JP5693951B2 - プロテインキナーゼの阻害剤 - Google Patents

プロテインキナーゼの阻害剤 Download PDF

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JP5693951B2
JP5693951B2 JP2010504681A JP2010504681A JP5693951B2 JP 5693951 B2 JP5693951 B2 JP 5693951B2 JP 2010504681 A JP2010504681 A JP 2010504681A JP 2010504681 A JP2010504681 A JP 2010504681A JP 5693951 B2 JP5693951 B2 JP 5693951B2
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alkyl
phenyl
compound
pain
methoxy
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JP2011502956A (ja
JP2011502956A5 (OSRAM
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ワブニトズ プヒリププ
ワブニトズ プヒリププ
スチャウエルテ ヘイケ
スチャウエルテ ヘイケ
アルルゲイエル ハンス
アルルゲイエル ハンス
アウグストイン マルトイン
アウグストイン マルトイン
ゼイトルマンン ルトズ
ゼイトルマンン ルトズ
エー.プレイスス ミチャエル
エー.プレイスス ミチャエル
ストウムム ガブリエレ
ストウムム ガブリエレ
ムエルレル アンケ
ムエルレル アンケ
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アストラゼネカ エービー
アストラゼネカ エービー
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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
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JP2010504681A 2007-04-24 2008-04-24 プロテインキナーゼの阻害剤 Expired - Fee Related JP5693951B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EPPCT/EP2007/003602 2007-04-24
EP2007003602 2007-04-24
PCT/EP2008/054975 WO2008129070A1 (en) 2007-04-24 2008-04-24 Inhibitors of protein kinases

Publications (3)

Publication Number Publication Date
JP2011502956A JP2011502956A (ja) 2011-01-27
JP2011502956A5 JP2011502956A5 (OSRAM) 2011-06-16
JP5693951B2 true JP5693951B2 (ja) 2015-04-01

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JP2010504681A Expired - Fee Related JP5693951B2 (ja) 2007-04-24 2008-04-24 プロテインキナーゼの阻害剤

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US (1) US8436007B2 (OSRAM)
JP (1) JP5693951B2 (OSRAM)
ES (1) ES2539518T3 (OSRAM)
WO (1) WO2008129070A1 (OSRAM)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2137166B1 (en) * 2007-04-24 2012-05-30 Ingenium Pharmaceuticals GmbH 4, 6-disubstituted aminopyrimidine derivatives as inhibitors of protein kinases
WO2008129069A1 (en) * 2007-04-24 2008-10-30 Ingenium Pharmaceuticals Gmbh Inhibitors of protein kinases
ES2539518T3 (es) 2007-04-24 2015-07-01 Astrazeneca Ab Inhibidores de proteínas quinasas
CN102481327B (zh) 2009-07-08 2015-01-28 乔本生医股份有限公司 一种龙眼核萃取物的制备方法与应用
JP2013107824A (ja) * 2010-03-17 2013-06-06 Dainippon Sumitomo Pharma Co Ltd 新規単環ピリミジン誘導体
EA026917B1 (ru) * 2010-03-22 2017-05-31 Лид Дискавери Сентр Гмбх Фармацевтически активные производные двузамещенного триазина
WO2012066065A1 (en) * 2010-11-17 2012-05-24 Novartis Ag Phenyl-heteroaryl amine compounds and their uses
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