JP5531370B2 - プロスタグランジンd2受容体のアンタゴニスト - Google Patents

プロスタグランジンd2受容体のアンタゴニスト Download PDF

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JP5531370B2
JP5531370B2 JP2011516892A JP2011516892A JP5531370B2 JP 5531370 B2 JP5531370 B2 JP 5531370B2 JP 2011516892 A JP2011516892 A JP 2011516892A JP 2011516892 A JP2011516892 A JP 2011516892A JP 5531370 B2 JP5531370 B2 JP 5531370B2
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phenyl
compound
phenoxy
acetic acid
methoxy
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JP2011526930A (ja
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ジョン ハワード ハッチンソン
トーマス ジョン サイダース
ボウェイ ワン
ジーニー エム. アルダ
ブライアン アンドリュー スターンズ
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パンミラ ファーマシューティカルズ,エルエルシー.
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • C07C317/28Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
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    • C07D263/18Oxygen atoms
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  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Hydrogenated Pyridines (AREA)
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JP2011516892A 2008-07-03 2009-07-02 プロスタグランジンd2受容体のアンタゴニスト Expired - Fee Related JP5531370B2 (ja)

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US7831108P 2008-07-03 2008-07-03
US61/078,311 2008-07-03
PCT/US2009/049621 WO2010003120A2 (en) 2008-07-03 2009-07-02 Antagonists of prostaglandin d2 receptors

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JP2011526930A JP2011526930A (ja) 2011-10-20
JP2011526930A5 JP2011526930A5 (https=) 2012-08-16
JP5531370B2 true JP5531370B2 (ja) 2014-06-25

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