JP5925809B2 - 三環系ピロロ誘導体、その調製方法およびそのキナーゼ阻害剤としての使用 - Google Patents

三環系ピロロ誘導体、その調製方法およびそのキナーゼ阻害剤としての使用 Download PDF

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JP5925809B2
JP5925809B2 JP2013550833A JP2013550833A JP5925809B2 JP 5925809 B2 JP5925809 B2 JP 5925809B2 JP 2013550833 A JP2013550833 A JP 2013550833A JP 2013550833 A JP2013550833 A JP 2013550833A JP 5925809 B2 JP5925809 B2 JP 5925809B2
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formula
compound
methyl
pyrrolo
quinazoline
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JP2014503567A (ja
JP2014503567A5 (enExample
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カルダレツリ，マリーナ
アンジヨリニ，マウロ
ベリア，イタロ
ブラスカ，マリア・ガブリエツラ
カスシエツリ，フランチエスコ
ダレツシオ，ロベルト
ロンバルデイ・ボルジア，アンドレア
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ネルビアーノ・メデイカル・サイエンシーズ・エツセ・エルレ・エルレ
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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JP2013550833A 2011-01-26 2012-01-19 三環系ピロロ誘導体、その調製方法およびそのキナーゼ阻害剤としての使用 Active JP5925809B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11152190 2011-01-26
EP11152190.2 2011-01-26
PCT/EP2012/050773 WO2012101032A1 (en) 2011-01-26 2012-01-19 Tricyclic pyrrolo derivatives, process for their preparation and their use as kinase inhibitors

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JP2015203440A Division JP6118383B2 (ja) 2011-01-26 2015-10-15 三環系ピロロ誘導体、その調製方法およびそのキナーゼ阻害剤としての使用

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JP2014503567A JP2014503567A (ja) 2014-02-13
JP2014503567A5 JP2014503567A5 (enExample) 2015-03-05
JP5925809B2 true JP5925809B2 (ja) 2016-05-25

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JP2015203440A Active JP6118383B2 (ja) 2011-01-26 2015-10-15 三環系ピロロ誘導体、その調製方法およびそのキナーゼ阻害剤としての使用

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US (2) US8975267B2 (enExample)
EP (1) EP2668190B1 (enExample)
JP (2) JP5925809B2 (enExample)
CN (1) CN103339134B (enExample)
BR (1) BR112013018515B1 (enExample)
ES (1) ES2602791T3 (enExample)
RU (1) RU2591191C2 (enExample)
WO (1) WO2012101032A1 (enExample)

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RU2013139353A (ru) 2015-03-10
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US20150141408A1 (en) 2015-05-21
US8975267B2 (en) 2015-03-10
EP2668190B1 (en) 2016-08-17
CN103339134B (zh) 2015-12-23
HK1189229A1 (zh) 2014-05-30
JP6118383B2 (ja) 2017-04-19
US20130296305A1 (en) 2013-11-07
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