JPS5818345A - 環状ヘキサペプチドの製法 - Google Patents

環状ヘキサペプチドの製法

Info

Publication number
JPS5818345A
JPS5818345A JP57122252A JP12225282A JPS5818345A JP S5818345 A JPS5818345 A JP S5818345A JP 57122252 A JP57122252 A JP 57122252A JP 12225282 A JP12225282 A JP 12225282A JP S5818345 A JPS5818345 A JP S5818345A
Authority
JP
Japan
Prior art keywords
phe
tyr
ala
lys
val
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP57122252A
Other languages
English (en)
Japanese (ja)
Inventor
ラス・エフ・ナツト
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of JPS5818345A publication Critical patent/JPS5818345A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/16—Somatostatin; related peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Medicinal Chemistry (AREA)
  • Zoology (AREA)
  • Biochemistry (AREA)
  • Toxicology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP57122252A 1981-07-15 1982-07-15 環状ヘキサペプチドの製法 Pending JPS5818345A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/283,404 US4374060A (en) 1981-07-15 1981-07-15 Process for the preparation of cyclic hexapeptide
US283404 1988-12-12

Publications (1)

Publication Number Publication Date
JPS5818345A true JPS5818345A (ja) 1983-02-02

Family

ID=23085903

Family Applications (1)

Application Number Title Priority Date Filing Date
JP57122252A Pending JPS5818345A (ja) 1981-07-15 1982-07-15 環状ヘキサペプチドの製法

Country Status (9)

Country Link
US (1) US4374060A (OSRAM)
EP (1) EP0070021B1 (OSRAM)
JP (1) JPS5818345A (OSRAM)
AT (1) ATE17359T1 (OSRAM)
CA (1) CA1216845A (OSRAM)
DK (1) DK316382A (OSRAM)
ES (1) ES513937A0 (OSRAM)
GR (1) GR76860B (OSRAM)
PT (1) PT75192B (OSRAM)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59148124A (ja) * 1983-02-15 1984-08-24 Konishiroku Photo Ind Co Ltd 磁気記録媒体の製造方法
JPH0748272A (ja) * 1987-07-10 1995-02-21 Sandoz Ag ソマトスタチン類に関する改良
JPWO2020262590A1 (OSRAM) * 2019-06-28 2020-12-30

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4584172A (en) * 1982-09-27 1986-04-22 Aluminum Company Of America Method of making composition suitable for use as inert electrode having good electrical conductivity and mechanical properties
US4508711A (en) * 1983-04-18 1985-04-02 American Cyanamid Company Cyclic pentapeptide displaying somatostatin antagonism and method of treatment of mammals therewith
FR2645870B1 (fr) * 1989-04-12 1993-01-22 Bioetica Sa Procede de reticulation du collagene par le diphenylphosphorylazide, collagene reticule ainsi obtenu et biomateriaux a base de collagene ainsi reticules
US6117841A (en) * 1997-05-30 2000-09-12 Warner-Lambert Company Substituted peptidylamine calcium channel blockers
CN116621941B (zh) * 2022-05-19 2024-07-09 浙江湃肽生物股份有限公司 一种抗皮肤衰老环六肽类化合物及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4102877A (en) * 1976-07-28 1978-07-25 Merck & Co., Inc. Cyclization of peptides
CA1101843A (en) * 1976-08-02 1981-05-26 Daniel F. Veber Cyclic hexapeptides useful for increasing feed efficiency
SU1219587A1 (ru) * 1978-09-29 1986-03-23 Ордена Трудового Красного Знамени Институт Органического Синтеза Ан Латвсср Циклические аналоги каллидина и других пахикининов,обладающие пролонгированным гипотензивным действием в сочетании с низкой или полностью отсутствующей миотропной активностью
US4310518A (en) * 1979-10-31 1982-01-12 Merck & Co., Inc. Cyclic hexapeptide somatostatin analogs
NZ195303A (en) * 1979-10-31 1984-10-19 Merck & Co Inc Cyclic hexapeptide somatostatin analogues,and pharmaceutical compositions
US4235886A (en) * 1979-10-31 1980-11-25 Merck & Co., Inc. Cyclic hexapeptide somatostatin analogs

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS59148124A (ja) * 1983-02-15 1984-08-24 Konishiroku Photo Ind Co Ltd 磁気記録媒体の製造方法
JPH0748272A (ja) * 1987-07-10 1995-02-21 Sandoz Ag ソマトスタチン類に関する改良
JPWO2020262590A1 (OSRAM) * 2019-06-28 2020-12-30
WO2020262590A1 (ja) * 2019-06-28 2020-12-30 味の素株式会社 環状ペプチドの製造方法

Also Published As

Publication number Publication date
EP0070021A1 (en) 1983-01-19
DK316382A (da) 1983-01-16
PT75192B (en) 1985-10-04
ES8305702A1 (es) 1983-04-16
EP0070021B1 (en) 1986-01-08
ATE17359T1 (de) 1986-01-15
PT75192A (en) 1982-08-01
GR76860B (OSRAM) 1984-09-04
CA1216845A (en) 1987-01-20
ES513937A0 (es) 1983-04-16
US4374060A (en) 1983-02-15

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