IE66524B1 - A process for the preparation of peptides by solid-phase synthesis - Google Patents

A process for the preparation of peptides by solid-phase synthesis

Info

Publication number
IE66524B1
IE66524B1 IE305191A IE305191A IE66524B1 IE 66524 B1 IE66524 B1 IE 66524B1 IE 305191 A IE305191 A IE 305191A IE 305191 A IE305191 A IE 305191A IE 66524 B1 IE66524 B1 IE 66524B1
Authority
IE
Ireland
Prior art keywords
labile
acid
formula
protective group
cooh
Prior art date
Application number
IE305191A
Other languages
English (en)
Other versions
IE913051A1 (en
Inventor
Gerhard Breipohl
Jochen Knolle
Wolfgang Koenig
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of IE913051A1 publication Critical patent/IE913051A1/en
Publication of IE66524B1 publication Critical patent/IE66524B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IE305191A 1990-08-30 1991-08-29 A process for the preparation of peptides by solid-phase synthesis IE66524B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4027394 1990-08-30

Publications (2)

Publication Number Publication Date
IE913051A1 IE913051A1 (en) 1992-03-11
IE66524B1 true IE66524B1 (en) 1996-01-10

Family

ID=6413202

Family Applications (1)

Application Number Title Priority Date Filing Date
IE305191A IE66524B1 (en) 1990-08-30 1991-08-29 A process for the preparation of peptides by solid-phase synthesis

Country Status (22)

Country Link
EP (1) EP0475184B1 (https=)
JP (1) JP3177269B2 (https=)
KR (1) KR100203548B1 (https=)
AU (1) AU646488B2 (https=)
CA (1) CA2050216C (https=)
CZ (1) CZ282881B6 (https=)
DE (1) DE59104538D1 (https=)
DK (1) DK0475184T3 (https=)
ES (1) ES2069148T3 (https=)
FI (1) FI102380B (https=)
GR (1) GR3015359T3 (https=)
HU (1) HU208838B (https=)
IE (1) IE66524B1 (https=)
IL (1) IL99338A (https=)
NO (1) NO300216B1 (https=)
NZ (1) NZ239575A (https=)
PL (1) PL167504B1 (https=)
PT (1) PT98813B (https=)
RU (1) RU2036200C1 (https=)
SK (1) SK280319B6 (https=)
TW (1) TW295589B (https=)
ZA (1) ZA916848B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9112825D0 (en) * 1991-06-14 1991-07-31 Ici Plc Process for making peptides
GB9727123D0 (en) * 1997-12-22 1998-02-25 Int Centre Genetic Eng & Bio Synthesis of diamines
ES2154590B1 (es) 1999-05-20 2001-11-01 Lipotec Sa Procedimiento de sintesis de peptidos en fase solida
MX2007008781A (es) 2005-01-21 2007-09-11 Astex Therapeutics Ltd Compuestos farmaceuticos.
WO2008044041A1 (en) 2006-10-12 2008-04-17 Astex Therapeutics Limited Pharmaceutical combinations
JP5528807B2 (ja) 2006-10-12 2014-06-25 アステックス、セラピューティックス、リミテッド 複合薬剤
CN105189465B (zh) 2013-03-21 2019-02-26 赛诺菲-安万特德国有限公司 合成含有乙内酰脲的肽产物
WO2014147129A1 (en) 2013-03-21 2014-09-25 Sanofi-Aventis Deutschland Gmbh Synthesis of cyclic imide containing peptide products

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0322348B1 (de) * 1987-12-22 1994-02-02 Hoechst Aktiengesellschaft Säurelabile Ankergruppen zur Synthese von Peptidamiden mittels Festphasenmethode

Also Published As

Publication number Publication date
AU646488B2 (en) 1994-02-24
CA2050216A1 (en) 1992-03-01
FI102380B1 (fi) 1998-11-30
AU8340291A (en) 1992-03-05
IE913051A1 (en) 1992-03-11
PL167504B1 (pl) 1995-09-30
SK280319B6 (sk) 1999-11-08
PT98813B (pt) 1999-01-29
NO913396L (no) 1992-03-02
HUT60749A (en) 1992-10-28
KR100203548B1 (ko) 1999-06-15
DK0475184T3 (da) 1995-06-26
DE59104538D1 (de) 1995-03-23
HU208838B (en) 1994-01-28
CZ282881B6 (cs) 1997-11-12
IL99338A0 (en) 1992-07-15
KR920004421A (ko) 1992-03-27
GR3015359T3 (en) 1995-06-30
HU912825D0 (en) 1992-10-28
CS266691A3 (en) 1992-03-18
PL291561A1 (en) 1992-07-13
FI102380B (fi) 1998-11-30
RU2036200C1 (ru) 1995-05-27
TW295589B (https=) 1997-01-11
NZ239575A (en) 1993-07-27
ZA916848B (en) 1992-04-29
EP0475184A1 (de) 1992-03-18
NO300216B1 (no) 1997-04-28
ES2069148T3 (es) 1995-05-01
IL99338A (en) 1996-05-14
FI914064L (fi) 1992-03-01
CA2050216C (en) 2003-03-11
NO913396D0 (no) 1991-08-29
FI914064A0 (fi) 1991-08-28
JPH04230697A (ja) 1992-08-19
PT98813A (pt) 1992-07-31
JP3177269B2 (ja) 2001-06-18
EP0475184B1 (de) 1995-02-08

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Legal Events

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MK9A Patent expired