JPH02501929A - 医学的使用 - Google Patents
医学的使用Info
- Publication number
- JPH02501929A JPH02501929A JP63508894A JP50889488A JPH02501929A JP H02501929 A JPH02501929 A JP H02501929A JP 63508894 A JP63508894 A JP 63508894A JP 50889488 A JP50889488 A JP 50889488A JP H02501929 A JPH02501929 A JP H02501929A
- Authority
- JP
- Japan
- Prior art keywords
- treatment
- compound
- prevention
- formula
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/10—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
- A61P5/12—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH for decreasing, blocking or antagonising the activity of the posterior pituitary hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE8704248A SE8704248D0 (sv) | 1987-10-30 | 1987-10-30 | Medical use |
SE8704248-7 | 1987-10-30 |
Publications (1)
Publication Number | Publication Date |
---|---|
JPH02501929A true JPH02501929A (ja) | 1990-06-28 |
Family
ID=20370069
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP63508894A Pending JPH02501929A (ja) | 1987-10-30 | 1988-10-27 | 医学的使用 |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP0339071A1 (ko) |
JP (1) | JPH02501929A (ko) |
KR (1) | KR890701587A (ko) |
AU (1) | AU2620388A (ko) |
DK (1) | DK322189A (ko) |
HU (1) | HU203663B (ko) |
IL (1) | IL88205A0 (ko) |
SE (1) | SE8704248D0 (ko) |
WO (1) | WO1989003833A1 (ko) |
Families Citing this family (24)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1327796C (en) * | 1987-07-16 | 1994-03-15 | Jorg Senn-Bilfinger | Diazoles |
US5081253A (en) * | 1989-12-21 | 1992-01-14 | American Home Products Corporation | Imidazo(4,5-c)pyridines as antiosteoporotic agents |
US5464843A (en) * | 1992-06-23 | 1995-11-07 | G.D. Searle & Co. | Imidazo[1,2-a]pyridinyldiacid compounds for cognitive enhancement and for treatment of cognitive disorders and neutrotoxic injury |
JPH11505524A (ja) * | 1995-05-01 | 1999-05-21 | 藤沢薬品工業株式会社 | イミダゾ1,2−aピリジンおよびイミダゾ1,2−aピリデジン誘導体、および骨吸収阻害剤としてのその用途 |
GB9518552D0 (en) * | 1995-09-11 | 1995-11-08 | Fujisawa Pharmaceutical Co | New heterocyclic compounds |
US7709468B2 (en) | 2005-09-02 | 2010-05-04 | Abbott Laboratories | Imidazo based heterocycles |
WO2012087833A1 (en) | 2010-12-22 | 2012-06-28 | Abbott Laboratories | Hepatitis c inhibitors and uses thereof |
DE102012200349A1 (de) | 2012-01-11 | 2013-07-11 | Bayer Intellectual Property Gmbh | Substituierte annellierte Pyrimidine und Triazine und ihre Verwendung |
US9624214B2 (en) | 2012-11-05 | 2017-04-18 | Bayer Pharma Aktiengesellschaft | Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
US8796305B2 (en) | 2012-11-05 | 2014-08-05 | Bayer Pharma Aktiengesellschaft | Carboxy-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
US9126998B2 (en) | 2012-11-05 | 2015-09-08 | Bayer Pharma AG | Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
US8778964B2 (en) | 2012-11-05 | 2014-07-15 | Bayer Pharma Aktiengesellschaft | Hydroxy-substituted imidazo[1,2-a]-pyridinecarboxamides and their use |
CA2914100A1 (en) | 2013-06-04 | 2014-12-11 | Bayer Pharma Aktiengesellschaft | 3-aryl-substituted imidazo[1,2-a]pyridines and the use thereof |
JP2016523944A (ja) | 2013-07-10 | 2016-08-12 | バイエル・ファルマ・アクティエンゲゼルシャフト | ベンジル−1H−ピラゾロ[3,4−b]ピリジンおよびその使用 |
CN106459090A (zh) | 2014-02-19 | 2017-02-22 | 拜耳制药股份公司 | 3‑(嘧啶‑2‑基)咪唑并[1,2‑a]吡啶 |
EP3119777A1 (de) | 2014-03-21 | 2017-01-25 | Bayer Pharma Aktiengesellschaft | Cyano-substituierte imidazo[1,2-a]pyridincarboxamide und ihre verwendung |
EP3137463A1 (de) * | 2014-05-02 | 2017-03-08 | Bayer Pharma Aktiengesellschaft | Enantiomere des n-(2-amino-5-fluor-2-methylpentyl)-8-[(2,6-difluorbenzyl)oxy]-2-methylimidazo[1,2-a]pyridin-3-carboxamids sowie der di- and tri-fluor-derivate zur behandlung von kardiovaskulären erkrankungen |
EP3137465A1 (de) * | 2014-05-02 | 2017-03-08 | Bayer Pharma Aktiengesellschaft | 6-chlor-substituierte imidazo[1,2-a]pyridincarboxamide und ihre verwendung als stimulatoren der löslichen guanylatcyclase |
JP2017514899A (ja) * | 2014-05-02 | 2017-06-08 | バイエル・ファルマ・アクティエンゲゼルシャフト | ヘテロシクリル−およびヘテロアリール−置換イミダゾ[1,2−a]ピリジンおよびその使用 |
CN107001361A (zh) | 2014-12-02 | 2017-08-01 | 拜耳医药股份有限公司 | 杂芳基取代的咪唑并[1,2‑a]吡啶及其用途 |
EP3227286B1 (de) | 2014-12-02 | 2018-12-26 | Bayer Pharma Aktiengesellschaft | Substituierte pyrazolo[1,5-a]pyridine und imidazo[1,2-a]pyrazine und ihre verwendung |
JP2018505885A (ja) | 2015-02-05 | 2018-03-01 | バイエル・ファルマ・アクティエンゲゼルシャフト | 置換ピラゾロ[1,5−a]−ピリジン−3−カルボキサミドおよびその使用 |
WO2016124564A1 (de) | 2015-02-05 | 2016-08-11 | Bayer Pharma Aktiengesellschaft | N-substituierte 8-[(2,6-difluorbenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyrazin-3-carboxamid-derivate als stimulatoren der löslichen guanylatcyclase (sgc) zur behandlung von kardiovaskulären erkrankungen |
WO2018184976A1 (de) | 2017-04-05 | 2018-10-11 | Bayer Pharma Aktiengesellschaft | Substituierte imidazo[1,2-a]pyridincarboxamide und ihre verwendung |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0068378B1 (en) * | 1981-06-26 | 1986-03-05 | Schering Corporation | Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them |
US4468400A (en) * | 1982-12-20 | 1984-08-28 | Schering Corporation | Antiulcer tricyclic imidazo [1,2-a]pyridines |
DE3446778A1 (de) * | 1984-12-21 | 1986-07-03 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue imidazoderivate, ihre herstellung und diese verbindungen enthaltende arzneimittel |
US4725601A (en) * | 1985-06-04 | 1988-02-16 | Fujisawa Pharmaceutical Co., Ltd. | Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers |
EP0228006A1 (en) * | 1985-12-16 | 1987-07-08 | Fujisawa Pharmaceutical Co., Ltd. | Imidazopyridine compounds and processes for preparation thereof |
-
1987
- 1987-10-30 SE SE8704248A patent/SE8704248D0/xx unknown
-
1988
- 1988-10-27 HU HU886708A patent/HU203663B/hu not_active IP Right Cessation
- 1988-10-27 EP EP88909620A patent/EP0339071A1/en not_active Withdrawn
- 1988-10-27 AU AU26203/88A patent/AU2620388A/en not_active Abandoned
- 1988-10-27 JP JP63508894A patent/JPH02501929A/ja active Pending
- 1988-10-27 WO PCT/SE1988/000576 patent/WO1989003833A1/en not_active Application Discontinuation
- 1988-10-27 KR KR1019890701209A patent/KR890701587A/ko not_active Application Discontinuation
- 1988-10-28 IL IL88205A patent/IL88205A0/xx unknown
-
1989
- 1989-06-28 DK DK322189A patent/DK322189A/da not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
DK322189D0 (da) | 1989-06-28 |
AU2620388A (en) | 1989-05-23 |
SE8704248D0 (sv) | 1987-10-30 |
WO1989003833A1 (en) | 1989-05-05 |
IL88205A0 (en) | 1989-06-30 |
DK322189A (da) | 1989-06-28 |
EP0339071A1 (en) | 1989-11-02 |
KR890701587A (ko) | 1989-12-21 |
HU203663B (en) | 1991-09-30 |
HUT51138A (en) | 1990-04-28 |
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