JP6589246B2 - イミダゾ［４，５‐ｃ］ピリジン由来のｓｓａｏ阻害剤 - Google Patents
イミダゾ［４，５‐ｃ］ピリジン由来のｓｓａｏ阻害剤 Download PDFInfo
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- JP6589246B2 JP6589246B2 JP2017515186A JP2017515186A JP6589246B2 JP 6589246 B2 JP6589246 B2 JP 6589246B2 JP 2017515186 A JP2017515186 A JP 2017515186A JP 2017515186 A JP2017515186 A JP 2017515186A JP 6589246 B2 JP6589246 B2 JP 6589246B2
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- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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| GBGB1416444.6A GB201416444D0 (en) | 2014-09-17 | 2014-09-17 | New compounds |
| GB1416444.6 | 2014-09-17 | ||
| PCT/GB2015/052691 WO2016042332A1 (en) | 2014-09-17 | 2015-09-17 | Imidazo[4,5-c]pyridine derived ssao inhibitors |
Publications (3)
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| JP2017532315A JP2017532315A (ja) | 2017-11-02 |
| JP2017532315A5 JP2017532315A5 (OSRAM) | 2019-08-15 |
| JP6589246B2 true JP6589246B2 (ja) | 2019-10-16 |
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| GB201304526D0 (en) * | 2013-03-13 | 2013-04-24 | Proximagen Ltd | New compounds |
| GB201416446D0 (en) * | 2014-09-17 | 2014-10-29 | Proximagen Ltd | New enzyme inhibitor compounds |
| WO2018027892A1 (en) | 2016-08-12 | 2018-02-15 | Eli Lilly And Company | Amino pyrimidine ssao inhibitors |
| WO2018148856A1 (en) | 2017-02-14 | 2018-08-23 | Eli Lilly And Company | Diazaspirodecanyl-pyrimidine compounds useful as ssao inhibitors |
| WO2022046779A1 (en) | 2020-08-25 | 2022-03-03 | Eli Lilly And Company | Polymorphs of an ssao inhibitor |
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| US6982286B2 (en) | 2001-07-12 | 2006-01-03 | Biotie Therapies Corp. | Carbocyclic hydrazino inhibitors of copper-containing amine oxidases |
| US20050096360A1 (en) | 2003-08-08 | 2005-05-05 | Salter-Cid Luisa M. | Inhibitors of semicarbazide-sensitive amine oxidase (SSAO) and VAP-1 mediated adhesion useful for treatment of diseases |
| JP2007504238A (ja) | 2003-09-04 | 2007-03-01 | アベンティス・ファーマスーティカルズ・インコーポレイテツド | ポリ（ａｄｐ−リボース）ポリメラーゼ（ｐａｒｐ）の阻害剤としての置換インドール |
| WO2007120528A2 (en) | 2006-03-31 | 2007-10-25 | La Jolla Pharmaceutical Company | Inhibitors of semicarbazide-sensitive amine oxidase (ssao) and vap-1 mediated adhesion useful for treatment and prevention of diseases |
| US7947723B2 (en) | 2008-02-01 | 2011-05-24 | Spelman College | Synthesis and anti-proliferative effect of benzimidazole derivatives |
| EP2328895B1 (en) * | 2008-09-16 | 2013-03-27 | Proximagen Limited | Pyrazolo[4,3-c]pyridine compounds and their use as inhibitors of SSAO |
| PT2334672E (pt) * | 2008-09-16 | 2014-01-02 | Proximagen Ltd | Compostos novos i |
| DK2376490T3 (da) | 2008-12-04 | 2013-04-15 | Proximagen Ltd | Imidazopyridinforbindelser |
| EP2417133A1 (en) | 2009-04-06 | 2012-02-15 | PTC Therapeutics, Inc. | Compounds and methods for antiviral treatment |
| GB201004311D0 (en) * | 2010-03-15 | 2010-04-28 | Proximagen Ltd | New enzyme inhibitor compounds |
| EP2518071A1 (en) * | 2011-04-29 | 2012-10-31 | Almirall, S.A. | Imidazopyridine derivatives as PI3K inhibitors |
| US9150574B2 (en) | 2011-09-14 | 2015-10-06 | Proximagen Limited | Enzyme inhibitor compounds |
| GB201115853D0 (en) | 2011-09-14 | 2011-10-26 | Proximagen Ltd | New enzyme inhibitor compounds |
| WO2013078254A1 (en) | 2011-11-22 | 2013-05-30 | Array Biopharma Inc. | Bicyclic heteroaryl derivatives as kinase inhibitors |
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| WO2015189534A1 (en) | 2014-06-12 | 2015-12-17 | Proximagen Limited | Vap-1 inhibitors for treating muscular dystrophy |
| GB201416446D0 (en) | 2014-09-17 | 2014-10-29 | Proximagen Ltd | New enzyme inhibitor compounds |
| CA3007768A1 (en) * | 2015-12-07 | 2017-06-15 | Benevolentai Cambridge Limited | Vap-1 inhibitors for treating pain |
| GB201709136D0 (en) * | 2017-06-08 | 2017-07-26 | Proximagen Ltd | New therapeutic uses of enzyme inhibitors |
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| AU2015316611A1 (en) | 2017-04-06 |
| GB201416444D0 (en) | 2014-10-29 |
| BR112017005324A2 (pt) | 2017-12-12 |
| US11530208B2 (en) | 2022-12-20 |
| ES2744548T3 (es) | 2020-02-25 |
| DK3194389T3 (da) | 2019-09-09 |
| AU2015316611B2 (en) | 2019-05-30 |
| US20170275281A1 (en) | 2017-09-28 |
| JP2017532315A (ja) | 2017-11-02 |
| EP3194389A1 (en) | 2017-07-26 |
| CA2961424A1 (en) | 2016-03-24 |
| IL251166B (en) | 2020-06-30 |
| PT3194389T (pt) | 2019-09-19 |
| HUE045827T2 (hu) | 2020-01-28 |
| WO2016042332A1 (en) | 2016-03-24 |
| PL3194389T3 (pl) | 2019-11-29 |
| CN107074853B (zh) | 2019-07-23 |
| IL251166A0 (en) | 2017-04-30 |
| EP3194389B1 (en) | 2019-08-07 |
| CN107074853A (zh) | 2017-08-18 |
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