JPS58172390A - インドリジノ〔８，７−ｂ〕インド−ル誘導体、その製造方法及び該誘導体を含む医薬製剤 - Google Patents

インドリジノ〔８，７−ｂ〕インド−ル誘導体、その製造方法及び該誘導体を含む医薬製剤

Info

Publication number
JPS58172390A
JPS58172390A JP58047356A JP4735683A JPS58172390A JP S58172390 A JPS58172390 A JP S58172390A JP 58047356 A JP58047356 A JP 58047356A JP 4735683 A JP4735683 A JP 4735683A JP S58172390 A JPS58172390 A JP S58172390A
Authority
JP
Japan
Prior art keywords
group
formula
hydrogen
lower alkyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP58047356A
Other languages
English (en)
Japanese (ja)
Inventor
ボルフガング・フロストル
アンゲロ・ストルニ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of JPS58172390A publication Critical patent/JPS58172390A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/58—Preparation of carboxylic acid halides
    • C07C51/60—Preparation of carboxylic acid halides by conversion of carboxylic acids or their anhydrides or esters, lactones, salts into halides with the same carboxylic acid part
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP58047356A 1982-03-24 1983-03-23 インドリジノ〔８，７−ｂ〕インド−ル誘導体、その製造方法及び該誘導体を含む医薬製剤 Pending JPS58172390A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH181182 1982-03-24
CH1811/826 1982-03-24

Publications (1)

Publication Number Publication Date
JPS58172390A true JPS58172390A (ja) 1983-10-11

Family

ID=4219154

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58047356A Pending JPS58172390A (ja) 1982-03-24 1983-03-23 インドリジノ〔８，７−ｂ〕インド−ル誘導体、その製造方法及び該誘導体を含む医薬製剤

Country Status (10)

Country Link
EP (1) EP0089926A3 (https=)
JP (1) JPS58172390A (https=)
AU (1) AU1275983A (https=)
DK (1) DK132283A (https=)
ES (1) ES520843A0 (https=)
FI (1) FI830939L (https=)
GR (1) GR79551B (https=)
NO (1) NO831034L (https=)
PT (1) PT76428B (https=)
ZA (1) ZA832038B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU582663B2 (en) * 1985-08-10 1989-04-06 John Wyeth & Brother Limited Sulphonamides
DE19708917B4 (de) * 1996-03-13 2006-05-24 Volkswagen Ag Axialkolbenpumpe zur Förderung eines Fluides
HRP20041026A2 (en) 2002-04-03 2005-06-30 Orion Corporation Polycyclic compounds as potent alpha2-adrenoceptor antagonists

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2478639A1 (fr) * 1980-03-20 1981-09-25 Sanofi Sa Nouveaux derives de l'indolizino (8,7-b) indole et intermediaires, leur procede de preparation et leur utilisation en therapeutique

Also Published As

Publication number Publication date
FI830939A7 (fi) 1983-09-25
DK132283D0 (da) 1983-03-23
FI830939L (fi) 1983-09-25
ES8500947A1 (es) 1984-11-01
EP0089926A3 (de) 1984-05-16
AU1275983A (en) 1983-09-29
ES520843A0 (es) 1984-11-01
NO831034L (no) 1983-09-26
FI830939A0 (fi) 1983-03-21
PT76428A (de) 1983-04-01
PT76428B (de) 1986-02-04
ZA832038B (en) 1983-12-28
EP0089926A2 (de) 1983-09-28
GR79551B (https=) 1984-10-30
DK132283A (da) 1983-09-25

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