JP6130398B2 - 新規アゼチジン誘導体、その医薬組成物及び使用 - Google Patents

新規アゼチジン誘導体、その医薬組成物及び使用 Download PDF

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JP6130398B2
JP6130398B2 JP2014549478A JP2014549478A JP6130398B2 JP 6130398 B2 JP6130398 B2 JP 6130398B2 JP 2014549478 A JP2014549478 A JP 2014549478A JP 2014549478 A JP2014549478 A JP 2014549478A JP 6130398 B2 JP6130398 B2 JP 6130398B2
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alkyl
group
cycloalkyl
heterocyclyl
phenyl
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JP2015503540A (ja
JP2015503540A5 (enExample
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ベルント ノッセ
ベルント ノッセ
マルティン フレック
マルティン フレック
ゲラルト ユルゲン ロート
ゲラルト ユルゲン ロート
ニクラス ハイネ
ニクラス ハイネ
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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JP2014549478A 2011-12-29 2012-12-28 新規アゼチジン誘導体、その医薬組成物及び使用 Expired - Fee Related JP6130398B2 (ja)

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EP11196046 2011-12-29
EP11196046.4 2011-12-29
PCT/EP2012/077025 WO2013098373A1 (en) 2011-12-29 2012-12-28 New azetidine derivatives, pharmaceutical compositions and uses thereof

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JP2015503540A JP2015503540A (ja) 2015-02-02
JP2015503540A5 JP2015503540A5 (enExample) 2016-02-18
JP6130398B2 true JP6130398B2 (ja) 2017-05-17

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MX2016002479A (es) * 2013-09-12 2016-05-31 Pfizer Uso de inhibidores de acetil-coa carboxilasa para tratar acne vulgaris.
EP3059225A4 (en) 2013-10-17 2017-09-06 Shionogi & Co., Ltd. Novel alkylene derivative
WO2015096651A1 (en) 2013-12-23 2015-07-02 Merck Sharp & Dohme Corp. Pyrimidone carboxamide compounds as pde2 inhibitors
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WO2016145614A1 (en) 2015-03-17 2016-09-22 Merck Sharp & Dohme Corp. Triazolyl pyrimidinone compounds as pde2 inhibitors
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