JPS62161791A - 2−メチルチアゾロ(4,5−c)キノリン誘導体よりなる薬剤、その製造方法及びそれを使用した中枢神経抑制剤 - Google Patents

2−メチルチアゾロ(4,5−c)キノリン誘導体よりなる薬剤、その製造方法及びそれを使用した中枢神経抑制剤

Info

Publication number
JPS62161791A
JPS62161791A JP61267868A JP26786886A JPS62161791A JP S62161791 A JPS62161791 A JP S62161791A JP 61267868 A JP61267868 A JP 61267868A JP 26786886 A JP26786886 A JP 26786886A JP S62161791 A JPS62161791 A JP S62161791A
Authority
JP
Japan
Prior art keywords
methylthiazolo
acid addition
quinoline
compound
addition salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP61267868A
Other languages
English (en)
Japanese (ja)
Inventor
ヨージェフ クノル
エディト ベレーニィ ネーエ ポルデルマン
カタリン ブダイ ネーエ シモニィ
ベルタ クノル
ジュザァ フュルツ
ユリア ティマール
ガブリエラ ジュイラ
イルディコー ニクリュア
ルイザ ペトオェーツ
アッティラ マーンディ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Egyt Gyogyszervegyeszeti Gyar
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of JPS62161791A publication Critical patent/JPS62161791A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP61267868A 1985-11-12 1986-11-12 2−メチルチアゾロ(4,5−c)キノリン誘導体よりなる薬剤、その製造方法及びそれを使用した中枢神経抑制剤 Pending JPS62161791A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU854302A HU196308B (en) 1985-11-12 1985-11-12 Process for producing pharmaceutical compositions containing 2-methyl-thiazolo/4,5-c/quinoline as active component
HU2251-4302/85 1985-11-12

Publications (1)

Publication Number Publication Date
JPS62161791A true JPS62161791A (ja) 1987-07-17

Family

ID=10967583

Family Applications (1)

Application Number Title Priority Date Filing Date
JP61267868A Pending JPS62161791A (ja) 1985-11-12 1986-11-12 2−メチルチアゾロ(4,5−c)キノリン誘導体よりなる薬剤、その製造方法及びそれを使用した中枢神経抑制剤

Country Status (15)

Country Link
US (1) US4778811A (enExample)
JP (1) JPS62161791A (enExample)
AU (1) AU587505B2 (enExample)
BE (1) BE905718A (enExample)
CH (1) CH669729A5 (enExample)
DE (1) DE3638573A1 (enExample)
FR (1) FR2589733A1 (enExample)
GB (1) GB2182561B (enExample)
HU (1) HU196308B (enExample)
IL (1) IL80609A0 (enExample)
IT (1) IT1214558B (enExample)
NL (1) NL8602877A (enExample)
SE (1) SE8604838L (enExample)
YU (1) YU192086A (enExample)
ZA (1) ZA868582B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU197019B (en) * 1985-11-12 1989-02-28 Egyt Gyogyszervegyeszeti Gyar Process for producing thiqzolo (4,5-c) quinoline derivatives and pharmaceuticals comprising same
HU199423B (en) * 1987-04-24 1990-02-28 Egyt Gyogyszervegyeszeti Gyar Process for producing 3-amino-4-/ethylthio/-quinoline and pharmaceutical compositions comprising such compounds
US4831040A (en) * 1988-02-01 1989-05-16 Rorer Pharmaceutical Corporation Method of prevention and treatment of peptic ulcers
US6110929A (en) 1998-07-28 2000-08-29 3M Innovative Properties Company Oxazolo, thiazolo and selenazolo [4,5-c]-quinolin-4-amines and analogs thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4666916A (en) * 1985-11-08 1987-05-19 Ciba-Geigy Corporation Hexahydro-(1)-benzo-(pyrano and thiopyrano) (4,3-C)pyridines, useful as serotin-2 blocking agents

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
J.AM.CHEM.SOC=1947 *

Also Published As

Publication number Publication date
GB8627042D0 (en) 1986-12-10
DE3638573A1 (de) 1987-05-14
NL8602877A (nl) 1987-06-01
IT1214558B (it) 1990-01-18
IT8622313A0 (it) 1986-11-12
CH669729A5 (enExample) 1989-04-14
ZA868582B (en) 1987-07-29
BE905718A (fr) 1987-05-07
AU587505B2 (en) 1989-08-17
FR2589733A1 (fr) 1987-05-15
HUT44562A (en) 1988-03-28
SE8604838L (sv) 1987-05-13
SE8604838D0 (sv) 1986-11-12
HU196308B (en) 1988-11-28
AU6508686A (en) 1987-05-14
GB2182561B (en) 1989-12-06
YU192086A (en) 1987-12-31
US4778811A (en) 1988-10-18
IL80609A0 (en) 1987-02-27
GB2182561A (en) 1987-05-20

Similar Documents

Publication Publication Date Title
NL8602878A (nl) Thiazolo4,5-cchinolinederivaten, werkwijze voor hun bereiding, alsmede dergelijke derivaten bevattende farmaceutische preparaten.
BG61367B2 (bg) Циклоалкилтриазоли
RU1779251C (ru) Способ получени 1-(4-аминофенил)-4-метил-7,8-метилендиокси-3,4-дигидро-5Н-2,3-бензодиазепина или его кислотно-аддитивных солей
EP1491212A1 (en) Remedy for sleep disturbance
US11141404B1 (en) Formulations and methods for treating acute cannabinoid overdose
JPS6136282A (ja) 窒素を含む複素環式化合物からなる医薬品とその製造方法
HK36793A (en) Ketone derivatives as medicaments for the treatment or prevention of the withdrawal syndrome
GB2243832A (en) 2-substituted 4-acetamido-5-chloro-n-[2-(diethylamino)ethyl]-benzamide derivative
JPH0354922B2 (enExample)
DE60026883T2 (de) Methoden und zusammensetzungen zur behandlung von schmerzen
US10604485B2 (en) Hydrobromide salt of N-(4-chloro-2-hydroxy-3-((3S)-3-piperidinylsulfonyl)phenyl-N′-(3-Fluoro-2-methylphenyl)urea
US3709996A (en) Pharmaceutical compositions containing n-cyclopropyl-1-aminoindane compounds and adapted for administration to obtain inhibition of monoamine oxidase enzyme and process
TW200940543A (en) Maleate, besylate and L-malate salts of 6-(5-chloro-2-pyridyl)-5-[(4-methyl-1-piperazinyl)carbonyloxy]-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyrazine
EP0788795A4 (en) PHARMACOLOGICALLY ACTIVE 2-MERCAPTOBENZIMIDAZOLE DERIVATIVES
US3946004A (en) Phenothiazines, phenoxazines and acridan bis-pyrrolinyl derivatives
US3086910A (en) Central nervous system depressants 3-(2'-pyridyl)-4-quinazolones
JPH05506441A (ja) 加齢関連記憶障害およびその他の認識障害の治療のための化合物
RU2073678C1 (ru) (s)-1-[(10-хлор-6,7-дигидро-4-оксо-3-фенил-4h-бензо/а/хинолизин-1-ил)карбонил]-3-этоксипирролидин, (s)-1-[(10-хлор-6,7-дигидро-4-оксо-3-фенил-4h-бензо/а/хинолизин-1-ил)карбонил]-3-оксипирролидин в качестве промежуточного продукта, композиция, обладающая гипнотическим неседативным действием
US4778811A (en) Pharmaceutical compositions of 2-methyl-thiazolo[4,5-c]quinoline
US4067983A (en) Pharmaceutical compositions and methods
JPH05507933A (ja) Cnsおよび抗高血圧活性を有する置換1―(アルコキシフェニル)ピペラジン類
HUT68215A (en) Use of 5ht1a receptor antagonist compounds for production of antitobacco medicament
DE2000775B2 (de) Substituierte 1,2,3,4-Tetrahydrobenzothieno [23-c] pyridin-Verbindungen, Verfahren zu ihrer Herstellung und pharmazeutische Zubereitung, die diese Verbindungen enthält
DE1770135A1 (de) Verfahren zur Herstellung von 2,4-Benzdiazepinen
CN115433116B (zh) 一种酰化吲哚啉类衍生物、组合物及其应用