JP6856657B2 - 血液学的悪性疾患および固形腫瘍の処置のためのｉｄｈ１阻害剤 - Google Patents

血液学的悪性疾患および固形腫瘍の処置のためのｉｄｈ１阻害剤 Download PDF

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JP6856657B2
JP6856657B2 JP2018544835A JP2018544835A JP6856657B2 JP 6856657 B2 JP6856657 B2 JP 6856657B2 JP 2018544835 A JP2018544835 A JP 2018544835A JP 2018544835 A JP2018544835 A JP 2018544835A JP 6856657 B2 JP6856657 B2 JP 6856657B2
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compound
flt3
idh1
aml
mutant
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JP2019510746A (ja
JP2019510746A5 (enExample
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マイケル アマタンジェロ，
マイケル アマタンジェロ，
シャオラン フー，
シャオラン フー，
アンジャン タクルタ，
アンジャン タクルタ，
ソン ウン チェ，
ソン ウン チェ，
ビン ウー，
ビン ウー，
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Celgene Corp
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Celgene Corp
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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JP2018544835A 2016-02-26 2016-12-02 血液学的悪性疾患および固形腫瘍の処置のためのｉｄｈ１阻害剤 Expired - Fee Related JP6856657B2 (ja)

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JP2021044546A JP2021102630A (ja) 2016-02-26 2021-03-18 血液学的悪性疾患および固形腫瘍の処置のためのｉｄｈ１阻害剤

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US201662300673P 2016-02-26 2016-02-26
US62/300,673 2016-02-26
PCT/US2016/064845 WO2017146795A1 (en) 2016-02-26 2016-12-02 Idh1 inhibitors for the treatment of haematological malignancies and solid tumours

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JP2018544835A Expired - Fee Related JP6856657B2 (ja) 2016-02-26 2016-12-02 血液学的悪性疾患および固形腫瘍の処置のためのｉｄｈ１阻害剤
JP2018544781A Expired - Fee Related JP6930991B2 (ja) 2016-02-26 2016-12-02 血液学的悪性腫瘍及び固形腫瘍の治療のためのｉｄｈ２阻害剤
JP2021044546A Withdrawn JP2021102630A (ja) 2016-02-26 2021-03-18 血液学的悪性疾患および固形腫瘍の処置のためのｉｄｈ１阻害剤

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JP2021044546A Withdrawn JP2021102630A (ja) 2016-02-26 2021-03-18 血液学的悪性疾患および固形腫瘍の処置のためのｉｄｈ１阻害剤

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US (3) US10137130B2 (enExample)
EP (2) EP3419593B1 (enExample)
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KR (2) KR20180113540A (enExample)
CN (1) CN109069410B (enExample)
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CA (2) CA3015757A1 (enExample)
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