KR101783471B1 - 치환된 1,3-디하이드로-2ｈ-인돌-2-온의 제조방법 - Google Patents

치환된 1,3-디하이드로-2ｈ-인돌-2-온의 제조방법 Download PDF

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Publication number
KR101783471B1
KR101783471B1 KR1020127031887A KR20127031887A KR101783471B1 KR 101783471 B1 KR101783471 B1 KR 101783471B1 KR 1020127031887 A KR1020127031887 A KR 1020127031887A KR 20127031887 A KR20127031887 A KR 20127031887A KR 101783471 B1 KR101783471 B1 KR 101783471B1
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KR
South Korea
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substituted
group
alkyl
formula
unsubstituted
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English (en)
Korean (ko)
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KR20130100913A (ko
Inventor
콘라드 시겔
군터 카리히
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바이엘 인텔렉쳐 프로퍼티 게엠베하
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Assigned to 바이엘 크롭사이언스 악티엔게젤샤프트 reassignment 바이엘 크롭사이언스 악티엔게젤샤프트 권리의 전부이전등록 Assignors: 바이엘 인텔렉쳐 프로퍼티 게엠베하
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C07D209/34—Oxygen atoms in position 2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
    • A01N43/38—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings condensed with carbocyclic rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
KR1020127031887A 2010-05-10 2011-05-06 치환된 1,3-디하이드로-2ｈ-인돌-2-온의 제조방법 Active KR101783471B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US33294910P 2010-05-10 2010-05-10
EP10162381 2010-05-10
US61/332,949 2010-05-10
EP10162381.7 2010-05-10
PCT/EP2011/057276 WO2011141364A1 (de) 2010-05-10 2011-05-06 Verfahren zur herstellung von substituierten 1,3-dihydro-2h-indol-2-onen

Publications (2)

Publication Number Publication Date
KR20130100913A KR20130100913A (ko) 2013-09-12
KR101783471B1 true KR101783471B1 (ko) 2017-09-29

Family

ID=42537445

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020127031887A Active KR101783471B1 (ko) 2010-05-10 2011-05-06 치환된 1,3-디하이드로-2ｈ-인돌-2-온의 제조방법

Country Status (12)

Country Link
US (1) US8563749B2 (cg-RX-API-DMAC10.html)
EP (1) EP2569283B1 (cg-RX-API-DMAC10.html)
JP (1) JP5815679B2 (cg-RX-API-DMAC10.html)
KR (1) KR101783471B1 (cg-RX-API-DMAC10.html)
CN (1) CN102985406B (cg-RX-API-DMAC10.html)
BR (1) BR112012028767B1 (cg-RX-API-DMAC10.html)
DK (1) DK2569283T3 (cg-RX-API-DMAC10.html)
ES (1) ES2523226T3 (cg-RX-API-DMAC10.html)
IL (1) IL222929A (cg-RX-API-DMAC10.html)
MX (1) MX2012012959A (cg-RX-API-DMAC10.html)
TW (1) TWI499583B (cg-RX-API-DMAC10.html)
WO (1) WO2011141364A1 (cg-RX-API-DMAC10.html)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3643210A1 (de) 2018-10-25 2020-04-29 Jura Elektroapparate AG Verfahren zum erzeugen eines kaffeegetränks in einem kaffeeautomaten

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4160032A (en) 1973-11-21 1979-07-03 Sandoz, Inc. Oxindoles as sleep-inducers
US4503073A (en) 1981-01-07 1985-03-05 A. H. Robins Company, Incorporated 2-Amino-3-(alkylthiobenzoyl)-phenylacetic acids
FI80270C (fi) * 1984-09-19 1990-05-10 Pfizer Foerfarande foer framstaellning av analgetiska och anti-inflammatoriska 1,3-diacyl-2-oxoindol-foereningar och mellanprodukter.
US5076835A (en) * 1990-05-31 1991-12-31 America Cyanamid Company Aryloxyspiroalkylindolinone herbicides
US5124347A (en) * 1991-07-31 1992-06-23 Warner-Lambert Co. 3-5-ditertiarybutylphenyl-4-hydroxymethylidene derivatives of 1,3-dihydro-2H-indole-2-ones as antiinflammatory agents
FR2708605A1 (fr) * 1993-07-30 1995-02-10 Sanofi Sa Dérivés du N-sulfonylindol-2-one, leur préparation, les compositions pharmaceutiques en contenant.

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Antiinflammatory agents. 2. Syntheses and antiinflammatory activity of substituted 2-aminophenylacetic acid derivatives. J.MED.CHEM.,1982.
Non-reductive Desulfenylation of 3-Thioalkyl-2-oxindoles. SYNLETT,1996.

Also Published As

Publication number Publication date
TWI499583B (zh) 2015-09-11
EP2569283B1 (de) 2014-08-27
IL222929A (en) 2015-06-30
MX2012012959A (es) 2012-12-17
DK2569283T3 (en) 2014-12-01
JP2013526498A (ja) 2013-06-24
WO2011141364A1 (de) 2011-11-17
ES2523226T3 (es) 2014-11-24
TW201206884A (en) 2012-02-16
JP5815679B2 (ja) 2015-11-17
BR112012028767A2 (pt) 2015-09-15
US8563749B2 (en) 2013-10-22
BR112012028767B1 (pt) 2021-04-27
CN102985406A (zh) 2013-03-20
KR20130100913A (ko) 2013-09-12
CN102985406B (zh) 2015-04-29
IL222929A0 (en) 2012-12-31
EP2569283A1 (de) 2013-03-20
US20110275832A1 (en) 2011-11-10

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