JP5818801B2 - 改善された製剤 - Google Patents

改善された製剤 Download PDF

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Publication number
JP5818801B2
JP5818801B2 JP2012533648A JP2012533648A JP5818801B2 JP 5818801 B2 JP5818801 B2 JP 5818801B2 JP 2012533648 A JP2012533648 A JP 2012533648A JP 2012533648 A JP2012533648 A JP 2012533648A JP 5818801 B2 JP5818801 B2 JP 5818801B2
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JP
Japan
Prior art keywords
aerosol formulation
suspension aerosol
fluticasone propionate
micrograms
formoterol fumarate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
JP2012533648A
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English (en)
Japanese (ja)
Other versions
JP2013507429A (ja
JP2013507429A5 (enExample
Inventor
ミュラーウォルツ ルディー
ミュラーウォルツ ルディー
フュエーク リーゼ−マリー
フュエーク リーゼ−マリー
Original Assignee
ヤゴテック アーゲー
ヤゴテック アーゲー
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41462451&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP5818801(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by ヤゴテック アーゲー, ヤゴテック アーゲー filed Critical ヤゴテック アーゲー
Publication of JP2013507429A publication Critical patent/JP2013507429A/ja
Publication of JP2013507429A5 publication Critical patent/JP2013507429A5/ja
Application granted granted Critical
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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/008—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2012533648A 2009-10-16 2010-10-15 改善された製剤 Active JP5818801B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0918150.4 2009-10-16
GBGB0918150.4A GB0918150D0 (en) 2009-10-16 2009-10-16 Improved formulations
PCT/EP2010/065569 WO2011045429A1 (en) 2009-10-16 2010-10-15 Improved formulations

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2015191177A Division JP2016040286A (ja) 2009-10-16 2015-09-29 改善された製剤

Publications (3)

Publication Number Publication Date
JP2013507429A JP2013507429A (ja) 2013-03-04
JP2013507429A5 JP2013507429A5 (enExample) 2015-05-21
JP5818801B2 true JP5818801B2 (ja) 2015-11-18

Family

ID=41462451

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2012533648A Active JP5818801B2 (ja) 2009-10-16 2010-10-15 改善された製剤
JP2015191177A Pending JP2016040286A (ja) 2009-10-16 2015-09-29 改善された製剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2015191177A Pending JP2016040286A (ja) 2009-10-16 2015-09-29 改善された製剤

Country Status (25)

Country Link
US (2) US20120263766A1 (enExample)
EP (2) EP2488157B1 (enExample)
JP (2) JP5818801B2 (enExample)
CN (1) CN102573791B (enExample)
AU (1) AU2010305695B2 (enExample)
BR (1) BR112012008969B1 (enExample)
CA (1) CA2776845C (enExample)
CL (1) CL2012000948A1 (enExample)
CY (1) CY1123918T1 (enExample)
DK (1) DK2488157T3 (enExample)
ES (1) ES2859629T3 (enExample)
GB (1) GB0918150D0 (enExample)
HR (1) HRP20210379T1 (enExample)
HU (1) HUE054030T2 (enExample)
IL (2) IL219162A0 (enExample)
LT (1) LT2488157T (enExample)
MX (1) MX372991B (enExample)
NZ (1) NZ599900A (enExample)
PL (1) PL2488157T3 (enExample)
PT (1) PT2488157T (enExample)
RS (1) RS61430B1 (enExample)
SI (1) SI2488157T1 (enExample)
SM (1) SMT202100150T1 (enExample)
WO (1) WO2011045429A1 (enExample)
ZA (1) ZA201202595B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016040286A (ja) * 2009-10-16 2016-03-24 ヤゴテック アーゲー 改善された製剤

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100496608C (zh) * 2001-03-30 2009-06-10 洁垢技术有限公司 药用气溶胶制剂
GB0323684D0 (en) 2003-10-09 2003-11-12 Jagotec Ag Improvements in or relating to organic compounds
GB0918149D0 (en) * 2009-10-16 2009-12-02 Jagotec Ag Improved medicinal aerosol formulation
WO2013127738A1 (de) * 2012-02-28 2013-09-06 Boehringer Ingelheim International Gmbh Neue treibgashaltige tiotropium-formulierung
RU2678992C2 (ru) 2012-04-11 2019-02-05 Сипла Лимитед Фармацевтическая композиция, содержащая арформотерол и флутиказона фуроат
GB201321712D0 (en) * 2013-12-09 2014-01-22 Pharmachemie Bv Dry Powder Inhaler
CN105963282B (zh) * 2016-05-04 2019-04-19 四川普锐特医药科技有限责任公司 一种医用定量吸入气雾剂
WO2018059390A1 (zh) * 2016-09-29 2018-04-05 广东东阳光药业有限公司 药物组合物

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6596260B1 (en) 1993-08-27 2003-07-22 Novartis Corporation Aerosol container and a method for storage and administration of a predetermined amount of a pharmaceutically active aerosol
EP1366777B1 (en) 1995-04-14 2005-06-15 SmithKline Beecham Corporation Metered dose inhaler for salmeterol
DE69622166T2 (de) 1995-04-14 2003-04-03 Smithkline Beecham Corp., Philadelphia Dosierinhalator für albuterol
JPH101442A (ja) * 1996-06-12 1998-01-06 Taisho Pharmaceut Co Ltd 鼻炎用点鼻薬
EP1393721B1 (en) * 1997-03-20 2008-11-26 Schering Corporation Dosage form of powder agglomerates
GB9903759D0 (en) * 1999-02-18 1999-04-14 Novartis Ag Organic compounds
EE05167B1 (et) * 2000-05-22 2009-06-15 Chiesi Farmaceutici S.P.A. Stabiilsed farmatseutilised lahuspreparaadid survestatud doseerivatele inhalaatoritele
US20060257324A1 (en) * 2000-05-22 2006-11-16 Chiesi Farmaceutici S.P.A. Pharmaceutical solution formulations for pressurised metered dose inhalers
AU2001289126A1 (en) 2000-09-18 2002-04-02 Glaxo Group Limited Metered dose inhaler can coated two or more times with fluorocarbon polymers
CN1635870A (zh) * 2000-10-09 2005-07-06 3M创新有限公司 药用气雾剂制剂
CN100496608C (zh) * 2001-03-30 2009-06-10 洁垢技术有限公司 药用气溶胶制剂
US6667344B2 (en) * 2001-04-17 2003-12-23 Dey, L.P. Bronchodilating compositions and methods
GB0201400D0 (en) * 2002-01-22 2002-03-13 Glaxo Group Ltd Novel apparatus and process
EP1531866A1 (en) * 2002-08-29 2005-05-25 Cipla Ltd. Pharmaceutical products and compositions comprising specific anticholinergic agents, beta-2 agonists and corticosteroids
GB0323684D0 (en) * 2003-10-09 2003-11-12 Jagotec Ag Improvements in or relating to organic compounds
GB0327727D0 (en) * 2003-11-28 2003-12-31 Quadrant Drug Delivery Ltd Viral microparticles
GB0410399D0 (en) * 2004-05-10 2004-06-16 Arakis Ltd The treatment of respiratory disease
GB0918150D0 (en) * 2009-10-16 2009-12-02 Jagotec Ag Improved formulations

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016040286A (ja) * 2009-10-16 2016-03-24 ヤゴテック アーゲー 改善された製剤

Also Published As

Publication number Publication date
PL2488157T3 (pl) 2021-06-28
CA2776845C (en) 2018-04-24
MX372991B (es) 2020-06-18
ES2859629T3 (es) 2021-10-04
NZ599900A (en) 2014-11-28
CN102573791B (zh) 2017-09-22
RS61430B1 (sr) 2021-03-31
GB0918150D0 (en) 2009-12-02
IL219162A0 (en) 2012-06-28
DK2488157T3 (da) 2021-01-25
HUE054030T2 (hu) 2021-08-30
US20180296468A2 (en) 2018-10-18
JP2016040286A (ja) 2016-03-24
CN102573791A (zh) 2012-07-11
CL2012000948A1 (es) 2012-12-14
BR112012008969B1 (pt) 2021-07-06
MX2012004338A (es) 2012-08-01
PT2488157T (pt) 2021-02-05
ZA201202595B (en) 2023-07-26
JP2013507429A (ja) 2013-03-04
CA2776845A1 (en) 2011-04-21
WO2011045429A1 (en) 2011-04-21
US20170281529A1 (en) 2017-10-05
SI2488157T1 (sl) 2021-02-26
EP2488157B1 (en) 2020-12-30
SMT202100150T1 (it) 2021-05-07
EP2488157A1 (en) 2012-08-22
US20120263766A1 (en) 2012-10-18
AU2010305695A1 (en) 2012-05-03
AU2010305695B2 (en) 2014-07-10
LT2488157T (lt) 2021-02-10
IL269369A (en) 2019-11-28
CY1123918T1 (el) 2022-05-27
BR112012008969A2 (pt) 2020-06-23
HRP20210379T1 (hr) 2021-04-16
EP3811928A1 (en) 2021-04-28

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