KE2592A - New penicillins, their preparation and their pharmaceutical use - Google Patents
New penicillins, their preparation and their pharmaceutical useInfo
- Publication number
- KE2592A KE2592A KE2592*UA KE259275A KE2592A KE 2592 A KE2592 A KE 2592A KE 259275 A KE259275 A KE 259275A KE 2592 A KE2592 A KE 2592A
- Authority
- KE
- Kenya
- Prior art keywords
- group
- carbon atoms
- formulμ
- compound
- general
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
- C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/30—Oxygen or sulfur atoms
- C07D233/32—One oxygen atom
- C07D233/38—One oxygen atom with acyl radicals or hetero atoms directly attached to ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
- C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
- C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2025414A DE2025414C3 (de) | 1970-05-25 | 1970-05-25 | Cyclische Acylureidophenylacetamidopenicillansäuren |
| DE19712104580 DE2104580C3 (de) | 1971-02-01 | 1971-02-01 | Acylureidopenicilline |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KE2592A true KE2592A (en) | 1976-01-09 |
Family
ID=25759178
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KE2592*UA KE2592A (en) | 1970-05-25 | 1975-12-22 | New penicillins, their preparation and their pharmaceutical use |
Country Status (28)
| Country | Link |
|---|---|
| JP (1) | JPS5538357B1 (no) |
| AR (2) | AR195267A1 (no) |
| AT (1) | AT307617B (no) |
| BE (1) | BE767647A (no) |
| BG (1) | BG23220A3 (no) |
| CA (1) | CA943128A (no) |
| CH (1) | CH562249A5 (no) |
| CS (1) | CS171230B2 (no) |
| CY (1) | CY829A (no) |
| DD (1) | DD91497B3 (no) |
| DK (1) | DK133679C (no) |
| EG (1) | EG10856A (no) |
| ES (4) | ES391532A1 (no) |
| FI (1) | FI54484C (no) |
| FR (1) | FR2100681B1 (no) |
| GB (1) | GB1301961A (no) |
| HU (1) | HU162205B (no) |
| IE (1) | IE35311B1 (no) |
| IL (1) | IL36905A (no) |
| KE (1) | KE2592A (no) |
| LU (1) | LU63203A1 (no) |
| NL (1) | NL172660C (no) |
| NO (1) | NO141164C (no) |
| PH (1) | PH14794A (no) |
| RO (2) | RO59157A (no) |
| SE (1) | SE395896B (no) |
| SU (1) | SU472507A3 (no) |
| YU (1) | YU130271A (no) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2354219A1 (de) * | 1973-10-30 | 1975-05-07 | Bayer Ag | Beta-lactam-antibiotica, ein verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
| US4039673A (en) | 1973-10-30 | 1977-08-02 | Bayer Aktiengesellschaft | Penicillins and cephalosporins and their production |
| GB1486349A (en) * | 1974-11-28 | 1977-09-21 | Bayer Ag | Beta-lactam antibiotics process for their preparation and their use as medicaments |
| DE2658906A1 (de) * | 1976-12-24 | 1978-07-06 | Bayer Ag | Beta-lactam-antibiotika, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
| GB1584400A (en) * | 1976-12-24 | 1981-02-11 | Bayer Ag | (2-oxo-imidazoliden-1-yl(carbonylamino)-acetamido-cephalosporins and penicillins |
| US4229348A (en) * | 1978-05-26 | 1980-10-21 | Chugai Seiyaku Kabushiki Kaisha | Penicillanic acid derivatives |
| JPS5732289A (en) | 1980-08-05 | 1982-02-20 | Chugai Pharmaceut Co Ltd | Alpha-substituted ureidobenzylpenicillin |
-
1971
- 1971-04-23 CH CH599071A patent/CH562249A5/xx not_active IP Right Cessation
- 1971-05-13 BG BG17580A patent/BG23220A3/xx unknown
- 1971-05-19 EG EG209/71A patent/EG10856A/xx active
- 1971-05-19 CS CS3646A patent/CS171230B2/cs unknown
- 1971-05-20 SU SU1661304A patent/SU472507A3/ru active
- 1971-05-21 LU LU63203D patent/LU63203A1/xx unknown
- 1971-05-21 IE IE643/71A patent/IE35311B1/xx unknown
- 1971-05-21 FI FI1401/71A patent/FI54484C/fi active
- 1971-05-24 NO NO1945/71A patent/NO141164C/no unknown
- 1971-05-24 SE SE7106667A patent/SE395896B/xx unknown
- 1971-05-24 DD DD71155301A patent/DD91497B3/de unknown
- 1971-05-24 AR AR235756A patent/AR195267A1/es active
- 1971-05-24 IL IL7136905A patent/IL36905A/xx unknown
- 1971-05-24 DK DK251071A patent/DK133679C/da active
- 1971-05-24 PH PH12493A patent/PH14794A/en unknown
- 1971-05-24 YU YU01302/71A patent/YU130271A/xx unknown
- 1971-05-25 GB GB1688071A patent/GB1301961A/en not_active Expired
- 1971-05-25 RO RO67014A patent/RO59157A/ro unknown
- 1971-05-25 CY CY829A patent/CY829A/xx unknown
- 1971-05-25 CA CA113,784A patent/CA943128A/en not_active Expired
- 1971-05-25 JP JP3524471A patent/JPS5538357B1/ja active Pending
- 1971-05-25 ES ES391532A patent/ES391532A1/es not_active Expired
- 1971-05-25 NL NLAANVRAGE7107175,A patent/NL172660C/xx not_active IP Right Cessation
- 1971-05-25 BE BE767647A patent/BE767647A/xx not_active IP Right Cessation
- 1971-05-25 AT AT450471A patent/AT307617B/de not_active IP Right Cessation
- 1971-05-25 RO RO7100078134A patent/RO62689A/ro unknown
- 1971-05-25 FR FR7118932A patent/FR2100681B1/fr not_active Expired
- 1971-05-25 HU HUBA2591A patent/HU162205B/hu unknown
-
1972
- 1972-05-24 ES ES403124A patent/ES403124A1/es not_active Expired
- 1972-05-24 ES ES403125A patent/ES403125A1/es not_active Expired
- 1972-05-24 ES ES403126A patent/ES403126A1/es not_active Expired
-
1973
- 1973-09-14 AR AR250097A patent/AR195946A1/es active
-
1975
- 1975-12-22 KE KE2592*UA patent/KE2592A/xx unknown
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