KR101716011B1 - Btk 활성의 억제제인 알킬화된 피페라진 화합물 - Google Patents

Btk 활성의 억제제인 알킬화된 피페라진 화합물 Download PDF

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KR101716011B1
KR101716011B1 KR1020147014782A KR20147014782A KR101716011B1 KR 101716011 B1 KR101716011 B1 KR 101716011B1 KR 1020147014782 A KR1020147014782 A KR 1020147014782A KR 20147014782 A KR20147014782 A KR 20147014782A KR 101716011 B1 KR101716011 B1 KR 101716011B1
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mmol
fluoro
methyl
phenyl
pyridin
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KR20140090227A (ko
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제임스 존 크로포드
웬디 비 영
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에프. 호프만-라 로슈 아게
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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KR1020147014782A 2011-11-03 2012-11-02 Btk 활성의 억제제인 알킬화된 피페라진 화합물 Expired - Fee Related KR101716011B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161555395P 2011-11-03 2011-11-03
US61/555,395 2011-11-03
PCT/US2012/063198 WO2013067277A1 (en) 2011-11-03 2012-11-02 Alkylated piperazine compounds as inhibitors of btk activity

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Publication Number Publication Date
KR20140090227A KR20140090227A (ko) 2014-07-16
KR101716011B1 true KR101716011B1 (ko) 2017-03-13

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US (3) US8729072B2 (enExample)
EP (1) EP2773639B1 (enExample)
JP (2) JP5976828B2 (enExample)
KR (1) KR101716011B1 (enExample)
CN (1) CN104024255B (enExample)
AR (1) AR088642A1 (enExample)
AU (1) AU2012332368A1 (enExample)
BR (1) BR112014010439A2 (enExample)
CA (1) CA2853970A1 (enExample)
CL (1) CL2014001158A1 (enExample)
CO (1) CO6950475A2 (enExample)
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EA (1) EA027561B1 (enExample)
IL (1) IL232280A0 (enExample)
IN (1) IN2014CN03265A (enExample)
MA (1) MA35725B1 (enExample)
MX (1) MX2014005289A (enExample)
PE (1) PE20141686A1 (enExample)
PH (1) PH12014500966A1 (enExample)
SG (1) SG11201401993RA (enExample)
TW (1) TW201326171A (enExample)
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RU2016101548A (ru) 2013-07-03 2017-08-08 Ф. Хоффманн-Ля Рош Аг Соединения амидов гетероарилпиридона и азапиридона
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