JPWO2023085396A5 - - Google Patents
Info
- Publication number
- JPWO2023085396A5 JPWO2023085396A5 JP2023559921A JP2023559921A JPWO2023085396A5 JP WO2023085396 A5 JPWO2023085396 A5 JP WO2023085396A5 JP 2023559921 A JP2023559921 A JP 2023559921A JP 2023559921 A JP2023559921 A JP 2023559921A JP WO2023085396 A5 JPWO2023085396 A5 JP WO2023085396A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- fluoro
- tetrahydropyrimidin
- carboxamido
- indazole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021184646 | 2021-11-12 | ||
| PCT/JP2022/042070 WO2023085396A1 (ja) | 2021-11-12 | 2022-11-11 | アルポート症候群を治療または予防するための医薬組成物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2023085396A1 JPWO2023085396A1 (https=) | 2023-05-19 |
| JPWO2023085396A5 true JPWO2023085396A5 (https=) | 2025-09-17 |
Family
ID=86335840
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023559921A Pending JPWO2023085396A1 (https=) | 2021-11-12 | 2022-11-11 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20250049806A1 (https=) |
| EP (1) | EP4431098A4 (https=) |
| JP (1) | JPWO2023085396A1 (https=) |
| WO (1) | WO2023085396A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4733297A1 (en) * | 2023-06-22 | 2026-04-29 | Antibody Therapeutics, Inc. | Integrin-inhibiting small molecule compound |
| CN118459367B (zh) * | 2024-07-09 | 2024-09-24 | 泰兴市广发金属设备制造厂 | 一种氟乙腈的制备方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL123164A (en) | 1995-08-30 | 2001-03-19 | Searle & Co | Meta-guanidine urea thiourea or azacyclic amino benzoic acid derivatives and pharmaceutical compositions containing them |
| ZA994406B (en) | 1998-03-04 | 2000-02-11 | Searle & Co | Meta-azacyclic amino benzoic acid and derivatives thereof. |
| US6372719B1 (en) | 1998-03-04 | 2002-04-16 | Jay Cunningham | ανβ3 integrin antagonists in combination with chemotherapeutic agents |
| KR20010042614A (ko) | 1998-04-10 | 2001-05-25 | 윌리암스 로저 에이 | 비트로넥틴 길항제로서 복소환식 글리실 베타-알라닌 유도체 |
| HUP0202048A3 (en) * | 1998-05-22 | 2006-11-28 | Boys Town Nat Res Hospital Oma | Use of alpha1betha1 integrin receptor inhibitors and tgf-betha1 inhibitors in the treatment of kidney disease |
| JP2006514050A (ja) * | 2002-12-20 | 2006-04-27 | ファルマシア・コーポレーション | インテグリン受容体アンタゴニスト誘導体としてのβ−アミノ酸化合物のR異性体 |
| WO2014015054A1 (en) | 2012-07-18 | 2014-01-23 | Saint Louis University | Beta amino acid derivatives as integrin antagonists |
| US8716226B2 (en) | 2012-07-18 | 2014-05-06 | Saint Louis University | 3,5 phenyl-substituted beta amino acid derivatives as integrin antagonists |
| SG11201805387RA (en) | 2015-12-30 | 2018-07-30 | Univ Saint Louis | Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists |
| KR20230011967A (ko) * | 2020-05-14 | 2023-01-25 | 유비이 가부시키가이샤 | 1,4,5,6-테트라하이드로피리미딘-2-아민 유도체 |
-
2022
- 2022-11-11 WO PCT/JP2022/042070 patent/WO2023085396A1/ja not_active Ceased
- 2022-11-11 JP JP2023559921A patent/JPWO2023085396A1/ja active Pending
- 2022-11-11 US US18/709,010 patent/US20250049806A1/en active Pending
- 2022-11-11 EP EP22892894.1A patent/EP4431098A4/en active Pending
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JPWO2023085396A5 (https=) | ||
| RU2315041C2 (ru) | Производные 2,6-хинолинила и 2,6-нафтила, фармацевтические композиции на их основе, их применение в качестве ингибиторов vla-4 и промежуточные соединения | |
| JP2012517479A5 (https=) | ||
| JP2021504443A5 (https=) | ||
| CN101622231B (zh) | 作为葡糖激酶激活剂的2,2,2-三取代的乙酰胺衍生物、它们的制造方法和药学应用 | |
| JP5488835B2 (ja) | 置換アセトフェノン化合物、その製造方法及び用途 | |
| CA2558585A1 (en) | Compounds, pharmaceutical compositions and methods for use in treating metabolic disorders | |
| JP2010513272A5 (https=) | ||
| PH12016501057B1 (en) | Pyrrolidinones as herbicides | |
| JP2006518763A5 (https=) | ||
| JP2008505874A5 (https=) | ||
| US9682938B2 (en) | Pyrazolone derivatives as nitroxyl donors | |
| JP2013517273A5 (https=) | ||
| JP2007519692A5 (https=) | ||
| RU2011104223A (ru) | Азотсодержащее ароматическое гетероциклическое соединение | |
| JP2005527625A5 (https=) | ||
| CN1095066A (zh) | 除草剂 | |
| JP2010513397A5 (https=) | ||
| JP4915715B2 (ja) | フェニルピリダジン誘導体及びこれを含有する医薬 | |
| JP2018521119A5 (https=) | ||
| JP2007308471A5 (https=) | ||
| RU2008141509A (ru) | Mglur5 модуляторы 1 | |
| JP2010540462A5 (https=) | ||
| HRP20171991T1 (hr) | Derivati pirolidin karbonske kiseline kao agonisti g-protein spojenog receptora (gpr43), farmaceutski pripravak i postupci za primjenu u liječenju poremećaja metabolizma | |
| RU2003112610A (ru) | Производные пиразола для лечения вирксных заболеваний |