JPH05255312A - 有機材料用安定剤として使用するための新規のテトラメチルピペリジン化合物 - Google Patents

有機材料用安定剤として使用するための新規のテトラメチルピペリジン化合物

Info

Publication number
JPH05255312A
JPH05255312A JP4355130A JP35513092A JPH05255312A JP H05255312 A JPH05255312 A JP H05255312A JP 4355130 A JP4355130 A JP 4355130A JP 35513092 A JP35513092 A JP 35513092A JP H05255312 A JPH05255312 A JP H05255312A
Authority
JP
Japan
Prior art keywords
group
carbon atoms
formula
same
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP4355130A
Other languages
English (en)
Japanese (ja)
Inventor
Valerio Borzatta
ボルザッタ ヴァレリオ
Graziano Vignali
ヴィニャリ グラジアノ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of JPH05255312A publication Critical patent/JPH05255312A/ja
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08KUse of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00Use of organic ingredients
    • C08K5/16Nitrogen-containing compounds
    • C08K5/34Heterocyclic compounds having nitrogen in the ring
    • C08K5/3442Heterocyclic compounds having nitrogen in the ring having two nitrogen atoms in the ring
    • C08K5/3445Five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Polymers & Plastics (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Materials For Photolithography (AREA)
  • Detergent Compositions (AREA)
JP4355130A 1991-12-17 1992-12-17 有機材料用安定剤として使用するための新規のテトラメチルピペリジン化合物 Pending JPH05255312A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT91A003374 1991-12-17
ITMI913374A IT1252227B (it) 1991-12-17 1991-12-17 Composti tetrametilpiperidinici atti all'impiego come stabilizzanti per materiali organici

Publications (1)

Publication Number Publication Date
JPH05255312A true JPH05255312A (ja) 1993-10-05

Family

ID=11361349

Family Applications (1)

Application Number Title Priority Date Filing Date
JP4355130A Pending JPH05255312A (ja) 1991-12-17 1992-12-17 有機材料用安定剤として使用するための新規のテトラメチルピペリジン化合物

Country Status (10)

Country Link
US (1) US5310767A (OSRAM)
EP (1) EP0548015B1 (OSRAM)
JP (1) JPH05255312A (OSRAM)
KR (1) KR100248537B1 (OSRAM)
BR (1) BR9205032A (OSRAM)
CA (1) CA2085379A1 (OSRAM)
DE (1) DE69207370T2 (OSRAM)
ES (1) ES2082434T3 (OSRAM)
IT (1) IT1252227B (OSRAM)
TW (1) TW242156B (OSRAM)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1263892B (it) * 1993-02-11 1996-09-05 Graziano Vignali Composti piperidin-triazinici atti all'impiego come stabilizzanti per materiali organici
US5721250A (en) * 1993-12-23 1998-02-24 Merck & Co. Inc. Di-and tri-substituted piperidines, pyrrolidines and hexahydro-1H-azepines promote release of growth hormone
AU780006B2 (en) 2000-03-06 2005-02-24 Acadia Pharmaceuticals, Inc. Azacyclic compounds for use in the treatment of serotonin related diseases
NZ571695A (en) 2001-12-28 2010-02-26 Acadia Pharm Inc Spiroazacyclic compounds as monoamine receptor for modulating 5-HT2A receptor-mediated events
US7253186B2 (en) 2002-06-24 2007-08-07 Carl-Magnus Andersson N-substituted piperidine derivatives as serotonin receptor agents
MXPA04012893A (es) 2002-06-24 2005-03-31 Acadia Pharm Inc Derivados de piperidina n-substituidos como agentes receptores de serotonina.
US7538222B2 (en) 2002-06-24 2009-05-26 Acadia Pharmaceuticals, Inc. N-substituted piperidine derivatives as serotonin receptor agents
PT1587789E (pt) 2003-01-16 2008-12-16 Acadia Pharm Inc Agonistas inversos selectivos para receptores 2a/2c da serotonina como agentes terapêuticos para doenças neurodegenerativas
US20050261278A1 (en) 2004-05-21 2005-11-24 Weiner David M Selective serotonin receptor inverse agonists as therapeutics for disease
US7820695B2 (en) 2004-05-21 2010-10-26 Acadia Pharmaceuticals, Inc. Selective serotonin receptor inverse agonists as therapeutics for disease
CA2580136C (en) 2004-09-27 2015-08-18 Acadia Pharmaceuticals Inc. Synthesis of n-(4-fluorobenzyl)-n-(1-methylpiperidin-4-yl)-n'-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and crystalline forms
US7790899B2 (en) 2004-09-27 2010-09-07 Acadia Pharmaceuticals, Inc. Synthesis of N-(4-fluorobenzyl)-N-(1-methylpiperidin-4-yl)-N′-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and crystalline forms
CA2681506C (en) 2007-03-19 2016-05-24 Perry Peters Combinations of 5-ht2a inverse agonists and antagonists with antipsychotics
TWI386451B (zh) * 2009-05-12 2013-02-21 Nanya Plastics Corp 一種pvc樹脂組成物及其製品
CA2992728A1 (en) 2015-07-20 2017-01-26 Acadia Pharmaceuticals Inc. Methods for preparing n-(4-fluorobenzyl)-n-(1-methylpiperidin-4-yl)-n'-(4-(2-methylpropyloxy)phenylmethyl)carbamide and its tartrate salt and polymorphic form c
WO2017165635A1 (en) 2016-03-25 2017-09-28 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome p450 modulators
US10953000B2 (en) 2016-03-25 2021-03-23 Acadia Pharmaceuticals Inc. Combination of pimavanserin and cytochrome P450 modulators
EP3558311A1 (en) 2016-12-20 2019-10-30 Acadia Pharmaceuticals Inc. Pimavanserin alone or in combination for use in the treatment of alzheimer's disease psychosis
EP3615028A1 (en) 2017-04-28 2020-03-04 Acadia Pharmaceuticals Inc. Pimavanserin for treating impulse control disorder
US20210077479A1 (en) 2017-08-30 2021-03-18 Acadia Pharmaceuticals Inc. Formulations of pimavanserin

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3684765A (en) * 1970-01-08 1972-08-15 Sankyo Co Stabilization of synthetic polymers
GB1393551A (en) * 1972-04-21 1975-05-07 Ciba Geigy Ag Piperidine derivatives
JPS557861B2 (OSRAM) * 1972-10-04 1980-02-28
IT1060458B (it) * 1975-12-18 1982-08-20 Chimosa Chimica Organica Spa Composti piperidil triazinici adatti per la stabilizzazione di polimeri sintetici e procedimento per la loro preparazione
IT1097753B (it) * 1978-07-28 1985-08-31 Chimosa Chimica Organica Spa Compcsti piperidinici, processo per la loro preparazione e loro impiego come stabil izzanti per polimeri sintetici
IT7921841A0 (it) * 1979-04-13 1979-04-13 Chimosa Chimica Organica Spa Nuovi composti piperidinici, processo per la loro preparazione e loro impiego come stabilizzanti per polimeri sintetici.
DE2944729A1 (de) * 1979-11-06 1981-05-14 Hoechst Ag, 6000 Frankfurt Neue triazinstabilisatoren
DE3382687D1 (de) * 1982-09-30 1993-07-01 Ciba Geigy Ag Mit bis-(polyalkylpiperidinyl-amino)-1,3,5-triazinen stabilisierte polyolefine.
JPS59122487A (ja) * 1982-12-28 1984-07-14 Sankyo Co Ltd ピペリジル−トリアジン−トリアミン誘導体及び高分子材料用安定剤
IT1193659B (it) * 1983-02-04 1988-07-21 Chimosa Chimica Organica Spa Composti piperidinil-triazinici utili come stabilizzanti per polimeri sintetici
JPS6181441A (ja) * 1984-09-28 1986-04-25 Adeka Argus Chem Co Ltd 高分子材料組成物
JPS6218444A (ja) * 1985-07-16 1987-01-27 Adeka Argus Chem Co Ltd 安定化された高分子材料組成物
IT1227334B (it) * 1988-08-04 1991-04-08 Ciba Geigy Spa Composti piperidin triazinici atti all'impiego come stabilizzanti per materiali organici.
IT1231329B (it) * 1989-07-28 1991-11-28 Ciba Geigy Spa Composti piperazin piperidinici atti all'impiego come stabilizzanti per materiali organici
IT1237129B (it) * 1989-11-10 1993-05-18 Valerio Borzatta Composti piperidin-triazinici atti all'impiego come stabilizzanti per materiali organici.
IT1243374B (it) * 1990-07-27 1994-06-10 Ciba Geigy Spa Composti piperidin-triazinici contenenti gruppi tetraidrofuranici o tetraidropiranici atti all'impiego come stabilizzanti per materiali organici
IT1243433B (it) * 1990-10-03 1994-06-10 Ciba Geigy Spa Composti piperidin-triazinici atti all'impiego come stabilizzanti per materiali organici
IT1243409B (it) * 1990-12-17 1994-06-10 Ciba Geigy Spa Composti piperidinici contenenti gruppi silenici atti all'impiego come stabilizzanti per materiali organici

Also Published As

Publication number Publication date
DE69207370D1 (de) 1996-02-15
CA2085379A1 (en) 1993-06-18
TW242156B (OSRAM) 1995-03-01
US5310767A (en) 1994-05-10
IT1252227B (it) 1995-06-05
EP0548015A1 (en) 1993-06-23
EP0548015B1 (en) 1996-01-03
KR100248537B1 (ko) 2000-04-01
ITMI913374A1 (it) 1993-06-17
ES2082434T3 (es) 1996-03-16
BR9205032A (pt) 1993-06-22
DE69207370T2 (de) 1996-11-14
ITMI913374A0 (it) 1991-12-17

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