JPS55105685A - Novel oxoimidazoquinoxaline derivatives*their manufacture*their use as drug and pharmaceutic composition containing them - Google Patents

Novel oxoimidazoquinoxaline derivatives*their manufacture*their use as drug and pharmaceutic composition containing them

Info

Publication number
JPS55105685A
JPS55105685A JP1376880A JP1376880A JPS55105685A JP S55105685 A JPS55105685 A JP S55105685A JP 1376880 A JP1376880 A JP 1376880A JP 1376880 A JP1376880 A JP 1376880A JP S55105685 A JPS55105685 A JP S55105685A
Authority
JP
Japan
Prior art keywords
oxoimidazoquinoxaline
drug
derivatives
novel
manufacture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1376880A
Other languages
English (en)
Other versions
JPH0144712B2 (ja
Inventor
Chiyaaruzu Baanzu Aran
Pooru Kei Deibitsudo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Publication of JPS55105685A publication Critical patent/JPS55105685A/ja
Publication of JPH0144712B2 publication Critical patent/JPH0144712B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
    • C07D241/40—Benzopyrazines
    • C07D241/44—Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP1376880A 1979-02-09 1980-02-08 Novel oxoimidazoquinoxaline derivatives*their manufacture*their use as drug and pharmaceutic composition containing them Granted JPS55105685A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7904648 1979-02-09

Publications (2)

Publication Number Publication Date
JPS55105685A true JPS55105685A (en) 1980-08-13
JPH0144712B2 JPH0144712B2 (ja) 1989-09-29

Family

ID=10503082

Family Applications (3)

Application Number Title Priority Date Filing Date
JP1376780A Pending JPS55105683A (en) 1978-02-08 1980-02-08 Novel heterotricyclic derivatives*their manufacture*their use as drug and pharmaceutic composition containing them
JP1376880A Granted JPS55105685A (en) 1979-02-09 1980-02-08 Novel oxoimidazoquinoxaline derivatives*their manufacture*their use as drug and pharmaceutic composition containing them
JP62290801A Pending JPS6456677A (en) 1979-02-09 1987-11-19 Novel heterotricyclic derivatives, manufacture and pharmacological composition

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP1376780A Pending JPS55105683A (en) 1978-02-08 1980-02-08 Novel heterotricyclic derivatives*their manufacture*their use as drug and pharmaceutic composition containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP62290801A Pending JPS6456677A (en) 1979-02-09 1987-11-19 Novel heterotricyclic derivatives, manufacture and pharmacological composition

Country Status (19)

Country Link
US (2) US4333934A (ja)
JP (3) JPS55105683A (ja)
AU (1) AU530820B2 (ja)
BE (2) BE881631A (ja)
CA (1) CA1131633A (ja)
CH (1) CH643257A5 (ja)
DE (1) DE3004750A1 (ja)
DK (1) DK54280A (ja)
ES (1) ES8102129A1 (ja)
FI (1) FI66868C (ja)
FR (1) FR2448535A1 (ja)
HU (1) HU178380B (ja)
IE (1) IE49388B1 (ja)
IL (1) IL59104A (ja)
IT (1) IT1144033B (ja)
NL (1) NL8000812A (ja)
PT (1) PT70804B (ja)
SE (1) SE441449B (ja)
ZA (1) ZA80234B (ja)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008520653A (ja) * 2004-11-17 2008-06-19 レクサン ファーマシューティカルズ インコーポレイテッド １−［（６，７−置換−アルコキシキノキサリニル）アミノカルボニル］−４−（ヘテロ）アリールピペラジン誘導体

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL66835A (en) * 1981-09-24 1988-05-31 Roussel Uclaf 1,4-disubstituted(1,2,4)triazolo(4,3-alpha)quinazolin-5(4h)-one derivatives and their salts,their preparation and pharmaceutical compositions containing them
US4472401A (en) * 1981-11-27 1984-09-18 Roussel Uclaf Pyrimido-quinoxalines having antiallergic properties
US4510143A (en) * 1982-02-17 1985-04-09 Roussel Uclaf Antiallergic pyrimido[1,2-a]quinoxalin-2-carboxylic acid derivatives
SE462338B (sv) * 1982-04-28 1990-06-11 Roussel Uclaf Nya imidazo /1,2-a/ kinoxaliner och deras salter, foerfarande foer framstaellning daerav samt farmaceutiska kompositioner innehaallande densamma
US4696928A (en) * 1985-09-09 1987-09-29 G. D. Searle & Co. Substituted dihydroimidazo[1,2-a]quinoxalines
US5055465A (en) * 1989-05-31 1991-10-08 Berlex Laboratories, Inc. Imidazoquinoxalinones, their aza analogs and process for their preparation
US5182386A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain imidazoquinoxalinones; a new class of gaba brain receptor ligands
GB9212486D0 (en) * 1992-06-12 1992-07-22 Erba Carlo Spa Derivatives of substituted imidazo benzoxazin-1-one and process for their preparation
DE4310523A1 (de) * 1993-03-31 1994-10-06 Basf Ag Imidazolo-chinoxalinone zur Behandlung zentralnervöser Erkrankungen
FR2722789B1 (fr) * 1994-07-20 1996-08-23 Rhone Poulenc Rorer Sa Derives d'acide imidazo (1,2-a)indeno(1,2-e) pyrazine-2-carboxylique, leur preparation et les medicaments les contenant
BR9509055A (pt) * 1994-09-30 1998-06-23 Basf Ag Imidazoloquinoxalinona uso da mesma e composiçao farmacêutica
CN1075498C (zh) * 1997-05-08 2001-11-28 车庆明 一种查尔酮c甙和它的用途
WO2001014348A1 (en) * 1999-08-20 2001-03-01 The Scripps Research Institute Formation of heterocycles
HUP0105406A3 (en) * 2001-12-21 2003-12-29 Sanofi Aventis Imidazo[1,2-a]quinolin derivatives, process for their preparation, pharmaceutical compositions thereof and intermediates
HUP0203976A3 (en) * 2002-11-15 2004-08-30 Sanofi Aventis Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them
JP2014532626A (ja) * 2011-10-21 2014-12-08 グラクソスミスクライン エルエルシー 自然免疫応答を増強する化合物および方法
JP6827237B2 (ja) * 2016-11-02 2021-02-10 株式会社大阪製薬 害虫駆除シート

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE759292A (fr) * 1969-11-27 1971-05-24 Allen & Hanburys Ltd Derives de xanthone, leur preparation et leur emploi
GB1538479A (en) * 1976-05-21 1979-01-17 Roussel Labor Ltd Imidazobenzoxazines
US4145419A (en) * 1976-05-21 1979-03-20 Roussel Uclaf Novel imidazobenzoxazines
US4075343A (en) * 1976-09-13 1978-02-21 Pfizer Inc. Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof
US4229452A (en) * 1977-01-07 1980-10-21 Westwood Pharmaceuticals, Inc. Treatment of inflammatory disorders with 4-trifluoromethylimidazo[1,2-a]quinoxaline
GB1596652A (en) * 1977-01-20 1981-08-26 Roussel Lab Ltd Imidazo (1,2-a) quinoline-2-carboxylic acid and derivatives
GB1576077A (en) * 1977-04-13 1980-10-01 Roussel Lab Ltd 4,5-dihydro-4-oxophyrrolo(1,2-)-quinoxaline-2-carboxylic acids and derivatives
SE444319B (sv) * 1977-11-18 1986-04-07 Roussel Uclaf Nya imidazobensoxazinderivat, forfarande for framstellning derav och farmaceutiska kompositioner innehallande dessa foreningar

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008520653A (ja) * 2004-11-17 2008-06-19 レクサン ファーマシューティカルズ インコーポレイテッド １−［（６，７−置換−アルコキシキノキサリニル）アミノカルボニル］−４−（ヘテロ）アリールピペラジン誘導体

Also Published As

Publication number Publication date
DK54280A (da) 1980-08-10
DE3004750A1 (de) 1980-08-21
IL59104A (en) 1984-02-29
FI66868C (fi) 1984-12-10
ES488386A0 (es) 1980-12-16
FI800391A (fi) 1980-08-10
US4333934A (en) 1982-06-08
CH643257A5 (fr) 1984-05-30
IL59104A0 (en) 1980-05-30
IE49388B1 (en) 1985-10-02
PT70804A (fr) 1980-03-01
SE441449B (sv) 1985-10-07
JPH0144712B2 (ja) 1989-09-29
JPS55105683A (en) 1980-08-13
AU5535180A (en) 1980-08-14
IT8047848A0 (it) 1980-02-08
PT70804B (fr) 1981-08-04
ES8102129A1 (es) 1980-12-16
BE881631A (fr) 1980-08-08
FI66868B (fi) 1984-08-31
JPS6456677A (en) 1989-03-03
FR2448535A1 (fr) 1980-09-05
NL8000812A (nl) 1980-08-12
US4474784A (en) 1984-10-02
AU530820B2 (en) 1983-07-28
IT1144033B (it) 1986-10-29
HU178380B (en) 1982-04-28
ZA80234B (en) 1981-08-26
BE881630A (fr) 1980-08-08
CA1131633A (en) 1982-09-14
SE8000205L (sv) 1980-08-10
IE800249L (en) 1980-08-09
FR2448535B1 (ja) 1983-10-21

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