JPS6037116B2 - ２―置換オキサゾロピリジン - Google Patents
２―置換オキサゾロピリジンInfo
- Publication number
- JPS6037116B2 JPS6037116B2 JP51089756A JP8975676A JPS6037116B2 JP S6037116 B2 JPS6037116 B2 JP S6037116B2 JP 51089756 A JP51089756 A JP 51089756A JP 8975676 A JP8975676 A JP 8975676A JP S6037116 B2 JPS6037116 B2 JP S6037116B2
- Authority
- JP
- Japan
- Prior art keywords
- formula
- lower alkyl
- formulas
- hydrogen
- pyridine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
- C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C63/00—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
- C07C63/68—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings containing halogen
- C07C63/72—Polycyclic acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/600,169 US4011326A (en) | 1975-07-29 | 1975-07-29 | 2-Substituted oxazolo[4,5-b]pyridine anti-inflammatory agents |
| US600169 | 1977-07-29 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5217495A JPS5217495A (en) | 1977-02-09 |
| JPS6037116B2 true JPS6037116B2 (ja) | 1985-08-24 |
Family
ID=24402575
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP51089756A Expired JPS6037116B2 (ja) | 1975-07-29 | 1976-07-29 | ２―置換オキサゾロピリジン |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US4011326A (enExample) |
| JP (1) | JPS6037116B2 (enExample) |
| AU (1) | AU505159B2 (enExample) |
| BE (1) | BE844577A (enExample) |
| CH (1) | CH603661A5 (enExample) |
| DE (1) | DE2633905A1 (enExample) |
| DK (1) | DK320276A (enExample) |
| ES (1) | ES450245A1 (enExample) |
| FR (1) | FR2319354A1 (enExample) |
| GB (1) | GB1497985A (enExample) |
| HU (1) | HU172167B (enExample) |
| NL (1) | NL7607794A (enExample) |
| SE (1) | SE431545B (enExample) |
| ZA (1) | ZA764527B (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH085368Y2 (ja) * | 1987-03-05 | 1996-02-14 | 日産自動車株式会社 | 内燃機関のコネクティングロッド |
| PT937075E (pt) * | 1996-11-11 | 2004-05-31 | Altana Pharma Ag | Novas imidazo- e oxazolo-piridinas como inibidores da fosfodiesterese |
| ATE327753T1 (de) | 2001-05-15 | 2006-06-15 | Hoffmann La Roche | Carbonsäure-substituierte oxazol-derivate zur verwendung als ppar-alpha und -gamma aktivatoren zur behandlung von diabetes |
| JP4202250B2 (ja) | 2001-07-25 | 2008-12-24 | バイオマリン ファーマシューティカル インコーポレイテッド | 血液脳関門輸送を調節するための組成物および方法 |
| RU2295520C2 (ru) * | 2002-07-03 | 2007-03-20 | Ф.Хоффманн-Ля Рош Аг | ПРОИЗВОДНЫЕ ОКСАЗОЛА И ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ СЕНСИБИЛИЗАТОРОВ ИНСУЛИНА, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ, ОБЛАДАЮЩАЯ АКТИВИРУЮЩИМ ДЕЙСТВИЕМ В ОТНОШЕНИИ PRARα И/ИЛИ PRARγ |
| EP1537091B1 (en) * | 2002-08-30 | 2010-10-06 | F. Hoffmann-La Roche AG | Novel 2-arylthiazole compounds as pparalpha and ppargamma agonists |
| JP4286782B2 (ja) * | 2002-09-12 | 2009-07-01 | エフ．ホフマン−ラ ロシュ アーゲー | 糖尿病の治療に有用な、ｐｐａｒアゴニストとしてのｎ−置換−１ｈ−インドール−５−プロピオン酸化合物 |
| RU2315767C2 (ru) * | 2002-11-25 | 2008-01-27 | Ф.Хоффманн-Ля Рош Аг | Индолилпроизводные, способ их получения, фармацевтическая композиция, способ лечения и/или профилактики заболеваний |
| EP3827747A1 (en) | 2005-04-28 | 2021-06-02 | Otsuka Pharmaceutical Co., Ltd. | Pharma-informatics system |
| CN101594878A (zh) | 2006-09-18 | 2009-12-02 | 雷普特药品公司 | 通过给予受体相关蛋白（rap）-缀合物对肝病症的治疗 |
| DK3395372T3 (da) | 2009-02-20 | 2022-04-19 | Enhanx Biopharm Inc | System til afgivelse af glutathion-baseret medikament |
| CN110075069A (zh) | 2009-05-06 | 2019-08-02 | 实验室护肤股份有限公司 | 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其应用 |
| US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3935195A (en) * | 1969-04-28 | 1976-01-27 | Sterling Drug Inc. | 4,4'-Stilbenebis-pyridooxazoles and related optical brighteners and polymeric compositions brightened thereby |
| FR2148362A1 (en) * | 1971-08-11 | 1973-03-23 | Ferlux | 2-amino-(4,5-b)-oxazolopyridine cpds - with analgesic,anti-inflammato anticonvulsant,muscle relaxant and diuretic activity |
| AR208500A1 (es) * | 1972-06-14 | 1977-02-15 | Merck & Co Inc | Procedimiento para la preparacion de derivados de oxazolo(4,5-b)-piridinas |
-
1975
- 1975-07-29 US US05/600,169 patent/US4011326A/en not_active Expired - Lifetime
-
1976
- 1976-07-14 NL NL7607794A patent/NL7607794A/xx not_active Application Discontinuation
- 1976-07-14 SE SE7608037A patent/SE431545B/xx not_active IP Right Cessation
- 1976-07-15 DK DK320276A patent/DK320276A/da not_active Application Discontinuation
- 1976-07-20 AU AU16052/76A patent/AU505159B2/en not_active Expired
- 1976-07-22 FR FR7622378A patent/FR2319354A1/fr active Granted
- 1976-07-23 CH CH947876A patent/CH603661A5/xx not_active IP Right Cessation
- 1976-07-26 GB GB31065/76A patent/GB1497985A/en not_active Expired
- 1976-07-28 BE BE169289A patent/BE844577A/xx not_active IP Right Cessation
- 1976-07-28 ES ES450245A patent/ES450245A1/es not_active Expired
- 1976-07-28 HU HU76ME00002006A patent/HU172167B/hu unknown
- 1976-07-28 ZA ZA00764527A patent/ZA764527B/xx unknown
- 1976-07-28 DE DE19762633905 patent/DE2633905A1/de not_active Ceased
- 1976-07-29 JP JP51089756A patent/JPS6037116B2/ja not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| CH603661A5 (enExample) | 1978-08-31 |
| US4011326A (en) | 1977-03-08 |
| SE7608037L (sv) | 1977-01-30 |
| DE2633905A1 (de) | 1977-02-17 |
| ES450245A1 (es) | 1979-05-16 |
| NL7607794A (nl) | 1977-02-01 |
| SE431545B (sv) | 1984-02-13 |
| AU505159B2 (en) | 1979-11-08 |
| HU172167B (hu) | 1978-06-28 |
| JPS5217495A (en) | 1977-02-09 |
| DK320276A (da) | 1977-01-30 |
| FR2319354B1 (enExample) | 1979-07-20 |
| GB1497985A (en) | 1978-01-12 |
| BE844577A (fr) | 1977-01-28 |
| AU1605276A (en) | 1978-01-26 |
| ZA764527B (en) | 1978-03-29 |
| FR2319354A1 (fr) | 1977-02-25 |
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