JPS60233073A - 抗高血圧性１，２‐ベンズイソチアゾールピペリジン - Google Patents
抗高血圧性１，２‐ベンズイソチアゾールピペリジンInfo
- Publication number
- JPS60233073A JPS60233073A JP60084681A JP8468185A JPS60233073A JP S60233073 A JPS60233073 A JP S60233073A JP 60084681 A JP60084681 A JP 60084681A JP 8468185 A JP8468185 A JP 8468185A JP S60233073 A JPS60233073 A JP S60233073A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- lower alkyl
- hydrogen
- acid addition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heart & Thoracic Surgery (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US603264 | 1984-04-23 | ||
| US06/603,264 US4528292A (en) | 1984-04-23 | 1984-04-23 | Antihypertensive 1,2-benzisothiazole piperidines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS60233073A true JPS60233073A (ja) | 1985-11-19 |
Family
ID=24414698
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP60084681A Pending JPS60233073A (ja) | 1984-04-23 | 1985-04-22 | 抗高血圧性１，２‐ベンズイソチアゾールピペリジン |
Country Status (17)
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4355037A (en) * | 1981-11-12 | 1982-10-19 | Hoechst-Roussel Pharmaceuticals | 3-(4-Piperidyl)-1,2-benzisoxales |
| US4352811A (en) * | 1981-11-12 | 1982-10-05 | Hoechst-Roussel Pharmaceuticals Inc. | 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles |
| US4458076A (en) * | 1983-05-31 | 1984-07-03 | Hoechst-Roussel Pharmaceuticals | 3-(4-Piperidinyl)-1,2-benzisothiazoles |
-
1984
- 1984-04-23 US US06/603,264 patent/US4528292A/en not_active Expired - Fee Related
-
1985
- 1985-04-17 EP EP85104676A patent/EP0159666B1/en not_active Expired
- 1985-04-17 DE DE8585104676T patent/DE3571031D1/de not_active Expired
- 1985-04-17 AT AT85104676T patent/ATE44031T1/de not_active IP Right Cessation
- 1985-04-18 PT PT80308A patent/PT80308B/pt not_active IP Right Cessation
- 1985-04-19 FI FI851565A patent/FI80692C/fi not_active IP Right Cessation
- 1985-04-22 KR KR1019850002693A patent/KR890000215B1/ko not_active Expired
- 1985-04-22 ZA ZA852984A patent/ZA852984B/xx unknown
- 1985-04-22 NZ NZ211865A patent/NZ211865A/xx unknown
- 1985-04-22 IL IL74981A patent/IL74981A/xx unknown
- 1985-04-22 ES ES542442A patent/ES8608515A1/es not_active Expired
- 1985-04-22 NO NO851606A patent/NO158421C/no unknown
- 1985-04-22 DK DK180185A patent/DK180185A/da not_active Application Discontinuation
- 1985-04-22 GR GR850963A patent/GR850963B/el unknown
- 1985-04-22 PH PH32169A patent/PH23312A/en unknown
- 1985-04-22 JP JP60084681A patent/JPS60233073A/ja active Pending
- 1985-04-23 AU AU41633/85A patent/AU581217B2/en not_active Ceased
-
1986
- 1986-01-28 ES ES551323A patent/ES8704941A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| FI851565A0 (fi) | 1985-04-19 |
| IL74981A (en) | 1990-01-18 |
| PT80308A (en) | 1985-05-01 |
| AU4163385A (en) | 1985-10-31 |
| FI851565L (fi) | 1985-10-24 |
| PT80308B (en) | 1987-02-10 |
| ES542442A0 (es) | 1986-06-16 |
| GR850963B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1985-11-25 |
| NZ211865A (en) | 1989-01-06 |
| EP0159666A2 (en) | 1985-10-30 |
| IL74981A0 (en) | 1985-08-30 |
| ES8608515A1 (es) | 1986-06-16 |
| NO158421C (no) | 1988-09-07 |
| DK180185D0 (da) | 1985-04-22 |
| FI80692C (fi) | 1990-07-10 |
| ES551323A0 (es) | 1987-04-16 |
| NO158421B (no) | 1988-05-30 |
| EP0159666A3 (en) | 1987-01-14 |
| NO851606L (no) | 1985-10-24 |
| PH23312A (en) | 1989-06-30 |
| ATE44031T1 (de) | 1989-06-15 |
| ES8704941A1 (es) | 1987-04-16 |
| US4528292A (en) | 1985-07-09 |
| FI80692B (fi) | 1990-03-30 |
| ZA852984B (en) | 1986-01-29 |
| EP0159666B1 (en) | 1989-06-14 |
| KR850007262A (ko) | 1985-12-02 |
| AU581217B2 (en) | 1989-02-16 |
| DE3571031D1 (en) | 1989-07-20 |
| KR890000215B1 (ko) | 1989-03-10 |
| DK180185A (da) | 1985-10-24 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2656189B2 (ja) | ベンゾイソチアゾールおよびベンゾイソキサゾール−３−カルボキサミド、その製法およびそれよりなる抗精神病剤 | |
| KR0123441B1 (ko) | 아릴 피페라지닐-헤테로사이클릭 화합물의 제조방법 | |
| JP3294961B2 (ja) | 新規イミダゾール誘導体及びその製造法 | |
| JP3018619B2 (ja) | ６，７−ジヒドロ−３−フェニル−１，２−ベンズイソオキサゾール−４（５ｈ）−オンおよびオール、その製法およびそれを含有する医薬 | |
| JPH02240068A (ja) | 中枢神経系に活性を有し、血圧降下活性を有するイミダゾール誘導体、それらの製造方法、ならびにそれらを含有する製薬組成物 | |
| JPH05507281A (ja) | ４−（１，２−ベンゾイソキサゾリル）ピペリジン抗精神病薬 | |
| JPH03388B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| HU176881B (en) | Process for producing derivatives of urea | |
| US3576808A (en) | N-4-phenyl-1-piperazinylalkyl-5-phenyl-oxazolidinones | |
| HU191076B (en) | Process for producing 6-fluoro/-3-(-1-heterocyclo-)-propyl/- 1,2-benzisoxazol derivatives and phrmaceiutical compositions containing them | |
| DE69227207T2 (de) | 1-Piperazinyl-2-butene und 2-butyne, Zwischenverbindungen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel | |
| JPH0699396B2 (ja) | 新規オキサゾロピリジン誘導体 | |
| JP2552494B2 (ja) | イミダゾチアジアジン誘導体及びその製造法 | |
| JPS60233073A (ja) | 抗高血圧性１，２‐ベンズイソチアゾールピペリジン | |
| CA2220140C (en) | (2-morpholinylmethyl)benzamide derivatives | |
| KR880001715B1 (ko) | 1-푸릴-3,4-디하이드로이소퀴놀린의 제조방법 | |
| CH628885A5 (en) | Piperidine derivative | |
| HU208970B (en) | Process for producing new thienloxyalkyl derivatives and pharmaceutical compositions comprising same | |
| JP2564719B2 (ja) | ８−アザビシクロ〔３．２．１〕オクチルアルキルチアゾリジノン類 | |
| US3225037A (en) | 10-[(amino- and acylamino-1-piperidyl) lower-alkyl]-phenothiazines | |
| EP0364091B1 (en) | Antipsychotic 4-(4-(3-benzisothiazolyl)-1-piperazinyl)butyl bridged bicyclic imides | |
| DE69223422T2 (de) | Benzothiadiazinderivate | |
| JPS58177980A (ja) | 新規なベンズイソオキサゾ−ル誘導体 | |
| KR890002093B1 (ko) | 융합된 방향족 옥사제핀 및 이의 황 동족체 및 이의 제조방법 | |
| EP0147691B1 (en) | Antihypertensive 3-aryl-1,2-benzisoxazolsulfonyl and-sulfinyl-alkanoic acids, a process for their preparation and their use for the preparation of medicaments |