JPH05509100A - ボンベシン拮抗薬 - Google Patents

ボンベシン拮抗薬

Info

Publication number
JPH05509100A
JPH05509100A JP3513218A JP51321891A JPH05509100A JP H05509100 A JPH05509100 A JP H05509100A JP 3513218 A JP3513218 A JP 3513218A JP 51321891 A JP51321891 A JP 51321891A JP H05509100 A JPH05509100 A JP H05509100A
Authority
JP
Japan
Prior art keywords
ala
pro
phe
formula
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP3513218A
Other languages
English (en)
Japanese (ja)
Inventor
クル，フレデリック，チャールズ
レバン，ヨハン，ヤコブ
Original Assignee
ザ　ウエルカム　ファウンデーション　リミテッド
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ザ　ウエルカム　ファウンデーション　リミテッド filed Critical ザ　ウエルカム　ファウンデーション　リミテッド
Publication of JPH05509100A publication Critical patent/JPH05509100A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • C07K7/086—Bombesin; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP3513218A 1990-07-31 1991-07-30 ボンベシン拮抗薬 Pending JPH05509100A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9016810.5 1990-07-31
GB909016810A GB9016810D0 (en) 1990-07-31 1990-07-31 Peptides

Publications (1)

Publication Number Publication Date
JPH05509100A true JPH05509100A (ja) 1993-12-16

Family

ID=10679953

Family Applications (1)

Application Number Title Priority Date Filing Date
JP3513218A Pending JPH05509100A (ja) 1990-07-31 1991-07-30 ボンベシン拮抗薬

Country Status (20)

Country Link
EP (1) EP0541654A1 (enExample)
JP (1) JPH05509100A (enExample)
AU (1) AU653544B2 (enExample)
CA (1) CA2088166A1 (enExample)
CZ (1) CZ8093A3 (enExample)
FI (1) FI930411A7 (enExample)
GB (1) GB9016810D0 (enExample)
HU (1) HUT63178A (enExample)
IE (1) IE912671A1 (enExample)
IL (1) IL99009A0 (enExample)
MC (1) MC2312A1 (enExample)
MY (1) MY107031A (enExample)
NO (1) NO930262D0 (enExample)
NZ (1) NZ239183A (enExample)
PL (1) PL167322B1 (enExample)
PT (1) PT98498A (enExample)
SK (1) SK3893A3 (enExample)
TW (1) TW234130B (enExample)
WO (1) WO1992002545A1 (enExample)
ZA (1) ZA915978B (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5723578A (en) * 1987-09-24 1998-03-03 The Administrators Of Tulane Educational Fund Peptide analogs of bombesin
US5877277A (en) 1987-09-24 1999-03-02 Biomeasure, Inc. Octapeptide bombesin analogs
US5436137A (en) * 1992-07-27 1995-07-25 Oregon Regional Primate Research Center DNA sequence which encodes a peptide capable of promoting acrosome reaction
US5620955A (en) * 1993-06-18 1997-04-15 Peptide Technologies Corporation Bombesin receptor antagonists and uses thereof
JP4954983B2 (ja) 2005-05-18 2012-06-20 ファーマサイエンス・インコーポレイテッド Ｂｉｒドメイン結合化合物
RU2418807C2 (ru) 2005-10-25 2011-05-20 Аегера Терапьютикс Инк. Соединения, связывающие bir домены iap
MX340870B (es) 2010-02-12 2016-07-27 Pharmascience Inc Compuestos de unión del dominio de repetición de inhibidores de proteínas de apoptosis de baculovirus.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU618029B2 (en) * 1987-11-02 1991-12-12 Imperial Chemical Industries Plc Polypeptide compounds

Also Published As

Publication number Publication date
EP0541654A1 (en) 1993-05-19
MC2312A1 (fr) 1993-09-27
ZA915978B (en) 1993-04-28
AU8311191A (en) 1992-03-02
MY107031A (en) 1995-08-30
WO1992002545A1 (en) 1992-02-20
PL167322B1 (pl) 1995-08-31
HU9300239D0 (en) 1993-04-28
NZ239183A (en) 1993-07-27
PT98498A (pt) 1992-05-29
GB9016810D0 (en) 1990-09-12
IE912671A1 (en) 1992-02-12
IL99009A0 (en) 1992-07-15
FI930411A0 (fi) 1993-01-29
NO930262L (no) 1993-01-26
PL297652A1 (enExample) 1992-07-13
CA2088166A1 (en) 1992-02-01
TW234130B (enExample) 1994-11-11
SK3893A3 (en) 1993-07-07
AU653544B2 (en) 1994-10-06
FI930411A7 (fi) 1993-01-29
CZ8093A3 (en) 1994-01-19
NO930262D0 (no) 1993-01-26
HUT63178A (en) 1993-07-28

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