KR101726893B1 - 멜라노코르틴 수용체-특이적 펩티드 - Google Patents

멜라노코르틴 수용체-특이적 펩티드 Download PDF

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KR101726893B1
KR101726893B1 KR1020127000543A KR20127000543A KR101726893B1 KR 101726893 B1 KR101726893 B1 KR 101726893B1 KR 1020127000543 A KR1020127000543 A KR 1020127000543A KR 20127000543 A KR20127000543 A KR 20127000543A KR 101726893 B1 KR101726893 B1 KR 101726893B1
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peptides
peptide
shock
artificial sequence
ser
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KR20120092089A (ko
Inventor
이-쿤 시
슈브 디. 살마
존 에이치. 도드
웨이 양
신 첸
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팔라틴 테크놀로지스 인코포레이티드
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A61K33/16—Fluorine compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/68—Melanocyte-stimulating hormone [MSH]
    • C07K14/685—Alpha-melanotropin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64—Cyclic peptides containing only normal peptide links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Inorganic Chemistry (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
KR1020127000543A 2009-06-08 2010-06-07 멜라노코르틴 수용체-특이적 펩티드 Active KR101726893B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18492909P 2009-06-08 2009-06-08
US61/184,929 2009-06-08
PCT/US2010/037589 WO2010144344A2 (en) 2009-06-08 2010-06-07 Melanocortin receptor-specific peptides

Publications (2)

Publication Number Publication Date
KR20120092089A KR20120092089A (ko) 2012-08-20
KR101726893B1 true KR101726893B1 (ko) 2017-04-13

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020127000543A Active KR101726893B1 (ko) 2009-06-08 2010-06-07 멜라노코르틴 수용체-특이적 펩티드

Country Status (14)

Country Link
US (4) US8846601B2 (https=)
EP (1) EP2440227B1 (https=)
JP (1) JP5805632B2 (https=)
KR (1) KR101726893B1 (https=)
CN (2) CN102458436B (https=)
AU (1) AU2010259008C1 (https=)
BR (1) BRPI1009644B1 (https=)
CA (1) CA2761607C (https=)
EA (1) EA020959B1 (https=)
IL (1) IL216843A (https=)
MX (1) MX2011013117A (https=)
NZ (1) NZ596617A (https=)
WO (1) WO2010144344A2 (https=)
ZA (1) ZA201200112B (https=)

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CA3166448A1 (en) * 2020-02-03 2021-08-12 Wei Yang Reverse amide-linked melanocortin receptor-specific cyclic peptides
CN114890958B (zh) * 2022-02-23 2023-10-20 四川警察学院 双光子染料化合物、其制备方法及其应用
CN115521356B (zh) * 2022-08-17 2024-04-02 桂林医学院 一种具有美白功效的多肽及其应用
CN119529031B (zh) * 2024-11-27 2025-12-05 润辉生物技术（威海）有限公司 一种环肽衍生物及其制备方法与应用

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Publication number Publication date
US8846601B2 (en) 2014-09-30
US20120178701A1 (en) 2012-07-12
US10179804B2 (en) 2019-01-15
CN105037502A (zh) 2015-11-11
CN102458436A (zh) 2012-05-16
US20160318977A1 (en) 2016-11-03
CA2761607A1 (en) 2010-12-16
US20190216887A1 (en) 2019-07-18
AU2010259008A1 (en) 2011-11-24
AU2010259008B2 (en) 2014-12-04
US9458201B2 (en) 2016-10-04
WO2010144344A2 (en) 2010-12-16
AU2010259008C1 (en) 2016-04-21
EA201190338A1 (ru) 2012-06-29
EP2440227A4 (en) 2013-03-20
US10632171B2 (en) 2020-04-28
CA2761607C (en) 2018-09-04
EA020959B1 (ru) 2015-03-31
ZA201200112B (en) 2013-06-26
EP2440227B1 (en) 2017-10-18
MX2011013117A (es) 2012-05-23
IL216843A0 (en) 2012-02-29
US20140357575A1 (en) 2014-12-04
JP5805632B2 (ja) 2015-11-04
CN102458436B (zh) 2015-06-03
EP2440227A2 (en) 2012-04-18
BRPI1009644A2 (pt) 2020-06-23
BRPI1009644B1 (pt) 2022-02-08
WO2010144344A3 (en) 2011-02-03
KR20120092089A (ko) 2012-08-20
JP2012529433A (ja) 2012-11-22
IL216843A (en) 2016-11-30
NZ596617A (en) 2014-04-30

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