KR101505419B1 - 나노분산액 - Google Patents

나노분산액 Download PDF

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Publication number
KR101505419B1
KR101505419B1 KR1020107014449A KR20107014449A KR101505419B1 KR 101505419 B1 KR101505419 B1 KR 101505419B1 KR 1020107014449 A KR1020107014449 A KR 1020107014449A KR 20107014449 A KR20107014449 A KR 20107014449A KR 101505419 B1 KR101505419 B1 KR 101505419B1
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KR
South Korea
Prior art keywords
nanodispersion
present
paclitaxel
water
drug
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Expired - Fee Related
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KR1020107014449A
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English (en)
Korean (ko)
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KR20100112564A (ko
Inventor
아제이 제이싱 코파데
서브하스 발라람 보우믹
엔. 아룰수다르
Original Assignee
썬 파마 어드밴스트 리서치 컴패니 리미티드
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40853553&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR101505419(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 썬 파마 어드밴스트 리서치 컴패니 리미티드 filed Critical 썬 파마 어드밴스트 리서치 컴패니 리미티드
Publication of KR20100112564A publication Critical patent/KR20100112564A/ko
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Publication of KR101505419B1 publication Critical patent/KR101505419B1/ko
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/51—Nanocapsules; Nanoparticles
    • A61K9/5107—Excipients; Inactive ingredients
    • A61K9/513—Organic macromolecular compounds; Dendrimers
    • A61K9/5138—Organic macromolecular compounds; Dendrimers obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/51—Nanocapsules; Nanoparticles
    • A61K9/5107—Excipients; Inactive ingredients
    • A61K9/513—Organic macromolecular compounds; Dendrimers
    • A61K9/5146—Organic macromolecular compounds; Dendrimers obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyamines, polyanhydrides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nanotechnology (AREA)
  • Physics & Mathematics (AREA)
  • Biomedical Technology (AREA)
  • Optics & Photonics (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Processes Of Treating Macromolecular Substances (AREA)
KR1020107014449A 2007-12-24 2008-12-23 나노분산액 Expired - Fee Related KR101505419B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN2527MU2007 2007-12-24
IN2527/MUM/2007 2007-12-24
PCT/IN2008/000857 WO2009087678A2 (en) 2007-12-24 2008-12-23 Nanodispersion

Publications (2)

Publication Number Publication Date
KR20100112564A KR20100112564A (ko) 2010-10-19
KR101505419B1 true KR101505419B1 (ko) 2015-03-30

Family

ID=40853553

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020107014449A Expired - Fee Related KR101505419B1 (ko) 2007-12-24 2008-12-23 나노분산액

Country Status (20)

Country Link
US (2) US8586062B2 (https=)
EP (2) EP2853264A1 (https=)
JP (2) JP5656643B2 (https=)
KR (1) KR101505419B1 (https=)
CN (1) CN101909614B (https=)
AP (1) AP2895A (https=)
AU (1) AU2008346121B2 (https=)
BR (1) BRPI0821514B8 (https=)
CA (1) CA2710525C (https=)
CO (1) CO6290681A2 (https=)
DK (1) DK2231144T3 (https=)
EA (1) EA016434B1 (https=)
ES (1) ES2509490T3 (https=)
IL (1) IL206584A0 (https=)
MX (1) MX2010007076A (https=)
NZ (1) NZ586343A (https=)
PL (1) PL2231144T3 (https=)
UA (1) UA100543C2 (https=)
WO (1) WO2009087678A2 (https=)
ZA (1) ZA201004450B (https=)

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CN102802624A (zh) * 2009-06-19 2012-11-28 太阳医药高级研发有限公司 药物的纳米分散体以及它的制备方法
CN102038635A (zh) * 2009-10-23 2011-05-04 天津天士力集团有限公司 一种含有pH值调节剂的紫杉烷类药物溶液及其制备方法
KR20110056042A (ko) * 2009-11-20 2011-05-26 주식회사유한양행 종양세포 표적지향을 위한 나노 입자 및 이의 제조방법
EA027666B1 (ru) 2010-05-03 2017-08-31 ТЕИКОКУ ФАРМА ЮСЭй, ИНК. Неводные лекарственные средства в форме проэмульсии на основе таксанов и способы их приготовления и использования
ES2385995B2 (es) * 2011-01-10 2013-05-21 Universidade De Santiago De Compostela Nanocápsulas con cubierta polimérica
CN102078300B (zh) * 2011-01-27 2012-01-11 海南美大制药有限公司 托拉塞米脂质体固体制剂
CN102366409B (zh) * 2011-09-14 2013-03-20 海南灵康制药有限公司 一种尼扎替丁脂质体固体制剂
JO3685B1 (ar) * 2012-10-01 2020-08-27 Teikoku Pharma Usa Inc صيغ التشتيت الجسيمي للتاكسين غير المائي وطرق استخدامها
US10736327B2 (en) 2013-03-14 2020-08-11 Griffith Foods International Inc. Natural fungicide composition
CA2950741C (en) * 2014-05-30 2023-03-28 Oms Investments, Inc. Nano-sized water-based dispersion compositions and methods of making thereof
KR101692314B1 (ko) * 2015-03-27 2017-01-03 주식회사 주빅 지용성 약물의 생분해성 고분자 내 용해 시스템: 스마트 폴리머 시스템
US20160346221A1 (en) 2015-06-01 2016-12-01 Autotelic Llc Phospholipid-coated therapeutic agent nanoparticles and related methods
EP3307242A4 (en) * 2015-06-09 2019-01-23 Sun Pharma Advanced Research Company Limited PICn-01
CN107551390A (zh) * 2017-08-21 2018-01-09 常熟佳禾生物科技有限公司 一种用于治疗乳腺小叶增生的中药文胸贴片及其制备方法
PL3768274T3 (pl) * 2018-03-19 2024-06-17 Epicyt Pharma Ab Kompozycje zawierające połączenie kwasu glikocholowego i kwasu masłowego lub kwasu oleinowego do zastosowania w leczeniu osteoporozy
US11877717B2 (en) 2019-12-17 2024-01-23 Emma Ruccio Method and apparatus for detecting scoliosis
US11423574B2 (en) 2019-12-17 2022-08-23 Emma Ruccio Method and apparatus for detecting scoliosis
PL3928772T3 (pl) * 2020-06-26 2024-10-07 Algiax Pharmaceuticals Gmbh Kompozycja nanocząstkowa
JP7745863B2 (ja) * 2021-04-12 2025-09-30 国立大学法人広島大学 難水溶性物質の可溶化方法および難水溶性物質の可溶化組成物

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Also Published As

Publication number Publication date
US20100297244A1 (en) 2010-11-25
US8586062B2 (en) 2013-11-19
JP2011507946A (ja) 2011-03-10
EP2231144B1 (en) 2014-07-02
CA2710525C (en) 2017-08-22
JP5656643B2 (ja) 2015-01-21
AP2010005314A0 (en) 2010-08-31
MX2010007076A (es) 2010-09-30
EA201070793A1 (ru) 2010-12-30
CN101909614A (zh) 2010-12-08
DK2231144T3 (da) 2014-10-13
KR20100112564A (ko) 2010-10-19
PL2231144T3 (pl) 2014-12-31
AU2008346121B2 (en) 2013-10-10
BRPI0821514A2 (pt) 2016-09-27
JP5937180B2 (ja) 2016-06-22
EA016434B1 (ru) 2012-04-30
US20140030352A1 (en) 2014-01-30
EP2231144A2 (en) 2010-09-29
AU2008346121A1 (en) 2009-07-16
BRPI0821514B1 (pt) 2020-03-10
EP2853264A1 (en) 2015-04-01
BRPI0821514B8 (pt) 2021-05-25
JP2015110565A (ja) 2015-06-18
UA100543C2 (ru) 2013-01-10
ZA201004450B (en) 2011-03-30
CO6290681A2 (es) 2011-06-20
IL206584A0 (en) 2010-12-30
CA2710525A1 (en) 2009-07-16
ES2509490T3 (es) 2014-10-17
EP2231144A4 (en) 2011-01-12
NZ586343A (en) 2012-03-30
WO2009087678A2 (en) 2009-07-16
AP2895A (en) 2014-05-31
WO2009087678A3 (en) 2009-09-11
CN101909614B (zh) 2015-04-15

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