KR100462441B1 - 성 호르몬 및 시클로덱스트린을 포함하는 비강 분무액을 제조하는 방법 - Google Patents

성 호르몬 및 시클로덱스트린을 포함하는 비강 분무액을 제조하는 방법 Download PDF

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Publication number
KR100462441B1
KR100462441B1 KR10-2001-7004679A KR20017004679A KR100462441B1 KR 100462441 B1 KR100462441 B1 KR 100462441B1 KR 20017004679 A KR20017004679 A KR 20017004679A KR 100462441 B1 KR100462441 B1 KR 100462441B1
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KR
South Korea
Prior art keywords
solution
cyclodextrin
estradiol
purified water
hormone
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR10-2001-7004679A
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English (en)
Korean (ko)
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KR20010073214A (ko
Inventor
질르 퐁크네끄땅
빠트리끄 우트리끄
Original Assignee
르 라보레또레 쎄르비에르
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Publication of KR20010073214A publication Critical patent/KR20010073214A/ko
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Publication of KR100462441B1 publication Critical patent/KR100462441B1/ko
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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40Cyclodextrins; Derivatives thereof

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Nanotechnology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Biotechnology (AREA)
  • General Engineering & Computer Science (AREA)
  • Medical Informatics (AREA)
  • Molecular Biology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Biophysics (AREA)
  • Reproductive Health (AREA)
  • Otolaryngology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR10-2001-7004679A 1998-10-14 1999-10-13 성 호르몬 및 시클로덱스트린을 포함하는 비강 분무액을 제조하는 방법 Expired - Fee Related KR100462441B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9812836A FR2784584B1 (fr) 1998-10-14 1998-10-14 Procede de preparation d'une solution pour pulverisation nasale contenant une ou plusieurs hormones sexuelles et une cyclodextrine
FR98/12836 1998-10-14

Publications (2)

Publication Number Publication Date
KR20010073214A KR20010073214A (ko) 2001-07-31
KR100462441B1 true KR100462441B1 (ko) 2004-12-17

Family

ID=9531516

Family Applications (1)

Application Number Title Priority Date Filing Date
KR10-2001-7004679A Expired - Fee Related KR100462441B1 (ko) 1998-10-14 1999-10-13 성 호르몬 및 시클로덱스트린을 포함하는 비강 분무액을 제조하는 방법

Country Status (21)

Country Link
EP (1) EP1121100B1 (https=)
JP (1) JP3911125B2 (https=)
KR (1) KR100462441B1 (https=)
CN (1) CN1323198A (https=)
AT (1) ATE237310T1 (https=)
AU (1) AU756441B2 (https=)
BR (1) BR9914532A (https=)
CA (1) CA2346567C (https=)
DE (1) DE69907005T2 (https=)
DK (1) DK1121100T3 (https=)
EA (1) EA003069B1 (https=)
ES (1) ES2197672T3 (https=)
FR (1) FR2784584B1 (https=)
HK (1) HK1040201A1 (https=)
HU (1) HUP0103968A3 (https=)
NO (1) NO20011673D0 (https=)
NZ (1) NZ510776A (https=)
PL (1) PL347322A1 (https=)
PT (1) PT1121100E (https=)
WO (1) WO2000021503A1 (https=)
ZA (1) ZA200102961B (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2827516B1 (fr) * 2001-07-19 2003-09-19 Servier Lab Composition pharmaceutique pour l'administration par voie nasale d'estradiol et de norethisterone
EP1661556A4 (en) * 2003-08-20 2010-05-19 Ajinomoto Kk MEDICAL PREPARATION WITH IMPROVED RESOLUTION CHARACTERISTICS
GB2482868A (en) * 2010-08-16 2012-02-22 Franciscus Wilhelmus Henricus Maria Merkus A testosterone liquid spray formulation for oromucosal administration
EA201490746A3 (ru) * 2011-10-07 2016-09-30 Флорида Стейт Юниверсити Рисеч Фондэйшн Применение прогестерона при профилактике и после острого периода для улучшения исходов, связанных с сотрясением мозга
CA2863500A1 (en) 2012-01-20 2013-07-25 Aratana Therapeutics Nv Eye drop composition
RU2753511C2 (ru) * 2017-05-31 2021-08-17 Аратана Терапьютикс, Инк. Композиция глазных капель

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8801670A (nl) * 1988-07-01 1990-02-01 Walter Adrianus Josephus Johan Farmaceutisch preparaat.
US5376645A (en) * 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
GB9012663D0 (en) * 1990-06-07 1990-08-01 Erba Carlo Spa Galenic formulations containing cyclodextrins
DE4207922A1 (de) * 1992-03-13 1993-09-23 Pharmatech Gmbh Wasserloesliche einschlussverbindungen und verfahren zu deren herstellung
BE1007402A5 (nl) * 1993-03-26 1995-06-06 Adir Nasale farmaceutische preparaten met progestagene stof.

Also Published As

Publication number Publication date
HUP0103968A2 (hu) 2002-04-29
FR2784584A1 (fr) 2000-04-21
BR9914532A (pt) 2001-11-06
ZA200102961B (en) 2001-11-20
EP1121100A1 (fr) 2001-08-08
ATE237310T1 (de) 2003-05-15
JP3911125B2 (ja) 2007-05-09
AU756441B2 (en) 2003-01-16
CA2346567A1 (fr) 2000-04-20
NZ510776A (en) 2002-10-25
KR20010073214A (ko) 2001-07-31
HUP0103968A3 (en) 2002-06-28
JP2002527374A (ja) 2002-08-27
NO20011673L (no) 2001-04-03
DE69907005T2 (de) 2004-03-18
EA003069B1 (ru) 2002-12-26
CN1323198A (zh) 2001-11-21
PT1121100E (pt) 2003-07-31
ES2197672T3 (es) 2004-01-01
DE69907005D1 (de) 2003-05-22
FR2784584B1 (fr) 2002-09-20
EA200100316A1 (ru) 2002-02-28
EP1121100B1 (fr) 2003-04-16
DK1121100T3 (da) 2003-07-21
PL347322A1 (en) 2002-03-25
NO20011673D0 (no) 2001-04-03
HK1040201A1 (zh) 2002-05-31
CA2346567C (fr) 2005-06-14
AU6096799A (en) 2000-05-01
WO2000021503A1 (fr) 2000-04-20

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