JP5886285B2 - Ｃｌｏｓｔｒｉｄｉｕｍ属に対する抗菌活性を有する化合物 - Google Patents
Ｃｌｏｓｔｒｉｄｉｕｍ属に対する抗菌活性を有する化合物 Download PDFInfo
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- JP5886285B2 JP5886285B2 JP2013522249A JP2013522249A JP5886285B2 JP 5886285 B2 JP5886285 B2 JP 5886285B2 JP 2013522249 A JP2013522249 A JP 2013522249A JP 2013522249 A JP2013522249 A JP 2013522249A JP 5886285 B2 JP5886285 B2 JP 5886285B2
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10171842 | 2010-08-04 | ||
| EP10171842.7 | 2010-08-04 | ||
| PCT/EP2011/063434 WO2012017030A1 (en) | 2010-08-04 | 2011-08-04 | Compounds with antibacterial activity against clostridium |
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| Publication Number | Publication Date |
|---|---|
| JP2013532714A JP2013532714A (ja) | 2013-08-19 |
| JP2013532714A5 JP2013532714A5 (enExample) | 2014-09-04 |
| JP5886285B2 true JP5886285B2 (ja) | 2016-03-16 |
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| EP (1) | EP2601193B1 (enExample) |
| JP (1) | JP5886285B2 (enExample) |
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| BR (1) | BR112013003675A8 (enExample) |
| CA (1) | CA2805358C (enExample) |
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| CO (1) | CO6680629A2 (enExample) |
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| ES (1) | ES2538998T3 (enExample) |
| HR (1) | HRP20150467T1 (enExample) |
| ME (1) | ME02061B (enExample) |
| MX (1) | MX2013001246A (enExample) |
| NZ (1) | NZ605850A (enExample) |
| PH (1) | PH12013500219A1 (enExample) |
| PL (1) | PL2601193T3 (enExample) |
| PT (1) | PT2601193E (enExample) |
| RS (1) | RS53990B1 (enExample) |
| SG (1) | SG187175A1 (enExample) |
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| TW (1) | TWI498330B (enExample) |
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Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9079935B2 (en) | 2012-08-13 | 2015-07-14 | The Board Of Regents Of The Nevada System Of Higher Education On Behalf Of The University Of Nevada, Las Vegas | Reducing risk of contracting Clostridium-difficile associated disease |
| WO2016127102A2 (en) | 2015-02-06 | 2016-08-11 | Ernesto Abel-Santos | Inhibiting germination of clostridium perfringens spores to reduce necrotic enteritis |
| GB201509326D0 (en) | 2015-05-29 | 2015-07-15 | Antibio Tx Aps | Novel use |
| KR101769204B1 (ko) * | 2015-08-04 | 2017-08-17 | 씨제이헬스케어 주식회사 | 크로마놀 유도체의 신규한 제조방법 |
| WO2023039159A2 (en) | 2021-09-09 | 2023-03-16 | Abel Santos Ernesto | Inhibitors of c. difficile spore germination |
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| EP2094714B1 (en) * | 2006-09-26 | 2012-08-15 | Crestone, Inc. | Substituted thienopyridone compounds with antibacterial activity |
| EP2091536B1 (en) * | 2006-09-26 | 2013-07-31 | Crestone, Inc. | Enantiomeric compounds with antibacterial activity |
| US8658670B2 (en) * | 2006-09-26 | 2014-02-25 | Crestone, Inc. | Methods and compounds for treatment of clostridium based infection |
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2011
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- 2011-08-04 SI SI201130439T patent/SI2601193T1/sl unknown
- 2011-08-04 ES ES11740921.9T patent/ES2538998T3/es active Active
- 2011-08-04 AU AU2011287584A patent/AU2011287584B2/en not_active Ceased
- 2011-08-04 DK DK11740921.9T patent/DK2601193T3/en active
- 2011-08-04 MX MX2013001246A patent/MX2013001246A/es not_active Application Discontinuation
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