JPS54128596A - Novel heptanoic ester and its preparation - Google Patents
Novel heptanoic ester and its preparationInfo
- Publication number
- JPS54128596A JPS54128596A JP3636478A JP3636478A JPS54128596A JP S54128596 A JPS54128596 A JP S54128596A JP 3636478 A JP3636478 A JP 3636478A JP 3636478 A JP3636478 A JP 3636478A JP S54128596 A JPS54128596 A JP S54128596A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- heptanoic
- theobromine
- ester
- novel
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Abstract
NEW MATERIAL:A heptanoic ester derivative of formula I: (R is 1W5C alkyl group).
EXAMPLE: 7-(Theobromin-1-yl)-3-oxo-heptanoic methyl ester.
USE: An intermediate for preparing 1-(5-oxohexyl)theobromine, which is a medicine having vesodilator and hematocytolysis actions with slight side effects.
PROCESS: A 1-(3-substituted-propyl)theobromine of formula II: (X is halogen, p- toluene sulfonyloxy) is reacted with dianions of acetoacetate of formula III: (M and M' are alkali metals) at a low temperature to give the desired compound of formula I. The compound of formula II can be obtained by reacting 1-(3-phenoxy-propyl) theobromine with a hydrohalogenic acid.
COPYRIGHT: (C)1979,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3636478A JPS5826914B2 (en) | 1978-03-29 | 1978-03-29 | New heptanoic acid ester derivatives and their production method |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3636478A JPS5826914B2 (en) | 1978-03-29 | 1978-03-29 | New heptanoic acid ester derivatives and their production method |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS54128596A true JPS54128596A (en) | 1979-10-05 |
JPS5826914B2 JPS5826914B2 (en) | 1983-06-06 |
Family
ID=12467769
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP3636478A Expired JPS5826914B2 (en) | 1978-03-29 | 1978-03-29 | New heptanoic acid ester derivatives and their production method |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5826914B2 (en) |
-
1978
- 1978-03-29 JP JP3636478A patent/JPS5826914B2/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
JPS5826914B2 (en) | 1983-06-06 |
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