JPWO2019195080A5 - - Google Patents

Download PDF

Info

Publication number
JPWO2019195080A5
JPWO2019195080A5 JP2020554100A JP2020554100A JPWO2019195080A5 JP WO2019195080 A5 JPWO2019195080 A5 JP WO2019195080A5 JP 2020554100 A JP2020554100 A JP 2020554100A JP 2020554100 A JP2020554100 A JP 2020554100A JP WO2019195080 A5 JPWO2019195080 A5 JP WO2019195080A5
Authority
JP
Japan
Prior art keywords
xrpd pattern
compound
values
crystal
characteristic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020554100A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021520357A5 (https=
JP2021520357A (ja
JP7350007B2 (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/024617 external-priority patent/WO2019195080A1/en
Publication of JP2021520357A publication Critical patent/JP2021520357A/ja
Publication of JP2021520357A5 publication Critical patent/JP2021520357A5/ja
Publication of JPWO2019195080A5 publication Critical patent/JPWO2019195080A5/ja
Priority to JP2023147376A priority Critical patent/JP7663642B2/ja
Application granted granted Critical
Publication of JP7350007B2 publication Critical patent/JP7350007B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020554100A 2018-04-02 2019-03-28 エラミプレチドの合成に有用な結晶性ジペプチド Active JP7350007B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023147376A JP7663642B2 (ja) 2018-04-02 2023-09-12 エラミプレチドの合成に有用な結晶性ジペプチド

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862651430P 2018-04-02 2018-04-02
US62/651,430 2018-04-02
PCT/US2019/024617 WO2019195080A1 (en) 2018-04-02 2019-03-28 Crystalline dipeptides useful in the synthesis of elamipretide

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023147376A Division JP7663642B2 (ja) 2018-04-02 2023-09-12 エラミプレチドの合成に有用な結晶性ジペプチド

Publications (4)

Publication Number Publication Date
JP2021520357A JP2021520357A (ja) 2021-08-19
JP2021520357A5 JP2021520357A5 (https=) 2022-03-30
JPWO2019195080A5 true JPWO2019195080A5 (https=) 2022-03-30
JP7350007B2 JP7350007B2 (ja) 2023-09-25

Family

ID=68101313

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020554100A Active JP7350007B2 (ja) 2018-04-02 2019-03-28 エラミプレチドの合成に有用な結晶性ジペプチド
JP2023147376A Active JP7663642B2 (ja) 2018-04-02 2023-09-12 エラミプレチドの合成に有用な結晶性ジペプチド

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023147376A Active JP7663642B2 (ja) 2018-04-02 2023-09-12 エラミプレチドの合成に有用な結晶性ジペプチド

Country Status (13)

Country Link
US (4) US10975118B2 (https=)
EP (2) EP3774844B1 (https=)
JP (2) JP7350007B2 (https=)
KR (2) KR102753323B1 (https=)
CN (2) CN112292388B (https=)
AU (1) AU2019249121B2 (https=)
CA (2) CA3280578A1 (https=)
DK (1) DK3774844T3 (https=)
ES (1) ES2941266T3 (https=)
FI (1) FI3774844T3 (https=)
IL (2) IL315355A (https=)
PT (1) PT3774844T (https=)
WO (1) WO2019195080A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115160402A (zh) * 2016-03-11 2022-10-11 隐形生物治疗公司 结晶盐形式
PT3774844T (pt) 2018-04-02 2023-03-28 Stealth Biotherapeutics Inc Dipeptídeos cristalinos úteis na síntese de elamipretida
CN117881411A (zh) 2021-06-01 2024-04-12 艾迪雅生物有限责任公司 用于眼部药物的延长释放药物递送系统和使用方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4711166B2 (ja) * 2004-08-03 2011-06-29 株式会社 液晶先端技術開発センター 結晶化装置、および結晶化方法
CA3022250A1 (en) * 2012-12-12 2014-06-12 Ariad Pharmaceuticals, Inc. Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide mono hydrochloride
CN104945453B (zh) * 2014-03-28 2018-06-26 江苏天士力帝益药业有限公司 吡唑衍生物的多晶型物
WO2016001042A1 (en) 2014-06-30 2016-01-07 Flamma S.P.A. Process for the production of d-arginyl-2,6-dimethyl-l-tyrosyl-l-lysyl-l-phenylalaninamide
US10633415B2 (en) * 2015-03-06 2020-04-28 Stealth Biotherapeutics Corp Processes for preparing pharmaceutically relevant peptides
CA3254279A1 (en) * 2015-06-03 2025-03-18 Triastek, Inc. PHARMACEUTICAL FORMS AND RELATED USES
CN115160402A (zh) * 2016-03-11 2022-10-11 隐形生物治疗公司 结晶盐形式
CN110087667A (zh) 2016-08-16 2019-08-02 隐形生物治疗公司 Elamipretide的基于N-羧基酸酐的规模合成
CN110914287A (zh) * 2017-04-05 2020-03-24 隐形生物治疗公司 Boc-d-arg-dmt-lys-(boc)-phe-nh2的结晶盐形式
PT3774844T (pt) 2018-04-02 2023-03-28 Stealth Biotherapeutics Inc Dipeptídeos cristalinos úteis na síntese de elamipretida

Similar Documents

Publication Publication Date Title
JP2021520357A5 (https=)
JP2021530451A5 (https=)
JP2018505199A5 (https=)
JP2009535462A5 (https=)
JPWO2019195080A5 (https=)
CN114206850A (zh) 作为crac抑制剂的2h-苯并吡喃衍生物
JP2007532560A5 (https=)
JP2010507590A5 (https=)
JP2019512542A5 (https=)
RU2007140801A (ru) Углеродсодержащая композиция для получения силицированных изделий
JPWO2021200153A5 (https=)
JPWO2019239387A5 (https=)
JPWO2021166802A5 (https=)
JPWO2022124344A5 (https=)
CN203854306U (zh) 一种磁性玻璃夹持装置
CN212628974U (zh) 一种散热器鳍片组卡点结构
CN216148145U (zh) 一种医用镊子
JPWO2021134045A5 (https=)
CN202668676U (zh) 一种pcb分板器
RU2005102294A (ru) Орбитальное зеркало
CN309884192S (zh) 麦克风配件(用于将麦克风固定于帽檐处)
CN209206164U (zh) 一种多功能折弯机机头
CN2867593Y (zh) 散热片的连接结构
CN115697329A (zh) Palovarotene在抗HBV病毒治疗中的用途
CN208242970U (zh) 一种西服兜盖快速制作装置