JP6443332B2 - 固形製剤用のコーティング剤並びにこれから形成された被膜及び被覆固形製剤 - Google Patents
固形製剤用のコーティング剤並びにこれから形成された被膜及び被覆固形製剤 Download PDFInfo
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- JP6443332B2 JP6443332B2 JP2015516935A JP2015516935A JP6443332B2 JP 6443332 B2 JP6443332 B2 JP 6443332B2 JP 2015516935 A JP2015516935 A JP 2015516935A JP 2015516935 A JP2015516935 A JP 2015516935A JP 6443332 B2 JP6443332 B2 JP 6443332B2
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- 229960004949 glycyrrhizic acid Drugs 0.000 description 1
- UYRUBYNTXSDKQT-UHFFFAOYSA-N glycyrrhizic acid Natural products CC1(C)C(CCC2(C)C1CCC3(C)C2C(=O)C=C4C5CC(C)(CCC5(C)CCC34C)C(=O)O)OC6OC(C(O)C(O)C6OC7OC(O)C(O)C(O)C7C(=O)O)C(=O)O UYRUBYNTXSDKQT-UHFFFAOYSA-N 0.000 description 1
- 235000019410 glycyrrhizin Nutrition 0.000 description 1
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- WTFXARWRTYJXII-UHFFFAOYSA-N iron(2+);iron(3+);oxygen(2-) Chemical compound [O-2].[O-2].[O-2].[O-2].[Fe+2].[Fe+3].[Fe+3] WTFXARWRTYJXII-UHFFFAOYSA-N 0.000 description 1
- SZVJSHCCFOBDDC-UHFFFAOYSA-N iron(II,III) oxide Inorganic materials O=[Fe]O[Fe]O[Fe]=O SZVJSHCCFOBDDC-UHFFFAOYSA-N 0.000 description 1
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- CVHZOJJKTDOEJC-UHFFFAOYSA-N saccharin Chemical compound C1=CC=C2C(=O)NS(=O)(=O)C2=C1 CVHZOJJKTDOEJC-UHFFFAOYSA-N 0.000 description 1
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- 239000011734 sodium Substances 0.000 description 1
- AJPJDKMHJJGVTQ-UHFFFAOYSA-M sodium dihydrogen phosphate Chemical compound [Na+].OP(O)([O-])=O AJPJDKMHJJGVTQ-UHFFFAOYSA-M 0.000 description 1
- DVQHRBFGRZHMSR-UHFFFAOYSA-N sodium methyl 2,2-dimethyl-4,6-dioxo-5-(N-prop-2-enoxy-C-propylcarbonimidoyl)cyclohexane-1-carboxylate Chemical compound [Na+].C=CCON=C(CCC)[C-]1C(=O)CC(C)(C)C(C(=O)OC)C1=O DVQHRBFGRZHMSR-UHFFFAOYSA-N 0.000 description 1
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- 235000019408 sucralose Nutrition 0.000 description 1
- BAQAVOSOZGMPRM-QBMZZYIRSA-N sucralose Chemical compound O[C@@H]1[C@@H](O)[C@@H](Cl)[C@@H](CO)O[C@@H]1O[C@@]1(CCl)[C@@H](O)[C@H](O)[C@@H](CCl)O1 BAQAVOSOZGMPRM-QBMZZYIRSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2813—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/282—Organic compounds, e.g. fats
- A61K9/2826—Sugars or sugar alcohols, e.g. sucrose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Inorganic Chemistry (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014072607 | 2014-03-31 | ||
| JP2014072607 | 2014-03-31 | ||
| PCT/JP2015/060039 WO2015152195A1 (ja) | 2014-03-31 | 2015-03-31 | 固形製剤用のコーティング剤並びにこれから形成された被膜及び被覆固形製剤 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2015152195A1 JPWO2015152195A1 (ja) | 2017-04-13 |
| JP6443332B2 true JP6443332B2 (ja) | 2018-12-26 |
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| JP2015516935A Active JP6443332B2 (ja) | 2014-03-31 | 2015-03-31 | 固形製剤用のコーティング剤並びにこれから形成された被膜及び被覆固形製剤 |
Country Status (11)
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| PT3868366T (pt) * | 2018-10-19 | 2024-03-25 | Towa Pharmaceutical Co Ltd | Preparação sólida revestida |
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| JPS5157814A (en) * | 1974-11-14 | 1976-05-20 | Sumitomo Chemical Co | Tsuyanoyoitoijono seizohoho |
| US4780315A (en) * | 1985-11-25 | 1988-10-25 | Eastman Kodak Company | Rumen-stable pellets |
| JP2003125706A (ja) | 2001-10-23 | 2003-05-07 | Lion Corp | 口中清涼製剤 |
| JP2006506357A (ja) * | 2002-10-11 | 2006-02-23 | ヴェクトゥラ リミテッド | 有機高分子物質との組み合わせで無機粒子を含み、かつ固体の網目状マトリックスを形成する医薬賦形剤、その組成物、製造および使用 |
| WO2005019286A1 (ja) * | 2003-08-20 | 2005-03-03 | Shionogi & Co., Ltd. | 新規コーティング組成物 |
| CN101632648A (zh) * | 2008-07-23 | 2010-01-27 | Ss制药株式会社 | 薄膜包衣制剂 |
| NZ592765A (en) * | 2008-08-14 | 2013-06-28 | Bioneer As | Tablets with a coating which impedes the release of an active ingredient |
| TWI438012B (zh) * | 2008-12-25 | 2014-05-21 | Toray Industries | 固態製劑用之塗覆劑及使用其之固態製劑 |
| PL2412369T3 (pl) | 2009-03-27 | 2017-02-28 | Toray Industries, Inc. | Powlekany preparat stały |
| TWI455733B (zh) | 2009-03-30 | 2014-10-11 | Toray Industries | 口腔內崩壞性被覆錠劑 |
| JP2010248106A (ja) | 2009-04-14 | 2010-11-04 | Dainippon Sumitomo Pharma Co Ltd | フィルムコーティング錠 |
| PL2508206T3 (pl) | 2009-11-30 | 2014-12-31 | Toray Industries | Środek powlekający do preparatu stałego i stały preparat zawierający ten środek |
| HUE026633T2 (en) | 2010-02-26 | 2016-06-28 | Toray Industries | Covered solid preparation |
| HUE041795T2 (hu) * | 2010-08-31 | 2019-05-28 | Toray Industries | Bevonószer szilárd gyógyszerészeti készítményhez, gyógyszerészeti filmkészítmény, és bevonatos szilárd gyógyszerészeti készítmény |
| WO2012147873A1 (ja) | 2011-04-28 | 2012-11-01 | 持田製薬株式会社 | 口腔内崩壊性に優れたコーティング組成物 |
-
2015
- 2015-03-24 TW TW104109294A patent/TWI658842B/zh active
- 2015-03-31 WO PCT/JP2015/060039 patent/WO2015152195A1/ja active Application Filing
- 2015-03-31 CN CN201580018244.5A patent/CN106456779B/zh active Active
- 2015-03-31 MX MX2016012171A patent/MX365922B/es active IP Right Grant
- 2015-03-31 JP JP2015516935A patent/JP6443332B2/ja active Active
- 2015-03-31 BR BR112016021123-5A patent/BR112016021123B1/pt active IP Right Grant
- 2015-03-31 KR KR1020167016379A patent/KR102207440B1/ko active IP Right Grant
- 2015-03-31 US US15/129,153 patent/US10022331B2/en active Active
- 2015-03-31 CA CA2938394A patent/CA2938394C/en active Active
- 2015-03-31 EP EP15772255.4A patent/EP3127555B8/en active Active
- 2015-03-31 ES ES15772255T patent/ES2713160T3/es active Active
Also Published As
| Publication number | Publication date |
|---|---|
| TW201542244A (zh) | 2015-11-16 |
| CN106456779A (zh) | 2017-02-22 |
| KR102207440B1 (ko) | 2021-01-26 |
| BR112016021123A2 (US06650917-20031118-M00005.png) | 2017-08-15 |
| CN106456779B (zh) | 2019-07-19 |
| US10022331B2 (en) | 2018-07-17 |
| EP3127555A4 (en) | 2017-11-22 |
| US20170105940A1 (en) | 2017-04-20 |
| WO2015152195A1 (ja) | 2015-10-08 |
| EP3127555B8 (en) | 2020-03-04 |
| CA2938394A1 (en) | 2015-10-08 |
| TWI658842B (zh) | 2019-05-11 |
| JPWO2015152195A1 (ja) | 2017-04-13 |
| MX2016012171A (es) | 2017-01-05 |
| EP3127555A1 (en) | 2017-02-08 |
| ES2713160T9 (es) | 2020-04-20 |
| EP3127555B1 (en) | 2018-12-12 |
| ES2713160T3 (es) | 2019-05-20 |
| KR20160137507A (ko) | 2016-11-30 |
| BR112016021123B1 (pt) | 2022-06-14 |
| MX365922B (es) | 2019-06-20 |
| CA2938394C (en) | 2022-03-29 |
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