KR101071048B1 - 3-할로-4,5-디히드로-1ｈ-피라졸의 제조 방법 - Google Patents

3-할로-4,5-디히드로-1ｈ-피라졸의 제조 방법 Download PDF

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Publication number
KR101071048B1
KR101071048B1 KR1020057001599A KR20057001599A KR101071048B1 KR 101071048 B1 KR101071048 B1 KR 101071048B1 KR 1020057001599 A KR1020057001599 A KR 1020057001599A KR 20057001599 A KR20057001599 A KR 20057001599A KR 101071048 B1 KR101071048 B1 KR 101071048B1
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KR
South Korea
Prior art keywords
formula
compound
alkyl
compounds
dihydro
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KR1020057001599A
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English (en)
Korean (ko)
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KR20050026043A (ko
Inventor
게리 데이비드 아니스
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이 아이 듀폰 디 네모아 앤드 캄파니
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Publication of KR20050026043A publication Critical patent/KR20050026043A/ko
Application granted granted Critical
Publication of KR101071048B1 publication Critical patent/KR101071048B1/ko
Assigned to 에프엠씨 코포레이션, 에프엠씨 아그로 싱가포르 피티이. 엘티디. reassignment 에프엠씨 코포레이션 권리의 전부이전등록 Assignors: 이 아이 듀폰 디 네모아 앤드 캄파니
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D231/08—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with oxygen or sulfur atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR1020057001599A 2002-07-31 2003-07-29 3-할로-4,5-디히드로-1ｈ-피라졸의 제조 방법 Expired - Lifetime KR101071048B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US40035602P 2002-07-31 2002-07-31
US60/400,356 2002-07-31
US44645103P 2003-02-11 2003-02-11
US60/446,451 2003-02-11

Publications (2)

Publication Number Publication Date
KR20050026043A KR20050026043A (ko) 2005-03-14
KR101071048B1 true KR101071048B1 (ko) 2011-10-06

Family

ID=31191368

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020057001599A Expired - Lifetime KR101071048B1 (ko) 2002-07-31 2003-07-29 3-할로-4,5-디히드로-1ｈ-피라졸의 제조 방법

Country Status (17)

Country Link
US (2) US7335780B2 (https=)
EP (2) EP1537097B1 (https=)
JP (1) JP4633462B2 (https=)
KR (1) KR101071048B1 (https=)
AT (2) ATE506356T1 (https=)
AU (2) AU2003257027B2 (https=)
BR (1) BRPI0313342B1 (https=)
CA (1) CA2494047C (https=)
DE (2) DE60336867D1 (https=)
DK (2) DK1537097T3 (https=)
ES (1) ES2334660T3 (https=)
IL (2) IL201407A (https=)
MX (2) MX338829B (https=)
PL (1) PL216029B1 (https=)
RU (1) RU2326877C2 (https=)
TW (1) TWI343376B (https=)
WO (1) WO2004011453A2 (https=)

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AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
DE60236600D1 (de) * 2001-08-13 2010-07-15 Du Pont Substituierte 1h-dihydropyrazole, ihre herstellung und verwendung
MY142967A (en) 2001-08-13 2011-01-31 Du Pont Method for controlling particular insect pests by applying anthranilamide compounds
EP1423379B1 (en) 2001-08-15 2008-05-28 E.I. du Pont de Nemours and Company Ortho-substituted aryl amides for controlling invertebrate pests
ES2319743T3 (es) 2001-08-16 2009-05-12 E.I. Du Pont De Nemours And Company Antranilamidas sustituidas para controlar plagas de invertebrados.
TWI283164B (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI326283B (en) 2002-07-31 2010-06-21 Du Pont Method for preparing fused oxazinones
WO2004046129A2 (en) * 2002-11-15 2004-06-03 E.I. Du Pont De Nemours And Company Novel anthranilamide insecticides
TWI289708B (en) 2002-12-25 2007-11-11 Qualcomm Mems Technologies Inc Optical interference type color display
SI1599463T1 (sl) 2003-01-28 2013-10-30 E.I. Du Pont De Nemours And Company Ciano antranilamidni insekticidi
TWI367882B (en) * 2003-03-26 2012-07-11 Du Pont Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates
KR20060008336A (ko) * 2003-06-12 2006-01-26 이 아이 듀폰 디 네모아 앤드 캄파니 융합된 옥사지논 제조 방법
US7342705B2 (en) 2004-02-03 2008-03-11 Idc, Llc Spatial light modulator with integrated optical compensation structure
RU2006139953A (ru) * 2004-04-13 2008-05-20 Е.И. Дюпон Де Немур Энд Компани (Us) Антраниламидные инсектициды
US7561323B2 (en) * 2004-09-27 2009-07-14 Idc, Llc Optical films for directing light towards active areas of displays
ES2413442T3 (es) * 2004-11-18 2013-07-16 E. I. Du Pont De Nemours And Company Insecticidas de antranilamida
TWI371449B (en) 2005-03-18 2012-09-01 Du Pont Conversion of 2-pyrazolines to ryrazoles using bromine
AU2006283181A1 (en) * 2005-08-24 2007-03-01 E. I. Du Pont De Nemours And Company Anthranilamides for controlling invertebrate pests
WO2008045200A2 (en) 2006-10-06 2008-04-17 Qualcomm Mems Technologies, Inc. Optical loss structure integrated in an illumination apparatus of a display
WO2008045207A2 (en) 2006-10-06 2008-04-17 Qualcomm Mems Technologies, Inc. Light guide
JP2009001541A (ja) * 2006-12-15 2009-01-08 Ishihara Sangyo Kaisha Ltd 新規ピラゾール化合物を中間体として用いるアントラニルアミド系化合物の製造方法
CN104496901B (zh) * 2006-12-15 2016-05-25 石原产业株式会社 邻氨基苯甲酰胺系化合物的制造方法
JP5507045B2 (ja) * 2006-12-15 2014-05-28 石原産業株式会社 アントラニルアミド系化合物の製造方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
US8068710B2 (en) 2007-12-07 2011-11-29 Qualcomm Mems Technologies, Inc. Decoupled holographic film and diffuser
CN101550130B (zh) * 2008-04-01 2012-11-07 中国中化股份有限公司 一种制备3-卤代-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酰卤的方法
JP5406581B2 (ja) * 2008-04-16 2014-02-05 石原産業株式会社 アントラニルアミド系化合物の製造方法
KR20140006007A (ko) 2011-01-28 2014-01-15 이 아이 듀폰 디 네모아 앤드 캄파니 2-아미노벤즈아미드 유도체의 제조 방법
EP2928471B1 (en) 2012-12-06 2020-10-14 Celgene Quanticel Research, Inc. Histone demethylase inhibitors
WO2020026259A1 (en) * 2018-07-31 2020-02-06 Sumitomo Chemical India Ltd. Ethyl 2-bromo-4-[2-(3-halopyridin-2-yl)-hydrazinyl]-4-oxobutanoate hbr salt, method of preparation and use thereof
EA202191554A1 (ru) 2018-12-03 2021-09-02 Фмк Корпорейшн Способ получения n-фенилпиразол-1-карбоксамидов
WO2021193432A1 (ja) 2020-03-25 2021-09-30 石原産業株式会社 シクラニリプロールの製造中間体の製造方法
CN114057686A (zh) * 2020-08-05 2022-02-18 沈阳中化农药化工研发有限公司 一种溴代吡唑羧酸酯类化合物的制备方法
US20240270726A1 (en) * 2021-06-04 2024-08-15 Pi Industries Ltd. A novel process for the preparation of anthranilic diamides
TW202342443A (zh) * 2022-01-31 2023-11-01 美商富曼西公司 用於製備３－溴－１－（３－氯吡啶－２－基）－４，５－二氫－１ｈ－吡唑－５－甲酸乙酯之方法
TW202409000A (zh) 2022-08-29 2024-03-01 美商富曼西公司 用於製備３－鹵代－４，５－二氫－１ｈ－吡唑之高效新方法

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US3577471A (en) * 1968-02-01 1971-05-04 Gulf Research Development Co Halogen interchange process
GB1410191A (en) * 1972-02-10 1975-10-15 Minnesota Mining & Mfg 3-chloro-1-aryl-2-pyrazolines
US5281571A (en) * 1990-10-18 1994-01-25 Monsanto Company Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles
MY138097A (en) * 2000-03-22 2009-04-30 Du Pont Insecticidal anthranilamides
US6838074B2 (en) * 2001-08-08 2005-01-04 Bristol-Myers Squibb Company Simultaneous imaging of cardiac perfusion and a vitronectin receptor targeted imaging agent
ITMI20011784A1 (it) 2001-08-13 2003-02-13 Atofina Processo per la preparazione di metacrilammide(maa)da acetoncianidrina
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
MY142967A (en) 2001-08-13 2011-01-31 Du Pont Method for controlling particular insect pests by applying anthranilamide compounds
TWI327566B (en) * 2001-08-13 2010-07-21 Du Pont Novel substituted ihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use
TWI283164B (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI326283B (en) 2002-07-31 2010-06-21 Du Pont Method for preparing fused oxazinones

Also Published As

Publication number Publication date
DE60330357D1 (de) 2010-01-14
IL165502A (en) 2010-05-31
EP1537097A2 (en) 2005-06-08
IL165502A0 (en) 2006-01-15
WO2004011453A2 (en) 2004-02-05
PL375409A1 (en) 2005-11-28
PL216029B1 (pl) 2014-02-28
AU2003257027B2 (en) 2010-09-16
WO2004011453A3 (en) 2004-03-18
MXPA05001117A (es) 2005-04-28
US20050215798A1 (en) 2005-09-29
AU2010257241A1 (en) 2011-01-13
US7705160B2 (en) 2010-04-27
IL201407A (en) 2013-01-31
BRPI0313342B1 (pt) 2016-04-19
DE60336867D1 (de) 2011-06-01
AU2010257241B2 (en) 2011-11-10
AU2003257027A1 (en) 2004-02-16
TWI343376B (en) 2011-06-11
EP1537097B1 (en) 2009-12-02
RU2005105325A (ru) 2005-07-20
BR0313342A (pt) 2005-07-12
TW200406383A (en) 2004-05-01
DK2100889T3 (da) 2011-08-08
ES2334660T3 (es) 2010-03-15
RU2326877C2 (ru) 2008-06-20
US20080108821A1 (en) 2008-05-08
JP4633462B2 (ja) 2011-02-16
EP2100889B1 (en) 2011-04-20
EP2100889A1 (en) 2009-09-16
JP2005534685A (ja) 2005-11-17
ATE506356T1 (de) 2011-05-15
KR20050026043A (ko) 2005-03-14
CA2494047A1 (en) 2004-02-05
ATE450523T1 (de) 2009-12-15
DK1537097T3 (da) 2010-04-12
CA2494047C (en) 2011-05-24
MX338829B (es) 2016-05-03
MX277756B (es) 2010-07-30
US7335780B2 (en) 2008-02-26

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