JPH07304761A - 不飽和タキサン化合物 - Google Patents

不飽和タキサン化合物

Info

Publication number
JPH07304761A
JPH07304761A JP7110678A JP11067895A JPH07304761A JP H07304761 A JPH07304761 A JP H07304761A JP 7110678 A JP7110678 A JP 7110678A JP 11067895 A JP11067895 A JP 11067895A JP H07304761 A JPH07304761 A JP H07304761A
Authority
JP
Japan
Prior art keywords
formula
compound
taxane derivative
protecting group
taxane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP7110678A
Other languages
English (en)
Japanese (ja)
Inventor
Nicola Mongelli
ニコラ・モンゲリ
Maria Menichincheri
マリア・メニチンチエリ
Bassini Domenico Fusar
ドメニコ・フサール・バツシーニ
Marina Ciomei
マリーナ・チオメイ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Pharmacia SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia SpA filed Critical Pharmacia SpA
Publication of JPH07304761A publication Critical patent/JPH07304761A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
JP7110678A 1994-05-09 1995-05-09 不飽和タキサン化合物 Pending JPH07304761A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9409131A GB9409131D0 (en) 1994-05-09 1994-05-09 Unsaturated taxane compounds
GB9409131.1 1994-05-09

Publications (1)

Publication Number Publication Date
JPH07304761A true JPH07304761A (ja) 1995-11-21

Family

ID=10754759

Family Applications (1)

Application Number Title Priority Date Filing Date
JP7110678A Pending JPH07304761A (ja) 1994-05-09 1995-05-09 不飽和タキサン化合物

Country Status (4)

Country Link
JP (1) JPH07304761A (it)
DE (1) DE19516631A1 (it)
GB (2) GB9409131D0 (it)
IT (1) IT1273612B (it)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998022451A1 (fr) * 1996-11-19 1998-05-28 Daiichi Pharmaceutical Co., Ltd. Derives taxol

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6315500A (en) * 1999-07-28 2001-02-13 Kobe Natural Products And Chemicals Co., Ltd. Multidrug-resistant cancer overcoming agents and process for producing the same
WO2003087078A1 (en) * 2002-04-05 2003-10-23 Natural Pharmaceuticals, Inc. Selective acylation of secondary hydroxyl groups

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2109861C (en) * 1992-12-04 1999-03-16 Shu-Hui Chen 6,7-modified paclitaxels
IL107950A (en) * 1992-12-15 2001-04-30 Upjohn Co b 7, b 8 - Matano - Taxols, their preparation and pharmaceutical preparations against malignant tumors containing them

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998022451A1 (fr) * 1996-11-19 1998-05-28 Daiichi Pharmaceutical Co., Ltd. Derives taxol

Also Published As

Publication number Publication date
DE19516631A1 (de) 1995-11-16
GB2289277A (en) 1995-11-15
ITMI950872A0 (it) 1995-04-28
GB9409131D0 (en) 1994-06-29
IT1273612B (it) 1997-07-08
GB2289277B (en) 1998-08-19
ITMI950872A1 (it) 1996-10-28
GB9509353D0 (en) 1995-06-28

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