KR100203548B1 - 고체상 합성에 의한 펩티드의 제조방법 - Google Patents

고체상 합성에 의한 펩티드의 제조방법 Download PDF

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Publication number
KR100203548B1
KR100203548B1 KR1019910014992A KR910014992A KR100203548B1 KR 100203548 B1 KR100203548 B1 KR 100203548B1 KR 1019910014992 A KR1019910014992 A KR 1019910014992A KR 910014992 A KR910014992 A KR 910014992A KR 100203548 B1 KR100203548 B1 KR 100203548B1
Authority
KR
South Korea
Prior art keywords
formula
resin
cooh
acid
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
KR1019910014992A
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English (en)
Korean (ko)
Other versions
KR920004421A (ko
Inventor
브라이폴 게르하르트
크놀레 요헨
퀘닉 볼프강
Original Assignee
무명씨
훽스트 악티엔게젤샤프트
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Publication date
Application filed by 무명씨, 훽스트 악티엔게젤샤프트 filed Critical 무명씨
Publication of KR920004421A publication Critical patent/KR920004421A/ko
Application granted granted Critical
Publication of KR100203548B1 publication Critical patent/KR100203548B1/ko
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1019910014992A 1990-08-30 1991-08-29 고체상 합성에 의한 펩티드의 제조방법 Expired - Lifetime KR100203548B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4027394 1990-08-30
DEP4027394.6 1990-08-30

Publications (2)

Publication Number Publication Date
KR920004421A KR920004421A (ko) 1992-03-27
KR100203548B1 true KR100203548B1 (ko) 1999-06-15

Family

ID=6413202

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019910014992A Expired - Lifetime KR100203548B1 (ko) 1990-08-30 1991-08-29 고체상 합성에 의한 펩티드의 제조방법

Country Status (22)

Country Link
EP (1) EP0475184B1 (https=)
JP (1) JP3177269B2 (https=)
KR (1) KR100203548B1 (https=)
AU (1) AU646488B2 (https=)
CA (1) CA2050216C (https=)
CZ (1) CZ282881B6 (https=)
DE (1) DE59104538D1 (https=)
DK (1) DK0475184T3 (https=)
ES (1) ES2069148T3 (https=)
FI (1) FI102380B (https=)
GR (1) GR3015359T3 (https=)
HU (1) HU208838B (https=)
IE (1) IE66524B1 (https=)
IL (1) IL99338A (https=)
NO (1) NO300216B1 (https=)
NZ (1) NZ239575A (https=)
PL (1) PL167504B1 (https=)
PT (1) PT98813B (https=)
RU (1) RU2036200C1 (https=)
SK (1) SK280319B6 (https=)
TW (1) TW295589B (https=)
ZA (1) ZA916848B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9112825D0 (en) * 1991-06-14 1991-07-31 Ici Plc Process for making peptides
GB9727123D0 (en) * 1997-12-22 1998-02-25 Int Centre Genetic Eng & Bio Synthesis of diamines
ES2154590B1 (es) 1999-05-20 2001-11-01 Lipotec Sa Procedimiento de sintesis de peptidos en fase solida
MX2007008781A (es) 2005-01-21 2007-09-11 Astex Therapeutics Ltd Compuestos farmaceuticos.
WO2008044041A1 (en) 2006-10-12 2008-04-17 Astex Therapeutics Limited Pharmaceutical combinations
JP5528807B2 (ja) 2006-10-12 2014-06-25 アステックス、セラピューティックス、リミテッド 複合薬剤
CN105189465B (zh) 2013-03-21 2019-02-26 赛诺菲-安万特德国有限公司 合成含有乙内酰脲的肽产物
WO2014147129A1 (en) 2013-03-21 2014-09-25 Sanofi-Aventis Deutschland Gmbh Synthesis of cyclic imide containing peptide products

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0322348B1 (de) * 1987-12-22 1994-02-02 Hoechst Aktiengesellschaft Säurelabile Ankergruppen zur Synthese von Peptidamiden mittels Festphasenmethode

Also Published As

Publication number Publication date
AU646488B2 (en) 1994-02-24
CA2050216A1 (en) 1992-03-01
FI102380B1 (fi) 1998-11-30
AU8340291A (en) 1992-03-05
IE913051A1 (en) 1992-03-11
PL167504B1 (pl) 1995-09-30
SK280319B6 (sk) 1999-11-08
PT98813B (pt) 1999-01-29
NO913396L (no) 1992-03-02
HUT60749A (en) 1992-10-28
DK0475184T3 (da) 1995-06-26
DE59104538D1 (de) 1995-03-23
HU208838B (en) 1994-01-28
CZ282881B6 (cs) 1997-11-12
IL99338A0 (en) 1992-07-15
KR920004421A (ko) 1992-03-27
GR3015359T3 (en) 1995-06-30
HU912825D0 (en) 1992-10-28
CS266691A3 (en) 1992-03-18
PL291561A1 (en) 1992-07-13
IE66524B1 (en) 1996-01-10
FI102380B (fi) 1998-11-30
RU2036200C1 (ru) 1995-05-27
TW295589B (https=) 1997-01-11
NZ239575A (en) 1993-07-27
ZA916848B (en) 1992-04-29
EP0475184A1 (de) 1992-03-18
NO300216B1 (no) 1997-04-28
ES2069148T3 (es) 1995-05-01
IL99338A (en) 1996-05-14
FI914064L (fi) 1992-03-01
CA2050216C (en) 2003-03-11
NO913396D0 (no) 1991-08-29
FI914064A0 (fi) 1991-08-28
JPH04230697A (ja) 1992-08-19
PT98813A (pt) 1992-07-31
JP3177269B2 (ja) 2001-06-18
EP0475184B1 (de) 1995-02-08

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