JPS5872565A - ピペリジン誘導体およびその製造方法 - Google Patents

ピペリジン誘導体およびその製造方法

Info

Publication number
JPS5872565A
JPS5872565A JP56170536A JP17053681A JPS5872565A JP S5872565 A JPS5872565 A JP S5872565A JP 56170536 A JP56170536 A JP 56170536A JP 17053681 A JP17053681 A JP 17053681A JP S5872565 A JPS5872565 A JP S5872565A
Authority
JP
Japan
Prior art keywords
formula
mol
water
substituted
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP56170536A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6135177B2 (enExample
Inventor
シユナイダ−・ロ−ランド
ヴアロラン・クリスチヤン
ビツグ・デニス
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to CA000388595A priority Critical patent/CA1173039A/en
Priority to ZA817373A priority patent/ZA817373B/xx
Priority to IE2500/81A priority patent/IE51707B1/en
Priority to NO813577A priority patent/NO153890C/no
Priority to DK469381A priority patent/DK157853C/da
Priority to JP56170536A priority patent/JPS5872565A/ja
Priority to PT73875A priority patent/PT73875B/pt
Priority to NZ198748A priority patent/NZ198748A/en
Priority to GR66337A priority patent/GR75364B/el
Priority to FI813330A priority patent/FI77850C/fi
Priority to ES506500A priority patent/ES506500A0/es
Priority to AU76769/81A priority patent/AU545739B2/en
Publication of JPS5872565A publication Critical patent/JPS5872565A/ja
Publication of JPS6135177B2 publication Critical patent/JPS6135177B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP56170536A 1981-10-23 1981-10-23 ピペリジン誘導体およびその製造方法 Granted JPS5872565A (ja)

Priority Applications (12)

Application Number Priority Date Filing Date Title
CA000388595A CA1173039A (en) 1981-10-23 1981-10-23 4-benzyloxypiperidine compounds
ZA817373A ZA817373B (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
IE2500/81A IE51707B1 (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
NO813577A NO153890C (no) 1981-10-23 1981-10-23 Analogifremgangsmaate for fremstilling av terapeutisk aktive piperidinderivater.
DK469381A DK157853C (da) 1981-10-23 1981-10-23 Analogifremgangsmaade til fremstilling af 4-benzyloxypiperidinderivater
JP56170536A JPS5872565A (ja) 1981-10-23 1981-10-23 ピペリジン誘導体およびその製造方法
PT73875A PT73875B (fr) 1981-10-23 1981-10-23 Procede de preparation de derives de piperidine applicables en therapeutique
NZ198748A NZ198748A (en) 1981-10-23 1981-10-23 Piperidine derivatives and pharmaceutical compositions
GR66337A GR75364B (enExample) 1981-10-23 1981-10-23
FI813330A FI77850C (fi) 1981-10-23 1981-10-23 Foerfarande foer framstaellning av 4-bensyloxi- eller 4-naftylmetoxipiperidinderivat, vilka har antidepressiv verkan.
ES506500A ES506500A0 (es) 1981-10-23 1981-10-23 Procedimiento de preparacion de derivados de piperidina
AU76769/81A AU545739B2 (en) 1981-10-23 1981-10-23 Piperidine derivatives

Applications Claiming Priority (12)

Application Number Priority Date Filing Date Title
CA000388595A CA1173039A (en) 1981-10-23 1981-10-23 4-benzyloxypiperidine compounds
ZA817373A ZA817373B (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
IE2500/81A IE51707B1 (en) 1981-10-23 1981-10-23 Piperidine derivatives,their preparation and pharmaceutical compositions containing them
NO813577A NO153890C (no) 1981-10-23 1981-10-23 Analogifremgangsmaate for fremstilling av terapeutisk aktive piperidinderivater.
DK469381A DK157853C (da) 1981-10-23 1981-10-23 Analogifremgangsmaade til fremstilling af 4-benzyloxypiperidinderivater
JP56170536A JPS5872565A (ja) 1981-10-23 1981-10-23 ピペリジン誘導体およびその製造方法
PT73875A PT73875B (fr) 1981-10-23 1981-10-23 Procede de preparation de derives de piperidine applicables en therapeutique
NZ198748A NZ198748A (en) 1981-10-23 1981-10-23 Piperidine derivatives and pharmaceutical compositions
GR66337A GR75364B (enExample) 1981-10-23 1981-10-23
FI813330A FI77850C (fi) 1981-10-23 1981-10-23 Foerfarande foer framstaellning av 4-bensyloxi- eller 4-naftylmetoxipiperidinderivat, vilka har antidepressiv verkan.
ES506500A ES506500A0 (es) 1981-10-23 1981-10-23 Procedimiento de preparacion de derivados de piperidina
AU76769/81A AU545739B2 (en) 1981-10-23 1981-10-23 Piperidine derivatives

Publications (2)

Publication Number Publication Date
JPS5872565A true JPS5872565A (ja) 1983-04-30
JPS6135177B2 JPS6135177B2 (enExample) 1986-08-12

Family

ID=27582840

Family Applications (1)

Application Number Title Priority Date Filing Date
JP56170536A Granted JPS5872565A (ja) 1981-10-23 1981-10-23 ピペリジン誘導体およびその製造方法

Country Status (12)

Country Link
JP (1) JPS5872565A (enExample)
AU (1) AU545739B2 (enExample)
CA (1) CA1173039A (enExample)
DK (1) DK157853C (enExample)
ES (1) ES506500A0 (enExample)
FI (1) FI77850C (enExample)
GR (1) GR75364B (enExample)
IE (1) IE51707B1 (enExample)
NO (1) NO153890C (enExample)
NZ (1) NZ198748A (enExample)
PT (1) PT73875B (enExample)
ZA (1) ZA817373B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH04356462A (ja) * 1990-03-28 1992-12-10 Du Pont Merck Pharmaceut Co 向精神薬または植物の真菌殺菌剤としてのピペリジンエーテル誘導体

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02148948U (enExample) * 1989-05-17 1990-12-18
JPH0535676U (ja) * 1991-06-06 1993-05-14 株式会社カネマス 乾燥海草の水戻し用パツク

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH04356462A (ja) * 1990-03-28 1992-12-10 Du Pont Merck Pharmaceut Co 向精神薬または植物の真菌殺菌剤としてのピペリジンエーテル誘導体

Also Published As

Publication number Publication date
FI77850C (fi) 1989-05-10
ES8206476A1 (es) 1982-08-16
DK469381A (da) 1983-04-24
IE51707B1 (en) 1987-02-18
DK157853B (da) 1990-02-26
AU545739B2 (en) 1985-08-01
FI813330L (fi) 1983-04-24
DK157853C (da) 1990-08-06
NO813577L (no) 1983-04-25
IE812500L (en) 1983-04-21
JPS6135177B2 (enExample) 1986-08-12
NZ198748A (en) 1984-08-24
ES506500A0 (es) 1982-08-16
PT73875A (fr) 1981-11-01
FI77850B (fi) 1989-01-31
CA1173039A (en) 1984-08-21
NO153890B (no) 1986-03-03
GR75364B (enExample) 1984-07-13
ZA817373B (en) 1983-03-30
AU7676981A (en) 1983-04-28
NO153890C (no) 1986-06-11
PT73875B (fr) 1983-01-25

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