JPH11193289A5 - - Google Patents

Info

Publication number
JPH11193289A5
JPH11193289A5 JP1997366756A JP36675697A JPH11193289A5 JP H11193289 A5 JPH11193289 A5 JP H11193289A5 JP 1997366756 A JP1997366756 A JP 1997366756A JP 36675697 A JP36675697 A JP 36675697A JP H11193289 A5 JPH11193289 A5 JP H11193289A5
Authority
JP
Japan
Prior art keywords
group
general formula
compound represented
ring
optionally substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP1997366756A
Other languages
English (en)
Japanese (ja)
Other versions
JPH11193289A (ja
Filing date
Publication date
Application filed filed Critical
Priority to JP9366756A priority Critical patent/JPH11193289A/ja
Priority claimed from JP9366756A external-priority patent/JPH11193289A/ja
Priority to US09/367,841 priority patent/US6271223B1/en
Priority to CNB988028875A priority patent/CN1148372C/zh
Priority to CA002282458A priority patent/CA2282458A1/en
Priority to HU0002291A priority patent/HUP0002291A3/hu
Priority to CNB2004100396861A priority patent/CN1282643C/zh
Priority to EP98961598A priority patent/EP0970088A2/en
Priority to KR1019997007706A priority patent/KR20000075641A/ko
Priority to PCT/JP1998/005954 priority patent/WO1999033840A2/en
Priority to AU16906/99A priority patent/AU752095B2/en
Publication of JPH11193289A publication Critical patent/JPH11193289A/ja
Priority to US09/871,655 priority patent/US6624314B2/en
Priority to US10/615,836 priority patent/US7057036B2/en
Publication of JPH11193289A5 publication Critical patent/JPH11193289A5/ja
Pending legal-status Critical Current

Links

JP9366756A 1997-12-26 1997-12-26 ピロールスルホンアミド誘導体 Pending JPH11193289A (ja)

Priority Applications (12)

Application Number Priority Date Filing Date Title
JP9366756A JPH11193289A (ja) 1997-12-26 1997-12-26 ピロールスルホンアミド誘導体
US09/367,841 US6271223B1 (en) 1997-12-26 1998-10-25 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action
AU16906/99A AU752095B2 (en) 1997-12-26 1998-12-25 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha1-blocking action
EP98961598A EP0970088A2 (en) 1997-12-26 1998-12-25 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha1-blocking action
CA002282458A CA2282458A1 (en) 1997-12-26 1998-12-25 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action
HU0002291A HUP0002291A3 (en) 1997-12-26 1998-12-25 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha1-blocking action
CNB2004100396861A CN1282643C (zh) 1997-12-26 1998-12-25 用于制备具有5－羟色胺－2受体拮抗作用和α1－阻断作用的化合物的中间体及其制法
CNB988028875A CN1148372C (zh) 1997-12-26 1998-12-25 具有5－羟色胺－2受体拮抗作用和α1-阻断作用的吡咯噻嗪和吡咯硫杂吖庚因化合物
KR1019997007706A KR20000075641A (ko) 1997-12-26 1998-12-25 세로토닌-2 수용체 길항작용 및 알파 1-저해 작용을 갖는 피롤로티아진 및 피롤로티아제핀 화합물
PCT/JP1998/005954 WO1999033840A2 (en) 1997-12-26 1998-12-25 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha1-blocking action
US09/871,655 US6624314B2 (en) 1997-12-26 2001-06-04 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action
US10/615,836 US7057036B2 (en) 1997-12-26 2003-07-10 Pyrrolothiazine and pyrrolothiazepine compounds having serotonin-2 receptor antagonistic and alpha-1-blocking action

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP9366756A JPH11193289A (ja) 1997-12-26 1997-12-26 ピロールスルホンアミド誘導体

Publications (2)

Publication Number Publication Date
JPH11193289A JPH11193289A (ja) 1999-07-21
JPH11193289A5 true JPH11193289A5 (enExample) 2005-07-28

Family

ID=18487593

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9366756A Pending JPH11193289A (ja) 1997-12-26 1997-12-26 ピロールスルホンアミド誘導体

Country Status (9)

Country Link
US (3) US6271223B1 (enExample)
EP (1) EP0970088A2 (enExample)
JP (1) JPH11193289A (enExample)
KR (1) KR20000075641A (enExample)
CN (2) CN1148372C (enExample)
AU (1) AU752095B2 (enExample)
CA (1) CA2282458A1 (enExample)
HU (1) HUP0002291A3 (enExample)
WO (1) WO1999033840A2 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997020845A1 (fr) 1995-12-01 1997-06-12 Suntory Limited Derives de pyrroloazepine
JPH11193290A (ja) 1997-12-26 1999-07-21 Suntory Ltd ピロールスルホンアミド系化合物
JPH11193289A (ja) 1997-12-26 1999-07-21 Suntory Ltd ピロールスルホンアミド誘導体
US6960579B1 (en) 1998-05-19 2005-11-01 Alcon Manufacturing, Ltd. Serotonergic 5HT7 receptor compounds for treating ocular and CNS disorders
AU784462B2 (en) * 2000-03-31 2006-04-06 Purdue Research Foundation Phosphoramidate prodrugs
IL283725B2 (en) 2017-06-20 2024-04-01 Imbria Pharmaceuticals Inc Compositions and methods for increasing efficiency of cardiac metabolism
WO2020081361A1 (en) 2018-10-17 2020-04-23 Imbria Pharmaceuticals, Inc. Methods of treating rheumatic diseases using trimetazidine-based compounds
US11780811B2 (en) 2020-06-30 2023-10-10 Imbria Pharmaceuticals, Inc. Methods of synthesizing 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate
US11530184B2 (en) 2020-06-30 2022-12-20 Imbria Pharmaceuticals, Inc. Crystal forms of 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate
US11883396B2 (en) 2021-05-03 2024-01-30 Imbria Pharmaceuticals, Inc. Methods of treating kidney conditions using modified forms of trimetazidine

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US240178A (en) 1881-04-12 Feeding device for button-hole sewing-machines
US208631A (en) 1878-10-01 Improvement in trimmers for wax-thread sewing-machines
US236765A (en) 1881-01-18 Attoenet
JP3198117B2 (ja) 1990-02-07 2001-08-13 サントリー株式会社 ピロロアゼピン誘導体
US5075440A (en) 1990-05-03 1991-12-24 Ortho Pharmaceutical Corporation Novel pyrido[2,3-f](1,4)thiazepines and pyrido[3,2-b](1,5)benzothiazepines
FR2675802B1 (fr) * 1991-04-26 1993-12-24 Rhone Poulenc Rorer Sa Antiserotonines, leur preparation et les medicaments les contenant.
WO1993003032A1 (fr) 1991-08-07 1993-02-18 Suntory Limited Compose de pyrroloazepine
CA2093631C (en) 1991-08-07 2003-09-23 Akira Mizuno Pyrroloazepine derivative
IL108634A0 (en) * 1993-02-15 1994-05-30 Wellcome Found Hypolipidaemic heterocyclic compounds, their prepatation and pharmaceutical compositions containing them
AU690622B2 (en) * 1993-12-24 1998-04-30 Daiichi Suntory Pharma Co., Ltd Benzothiazine derivative
DE69630184T2 (de) 1995-11-02 2004-08-12 Daiichi Suntory Pharma Co., Ltd. Verfahren zur Herstellung von 1-substituierten Pyrrol-3-carbonsäure-Derivaten
WO1997020845A1 (fr) 1995-12-01 1997-06-12 Suntory Limited Derives de pyrroloazepine
JPH10251258A (ja) 1997-03-14 1998-09-22 Suntory Ltd ピロロアゼピン系化合物
JPH11193289A (ja) 1997-12-26 1999-07-21 Suntory Ltd ピロールスルホンアミド誘導体
JPH11193290A (ja) * 1997-12-26 1999-07-21 Suntory Ltd ピロールスルホンアミド系化合物

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