KR100559019B1 - 헤테로사이클릭 인덴 유사체의 제조 방법 - Google Patents

헤테로사이클릭 인덴 유사체의 제조 방법 Download PDF

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Publication number
KR100559019B1
KR100559019B1 KR1020037009790A KR20037009790A KR100559019B1 KR 100559019 B1 KR100559019 B1 KR 100559019B1 KR 1020037009790 A KR1020037009790 A KR 1020037009790A KR 20037009790 A KR20037009790 A KR 20037009790A KR 100559019 B1 KR100559019 B1 KR 100559019B1
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KR
South Korea
Prior art keywords
formula
alkyl
compound
phenyl
benzenesulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1020037009790A
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English (en)
Korean (ko)
Other versions
KR20030077007A (ko
Inventor
스칼론미켈란젤로
자이빅토마스
Original Assignee
에프. 호프만-라 로슈 아게
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by 에프. 호프만-라 로슈 아게 filed Critical 에프. 호프만-라 로슈 아게
Publication of KR20030077007A publication Critical patent/KR20030077007A/ko
Application granted granted Critical
Publication of KR100559019B1 publication Critical patent/KR100559019B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Hydrogenated Pyridines (AREA)
KR1020037009790A 2001-01-25 2002-01-22 헤테로사이클릭 인덴 유사체의 제조 방법 Expired - Fee Related KR100559019B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP01101584.9 2001-01-25
EP01101584 2001-01-25
PCT/EP2002/000583 WO2002059089A2 (en) 2001-01-25 2002-01-22 Process for the preparation of heterocyclic indene analogs

Publications (2)

Publication Number Publication Date
KR20030077007A KR20030077007A (ko) 2003-09-29
KR100559019B1 true KR100559019B1 (ko) 2006-03-10

Family

ID=8176288

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020037009790A Expired - Fee Related KR100559019B1 (ko) 2001-01-25 2002-01-22 헤테로사이클릭 인덴 유사체의 제조 방법

Country Status (9)

Country Link
US (2) US6777559B2 (https=)
EP (1) EP1355880A2 (https=)
JP (1) JP4056883B2 (https=)
KR (1) KR100559019B1 (https=)
CN (1) CN1266131C (https=)
CA (1) CA2434408C (https=)
JO (1) JO2433B1 (https=)
MX (1) MXPA03006606A (https=)
WO (1) WO2002059089A2 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004501191A (ja) * 2000-06-28 2004-01-15 テバ　ファーマシューティカル　インダストリーズ　リミティド カルベジロール
MXPA04006909A (es) 2002-01-15 2005-04-19 Teva Pharma Solidos cristalinos de carvedilol y procesos para su preparacion.
US20070191456A1 (en) * 2004-04-22 2007-08-16 Tarur Venkatasubramanian R Novel process for the preparation of 1-(9h-carbazol-4-yloxy)-3-[[2-(-methoxyphenoxy)-ethyl] amino]-propan-2-ol
GB0411273D0 (en) * 2004-05-20 2004-06-23 Cipla Ltd Process and product
US20070043099A1 (en) * 2005-06-09 2007-02-22 Igor Lifshitz Crystalline forms of carvedilol and processes for their preparation
WO2008002683A2 (en) * 2006-06-28 2008-01-03 Teva Pharmaceutical Industries Ltd. Polymorphous forms of carvedilol phosphate
WO2008038301A1 (en) * 2006-09-26 2008-04-03 Morepen Laboratories Limited A process for the preparation of carvedilol
US20080207726A1 (en) * 2007-02-26 2008-08-28 Santiago Ini Process for the purification of carvedilol or its salts thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2258431T3 (es) 1999-08-02 2006-09-01 F. Hoffmann-La Roche Ag Proceso para la preparacion de derivados de benzotiofeno.

Also Published As

Publication number Publication date
JP2004519465A (ja) 2004-07-02
EP1355880A2 (en) 2003-10-29
CA2434408A1 (en) 2002-08-01
WO2002059089A3 (en) 2002-10-31
JO2433B1 (en) 2008-04-17
MXPA03006606A (es) 2003-09-22
US20040127723A1 (en) 2004-07-01
WO2002059089A2 (en) 2002-08-01
KR20030077007A (ko) 2003-09-29
CN1487922A (zh) 2004-04-07
US7169935B2 (en) 2007-01-30
US20020099223A1 (en) 2002-07-25
JP4056883B2 (ja) 2008-03-05
CN1266131C (zh) 2006-07-26
CA2434408C (en) 2009-10-20
US6777559B2 (en) 2004-08-17

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