N CCOC(c1c[n](C)nc1C(F)F)=O Chemical compound CCOC(c1c[n](C)nc1C(F)F)=O MRQQMVMIANXDKC-UHFFFAOYSA-N 0.000 description 1
- BGABLBBBIZLHQH-UHFFFAOYSA-N CC[O](C(CC(C(F)F)=O)=O)=C Chemical compound CC[O](C(CC(C(F)F)=O)=O)=C BGABLBBBIZLHQH-UHFFFAOYSA-N 0.000 description 1
- RJPCAQUEBXGVIB-MFNQIRJZSA-N CN/C=C(\C(C(F)F)=N)/C(O)=O Chemical compound CN/C=C(\C(C(F)F)=N)/C(O)=O RJPCAQUEBXGVIB-MFNQIRJZSA-N 0.000 description 1
- MZGPCLIDFPCPTI-UHFFFAOYSA-N C[n]1nc(C(F)F)c(C(Cl)=O)c1 Chemical compound C[n]1nc(C(F)F)c(C(Cl)=O)c1 MZGPCLIDFPCPTI-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12167855.1 | 2012-05-14 | ||
| EP12167855 | 2012-05-14 | ||
| PCT/EP2013/059745 WO2013171134A1 (de) | 2012-05-14 | 2013-05-10 | Verfahren zum herstellen von 1-alkyl-3-fluoralkyl-1h-pyrazol-4-carbonsäurechloriden |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20150008400A KR20150008400A (ko) | 2015-01-22 |
| KR102006518B1 true KR102006518B1 (ko) | 2019-08-01 |
Family
ID=48520908
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020147031605A KR102006518B1 (ko) | 2012-05-14 | 2013-05-10 | 1-알킬-3-플루오로알킬-1h-피라졸-4-카르복실산 클로라이드의 제조 방법 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US9145369B2 (es) |
| EP (1) | EP2850066B1 (es) |
| JP (1) | JP6101345B2 (es) |
| KR (1) | KR102006518B1 (es) |
| CN (1) | CN104254523B (es) |
| BR (1) | BR112014028292B1 (es) |
| DK (1) | DK2850066T3 (es) |
| ES (1) | ES2568979T3 (es) |
| IL (1) | IL235490A (es) |
| MX (1) | MX348274B (es) |
| TW (1) | TWI586653B (es) |
| WO (1) | WO2013171134A1 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6462703B2 (ja) * | 2014-01-24 | 2019-01-30 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | １−アルキル−３−ジフルオロメチル−５−フルオロ−１ｈ−ピラゾール−４−カルバルデヒド類及び１−アルキル−３−ジフルオロメチル−５−フルオロ−１ｈ−ピラゾール−４−カルボキシレート類を調製する方法 |
| WO2016202254A1 (zh) * | 2015-06-19 | 2016-12-22 | 浙江永太科技股份有限公司 | 一种用于制备吡唑甲酸衍生物的方法及其中间体 |
| CN104945325B (zh) * | 2015-06-19 | 2017-04-05 | 浙江永太科技股份有限公司 | 一种吡唑甲酸衍生物的制备方法 |
| JP6911143B2 (ja) | 2018-11-07 | 2021-07-28 | 福建永晶科技股▲ふん▼有限公司Ｆｕｊｉａｎ Ｙｏｎｇｊｉｎｇ Ｔｅｃｈｎｏｌｏｇｙ Ｃｏ．， Ｌｔｄ | ピラゾール又はピリミジノンの新しい製造方法 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1993011117A1 (en) | 1991-12-06 | 1993-06-10 | Monsanto Company | Pyrazole carboxanilide fungicides |
| WO2004063165A1 (en) | 2003-01-06 | 2004-07-29 | Eli Lilly And Company | A pyrazole derivative as ppar modulator |
| EP2325173A1 (de) | 2009-11-19 | 2011-05-25 | Bayer CropScience AG | Verfahren zum Herstellen von 5-Fluor-1-alkyl-3-fluoralkyl-1H-pyrazol-4-carbonsäurechloriden |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GEP20094751B (en) | 2004-08-18 | 2009-08-10 | Pfizer | Inhibitors of hepatitis c virus rna-dependent rna polymerase, and compositions and treatments using the same |
| EA201000345A1 (ru) * | 2005-09-16 | 2010-06-30 | Синджента Партисипейшнс Аг | Способ получения амидов |
| AR056882A1 (es) | 2006-02-01 | 2007-10-31 | Bayer Cropscience Sa | Derivados del fungicida n- cicloalquil- bencil- amida |
| AR061791A1 (es) | 2006-06-30 | 2008-09-24 | Basf Ag | Compuestos de 1-(azolin-2-il)-amino-2-aril-1-heteroaril-etano sustituidos, composicion agricola y metodo para proteger plantas de cosecha |
| DE102007002674A1 (de) * | 2007-01-18 | 2008-07-24 | Bayer Cropscience Ag | Verfahren zum Herstellen von substituierten Pyrazolcarbonsäurechloriden |
| EP2008996A1 (en) | 2007-06-27 | 2008-12-31 | Syngeta Participations AG | Process for the production of pyrazoles |
| JP2010531829A (ja) | 2007-07-02 | 2010-09-30 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | 新規殺微生物剤 |
| JP5500582B2 (ja) * | 2009-02-09 | 2014-05-21 | 公益財団法人相模中央化学研究所 | ピラゾ−ル−４−カルボキサミド誘導体、それらの製造方法及びそれらを有効成分とする殺菌剤 |
| EP2595962B1 (en) | 2010-07-23 | 2018-07-11 | Solvay Sa | Process for the preparation of esters of 1-substituted-3-fluoroalkyl-pyrazole-4-carboxylic acids |
-
2013
- 2013-05-10 WO PCT/EP2013/059745 patent/WO2013171134A1/de active Application Filing
- 2013-05-10 MX MX2014013812A patent/MX348274B/es active IP Right Grant
- 2013-05-10 KR KR1020147031605A patent/KR102006518B1/ko active IP Right Grant
- 2013-05-10 CN CN201380022186.4A patent/CN104254523B/zh active Active
- 2013-05-10 EP EP13725092.4A patent/EP2850066B1/de active Active
- 2013-05-10 BR BR112014028292-7A patent/BR112014028292B1/pt active IP Right Grant
- 2013-05-10 JP JP2015512006A patent/JP6101345B2/ja active Active
- 2013-05-10 DK DK13725092.4T patent/DK2850066T3/en active
- 2013-05-10 ES ES13725092.4T patent/ES2568979T3/es active Active
- 2013-05-10 US US14/400,359 patent/US9145369B2/en active Active
- 2013-05-13 TW TW102116823A patent/TWI586653B/zh active
-
2014
- 2014-11-04 IL IL235490A patent/IL235490A/en active IP Right Grant
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1993011117A1 (en) | 1991-12-06 | 1993-06-10 | Monsanto Company | Pyrazole carboxanilide fungicides |
| WO2004063165A1 (en) | 2003-01-06 | 2004-07-29 | Eli Lilly And Company | A pyrazole derivative as ppar modulator |
| EP2325173A1 (de) | 2009-11-19 | 2011-05-25 | Bayer CropScience AG | Verfahren zum Herstellen von 5-Fluor-1-alkyl-3-fluoralkyl-1H-pyrazol-4-carbonsäurechloriden |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2850066B1 (de) | 2016-03-16 |
| MX2014013812A (es) | 2015-02-04 |
| EP2850066A1 (de) | 2015-03-25 |
| BR112014028292A2 (pt) | 2020-10-27 |
| US20150126748A1 (en) | 2015-05-07 |
| WO2013171134A1 (de) | 2013-11-21 |
| US9145369B2 (en) | 2015-09-29 |
| MX348274B (es) | 2017-06-02 |
| CN104254523A (zh) | 2014-12-31 |
| JP2015517509A (ja) | 2015-06-22 |
| ES2568979T3 (es) | 2016-05-05 |
| KR20150008400A (ko) | 2015-01-22 |
| BR112014028292B1 (pt) | 2021-07-20 |
| JP6101345B2 (ja) | 2017-03-22 |
| IL235490A (en) | 2016-07-31 |
| TW201400461A (zh) | 2014-01-01 |
| TWI586653B (zh) | 2017-06-11 |
| DK2850066T3 (en) | 2016-04-25 |
| CN104254523B (zh) | 2017-03-22 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP5802213B2 (ja) | ５−フッ素−１−アルキル−３−フルオロアルキル−１ｈ−ピラゾール−４−カルボン酸クロライドの製造方法 | |
| KR102006518B1 (ko) | 1-알킬-3-플루오로알킬-1h-피라졸-4-카르복실산 클로라이드의 제조 방법 | |
| JP2007326784A (ja) | １−置換−５−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法 | |
| JP6771475B2 (ja) | ３−クロロ−２−ビニルフェニルスルホネート類の製造方法 | |
| KR20060094534A (ko) | 플루오로메틸-치환된 헤테로사이클의 제조방법 | |
| WO2010122794A1 (ja) | ピラジンカルボン酸誘導体の製造方法及びその中間体 | |
| CN111825653A (zh) | 取代吡唑类化合物的制备及其作为邻氨基苯甲酰胺前体的用途 | |
| WO2010122793A1 (ja) | ピラジン誘導体の製造方法及びその中間体 | |
| JP5631741B2 (ja) | ピラジン誘導体類の製造方法及びその中間体類 | |
| TW202321195A (zh) | (2,2,2-三氟乙基)硫烷基苯胺衍生物的製備方法 | |
| JP5790195B2 (ja) | ピラゾール化合物の製造方法 | |
| JP2013006776A (ja) | ピラゾール化合物の製造方法 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A201 | Request for examination | ||
| E701 | Decision to grant or registration of patent right |