JPWO2021067335A5 - - Google Patents
Download PDFInfo
- Publication number
- JPWO2021067335A5 JPWO2021067335A5 JP2022520290A JP2022520290A JPWO2021067335A5 JP WO2021067335 A5 JPWO2021067335 A5 JP WO2021067335A5 JP 2022520290 A JP2022520290 A JP 2022520290A JP 2022520290 A JP2022520290 A JP 2022520290A JP WO2021067335 A5 JPWO2021067335 A5 JP WO2021067335A5
- Authority
- JP
- Japan
- Prior art keywords
- chemical formula
- pharmaceutically acceptable
- following chemical
- compound
- pharmaceutical composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962909006P | 2019-10-01 | 2019-10-01 | |
US62/909,006 | 2019-10-01 | ||
PCT/US2020/053369 WO2021067335A1 (en) | 2019-10-01 | 2020-09-30 | Benzoxazinone compounds as klk5/7 dual inhibitors |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2022551583A JP2022551583A (ja) | 2022-12-12 |
JPWO2021067335A5 true JPWO2021067335A5 (zh) | 2023-09-29 |
Family
ID=75274622
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2022520290A Pending JP2022551583A (ja) | 2019-10-01 | 2020-09-30 | Klk5/7デュアル阻害剤としてのベンゾキサジノン化合物 |
Country Status (12)
Country | Link |
---|---|
US (2) | US11643420B2 (zh) |
EP (1) | EP4037687A4 (zh) |
JP (1) | JP2022551583A (zh) |
KR (1) | KR20220091488A (zh) |
CN (1) | CN114615984A (zh) |
AU (1) | AU2020359526A1 (zh) |
BR (1) | BR112022005881A2 (zh) |
CA (1) | CA3151626A1 (zh) |
IL (1) | IL291398A (zh) |
MX (1) | MX2022003929A (zh) |
TW (1) | TW202126631A (zh) |
WO (1) | WO2021067335A1 (zh) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20200040103A1 (en) | 2018-03-14 | 2020-02-06 | Genentech, Inc. | Anti-klk5 antibodies and methods of use |
Family Cites Families (34)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3536809A (en) | 1969-02-17 | 1970-10-27 | Alza Corp | Medication method |
US3598123A (en) | 1969-04-01 | 1971-08-10 | Alza Corp | Bandage for administering drugs |
US3845770A (en) | 1972-06-05 | 1974-11-05 | Alza Corp | Osmatic dispensing device for releasing beneficial agent |
US3916899A (en) | 1973-04-25 | 1975-11-04 | Alza Corp | Osmotic dispensing device with maximum and minimum sizes for the passageway |
US4008719A (en) | 1976-02-02 | 1977-02-22 | Alza Corporation | Osmotic system having laminar arrangement for programming delivery of active agent |
ES8702440A1 (es) | 1984-10-04 | 1986-12-16 | Monsanto Co | Un procedimiento para la preparacion de una composicion de polipeptido inyectable sustancialmente no acuosa. |
IE58110B1 (en) | 1984-10-30 | 1993-07-14 | Elan Corp Plc | Controlled release powder and process for its preparation |
CA1309556C (en) | 1987-06-09 | 1992-10-27 | Masayuki Kokubo | 4h-3,1-benzoxazin-4-one compounds and pharmaceutical composition thereoffor the inhibition of serine proteases |
US5073543A (en) | 1988-07-21 | 1991-12-17 | G. D. Searle & Co. | Controlled release formulations of trophic factors in ganglioside-lipsome vehicle |
IT1229203B (it) | 1989-03-22 | 1991-07-25 | Bioresearch Spa | Impiego di acido 5 metiltetraidrofolico, di acido 5 formiltetraidrofolico e dei loro sali farmaceuticamente accettabili per la preparazione di composizioni farmaceutiche in forma a rilascio controllato attive nella terapia dei disturbi mentali organici e composizioni farmaceutiche relative. |
PH30995A (en) | 1989-07-07 | 1997-12-23 | Novartis Inc | Sustained release formulations of water soluble peptides. |
US5120548A (en) | 1989-11-07 | 1992-06-09 | Merck & Co., Inc. | Swelling modulated polymeric drug delivery device |
US5733566A (en) | 1990-05-15 | 1998-03-31 | Alkermes Controlled Therapeutics Inc. Ii | Controlled release of antiparasitic agents in animals |
US5580578A (en) | 1992-01-27 | 1996-12-03 | Euro-Celtique, S.A. | Controlled release formulations coated with aqueous dispersions of acrylic polymers |
TW333456B (en) | 1992-12-07 | 1998-06-11 | Takeda Pharm Ind Co Ltd | A pharmaceutical composition of sustained-release preparation the invention relates to a pharmaceutical composition of sustained-release preparation which comprises a physiologically active peptide. |
US5591767A (en) | 1993-01-25 | 1997-01-07 | Pharmetrix Corporation | Liquid reservoir transdermal patch for the administration of ketorolac |
US6087324A (en) | 1993-06-24 | 2000-07-11 | Takeda Chemical Industries, Ltd. | Sustained-release preparation |
IT1270594B (it) | 1994-07-07 | 1997-05-07 | Recordati Chem Pharm | Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida |
CA2224381A1 (en) | 1995-06-27 | 1997-01-16 | Takeda Chemical Industries, Ltd. | Method of producing sustained-release preparation |
TW448055B (en) | 1995-09-04 | 2001-08-01 | Takeda Chemical Industries Ltd | Method of production of sustained-release preparation |
JP2909418B2 (ja) | 1995-09-18 | 1999-06-23 | 株式会社資生堂 | 薬物の遅延放出型マイクロスフイア |
US5980945A (en) | 1996-01-16 | 1999-11-09 | Societe De Conseils De Recherches Et D'applications Scientifique S.A. | Sustained release drug formulations |
US6264970B1 (en) | 1996-06-26 | 2001-07-24 | Takeda Chemical Industries, Ltd. | Sustained-release preparation |
US6419961B1 (en) | 1996-08-29 | 2002-07-16 | Takeda Chemical Industries, Ltd. | Sustained release microcapsules of a bioactive substance and a biodegradable polymer |
CA2217134A1 (en) | 1996-10-09 | 1998-04-09 | Sumitomo Pharmaceuticals Co., Ltd. | Sustained release formulation |
ATE272394T1 (de) | 1996-10-31 | 2004-08-15 | Takeda Chemical Industries Ltd | Zubereitung mit verzögerter freisetzung |
ZA9711385B (en) | 1996-12-20 | 1999-06-18 | Takeda Chemical Industries Ltd | Method of producing a sustained-release preparation |
US5891474A (en) | 1997-01-29 | 1999-04-06 | Poli Industria Chimica, S.P.A. | Time-specific controlled release dosage formulations and method of preparing same |
US6613358B2 (en) | 1998-03-18 | 2003-09-02 | Theodore W. Randolph | Sustained-release composition including amorphous polymer |
NZ506985A (en) | 1998-03-31 | 2003-10-31 | Warner Lambert Co | Benzoxazinones/benzothiazinones as serine protease inhibitors |
KR19990085365A (ko) | 1998-05-16 | 1999-12-06 | 허영섭 | 지속적으로 약물 조절방출이 가능한 생분해성 고분자 미립구 및그 제조방법 |
US6248363B1 (en) | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
CA2525383C (en) | 2003-06-06 | 2012-03-06 | Arexis Ab | Use of heterocyclic compounds as scce inhibitors |
SI3097085T1 (sl) * | 2014-01-23 | 2020-11-30 | Sixera Pharma Ab | Derivati benzoksazinona za zdravljenje kožnih bolezni |
-
2020
- 2020-09-30 CA CA3151626A patent/CA3151626A1/en active Pending
- 2020-09-30 MX MX2022003929A patent/MX2022003929A/es unknown
- 2020-09-30 AU AU2020359526A patent/AU2020359526A1/en active Pending
- 2020-09-30 US US17/037,910 patent/US11643420B2/en active Active
- 2020-09-30 BR BR112022005881A patent/BR112022005881A2/pt unknown
- 2020-09-30 WO PCT/US2020/053369 patent/WO2021067335A1/en unknown
- 2020-09-30 JP JP2022520290A patent/JP2022551583A/ja active Pending
- 2020-09-30 KR KR1020227014268A patent/KR20220091488A/ko unknown
- 2020-09-30 TW TW109134275A patent/TW202126631A/zh unknown
- 2020-09-30 EP EP20872712.3A patent/EP4037687A4/en active Pending
- 2020-09-30 CN CN202080069819.7A patent/CN114615984A/zh active Pending
-
2022
- 2022-03-15 IL IL291398A patent/IL291398A/en unknown
-
2023
- 2023-04-03 US US18/295,009 patent/US20240067658A1/en active Pending
Similar Documents
Publication | Publication Date | Title |
---|---|---|
RU2606947C2 (ru) | Борсодержащие малые молекулы | |
JP5389668B2 (ja) | 皮膚浸透率の非常に高い1H−イミダゾ[4,5−c]キノリン−4−アミン及び関連化合物の正に荷電した水溶性プロドラッグ | |
TWI689490B (zh) | 用於治療纖維化之經取代之芳族化合物及相關方法 | |
JP2007530523A5 (zh) | ||
JP2001506267A (ja) | アミノステロールエステル化合物 | |
JP2002539243A (ja) | 受精能を向上させるための組成物 | |
JP2015519358A (ja) | スルフォラファンの単離及び精製 | |
JP2001525803A (ja) | 勃起機能不全治療用の薬剤の調製のためのミソプロストール及び/又はミソプロストール酸の用途 | |
JP2003515580A (ja) | (s)−2−エトキシ−3−〔4−(2−[4−メタンスルホニルオキシフェニル]エトキシ)フェニル〕プロパン酸の微粉砕形 | |
JPH0827081A (ja) | L−カルニチン塩および化粧用および皮膚病処置用医薬組成物 | |
JP2562475B2 (ja) | 新規化合物、医療組成物、及び炎症及び痛みの治療方法 | |
JP2003516327A (ja) | アテローム性動脈硬化の予防および/または治療方法 | |
CN108341752A (zh) | 抑制ssao/vap-1的胺类化合物及其在医药上的应用 | |
JPH08109131A (ja) | Hivプロテアーゼ抑制因子組成物 | |
US20230046317A1 (en) | Inhibitors of Glutathione S-Transferases (GSTS) and NAD(P)H:Quinone Oxidoreductase 1 (NQO1), Pharmaceutical Compositions, and Uses in Managing Cancer | |
US20220105082A1 (en) | New formulations containing leukotriene receptor antagonists | |
CN113101289A (zh) | 烟酰胺在制备治疗手足皮肤反应制剂中的应用 | |
US20180085345A1 (en) | Methods of tracking skin conditions using cyclolignan compounds | |
JPWO2021067335A5 (zh) | ||
EP3435990B1 (en) | Stable pharmaceutical compositions for topical administration and uses thereof | |
JPH10513186A (ja) | Hivプロテアーゼ阻害剤インジナビル及び逆転写酵素阻害剤3tcを必要に応じてazt、ddi、又はddcと共に用いるhiv感染の組合せ治療 | |
CN115925640A (zh) | ((3-氨甲酰-5-氟吡嗪-2-基)氧基)甲基异丁酸酯及其制备方法和应用 | |
TW201811307A (zh) | 2-(2-乙氧基-2-氧代乙基)(甲基)胺基-2-氧代乙基5-(十四烷氧基)呋喃-2-羧酸酯之皮膚調配物 | |
JP2003512425A (ja) | 6−メトキシ−2−ナフチル酢酸プロドラッグ | |
RU2004102398A (ru) | Производные бензо[g]хинолина для лечения глаукомы и близорукости |