ES2539518T3 - Inhibidores de proteínas quinasas - Google Patents

Inhibidores de proteínas quinasas Download PDF

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Publication number
ES2539518T3
ES2539518T3 ES08736527.6T ES08736527T ES2539518T3 ES 2539518 T3 ES2539518 T3 ES 2539518T3 ES 08736527 T ES08736527 T ES 08736527T ES 2539518 T3 ES2539518 T3 ES 2539518T3
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Prior art keywords
4alkyl
phenyl
diseases
pain
alkyl
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ES08736527.6T
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English (en)
Spanish (es)
Inventor
Philipp Wabnitz
Heike Schauerte
Hans Allgeier
Martin Augustin
Lutz Zeitlmann
Michael A. Pleiss
Gabriele Stumm
Anke Mueller
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AstraZeneca AB
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AstraZeneca AB
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
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  • Organic Chemistry (AREA)
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  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Vascular Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
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ES08736527.6T 2007-04-24 2008-04-24 Inhibidores de proteínas quinasas Active ES2539518T3 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP2007003602 2007-04-24
WOPCT/EP2007/003602 2007-04-24
PCT/EP2008/054975 WO2008129070A1 (en) 2007-04-24 2008-04-24 Inhibitors of protein kinases

Publications (1)

Publication Number Publication Date
ES2539518T3 true ES2539518T3 (es) 2015-07-01

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ID=39588050

Family Applications (1)

Application Number Title Priority Date Filing Date
ES08736527.6T Active ES2539518T3 (es) 2007-04-24 2008-04-24 Inhibidores de proteínas quinasas

Country Status (4)

Country Link
US (1) US8436007B2 (OSRAM)
JP (1) JP5693951B2 (OSRAM)
ES (1) ES2539518T3 (OSRAM)
WO (1) WO2008129070A1 (OSRAM)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2137166B1 (en) * 2007-04-24 2012-05-30 Ingenium Pharmaceuticals GmbH 4, 6-disubstituted aminopyrimidine derivatives as inhibitors of protein kinases
WO2008129069A1 (en) * 2007-04-24 2008-10-30 Ingenium Pharmaceuticals Gmbh Inhibitors of protein kinases
ES2539518T3 (es) 2007-04-24 2015-07-01 Astrazeneca Ab Inhibidores de proteínas quinasas
CN102481327B (zh) 2009-07-08 2015-01-28 乔本生医股份有限公司 一种龙眼核萃取物的制备方法与应用
JP2013107824A (ja) * 2010-03-17 2013-06-06 Dainippon Sumitomo Pharma Co Ltd 新規単環ピリミジン誘導体
EA026917B1 (ru) * 2010-03-22 2017-05-31 Лид Дискавери Сентр Гмбх Фармацевтически активные производные двузамещенного триазина
WO2012066065A1 (en) * 2010-11-17 2012-05-24 Novartis Ag Phenyl-heteroaryl amine compounds and their uses
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