JP5530923B2 - ホウ素含有小分子 - Google Patents

ホウ素含有小分子 Download PDF

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Publication number
JP5530923B2
JP5530923B2 JP2010513416A JP2010513416A JP5530923B2 JP 5530923 B2 JP5530923 B2 JP 5530923B2 JP 2010513416 A JP2010513416 A JP 2010513416A JP 2010513416 A JP2010513416 A JP 2010513416A JP 5530923 B2 JP5530923 B2 JP 5530923B2
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exemplary embodiment
substituted
compound
unsubstituted
salt
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Japanese (ja)
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JP2010530881A (ja
JP2010530881A5 (enExample
Inventor
ベイカー，スティーブン，ジェイ．
ヘルナンデス，ビンセント，エス
シャーマ，ラシュミ
ニエマン，ジェームス，エー．
勉 赤間
チャン，ヨン−カン
ジェイ． プラットナー，ジェイコブ
アリー，マイケル，リチャード，ケビン
シン，ラジェシャワー
シャ，イ
ジョウ，フチェン
モハマッド，ラヒム
メーディ ケラマネ，エル
ルー，シャオソン
ハ，ミン
フィリップス，ジェームス，ジー．
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アナコール ファーマシューティカルズ，インコーポレイテッド
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Application filed by アナコール ファーマシューティカルズ，インコーポレイテッド filed Critical アナコール ファーマシューティカルズ，インコーポレイテッド
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Publication of JP2010530881A5 publication Critical patent/JP2010530881A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/02—Local antiseptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2010513416A 2007-06-20 2008-06-19 ホウ素含有小分子 Active JP5530923B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US94529407P 2007-06-20 2007-06-20
US60/945,294 2007-06-20
US4117808P 2008-03-31 2008-03-31
US61/041,178 2008-03-31
PCT/US2008/067550 WO2008157726A1 (en) 2007-06-20 2008-06-19 Boron-containing small molecules

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014087397A Division JP2014148531A (ja) 2007-06-20 2014-04-21 ホウ素含有小分子

Publications (3)

Publication Number Publication Date
JP2010530881A JP2010530881A (ja) 2010-09-16
JP2010530881A5 JP2010530881A5 (enExample) 2011-08-04
JP5530923B2 true JP5530923B2 (ja) 2014-06-25

Family

ID=40156702

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2010513416A Active JP5530923B2 (ja) 2007-06-20 2008-06-19 ホウ素含有小分子
JP2014087397A Pending JP2014148531A (ja) 2007-06-20 2014-04-21 ホウ素含有小分子
JP2015187239A Active JP6570391B2 (ja) 2007-06-20 2015-09-24 ホウ素含有小分子

Family Applications After (2)

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JP2014087397A Pending JP2014148531A (ja) 2007-06-20 2014-04-21 ホウ素含有小分子
JP2015187239A Active JP6570391B2 (ja) 2007-06-20 2015-09-24 ホウ素含有小分子

Country Status (29)

Country Link
US (4) US7816344B2 (enExample)
EP (1) EP2164331B1 (enExample)
JP (3) JP5530923B2 (enExample)
KR (3) KR101578351B1 (enExample)
CN (2) CN101772302B (enExample)
AR (1) AR067105A1 (enExample)
AU (1) AU2008265630B2 (enExample)
BR (1) BRPI0813450B8 (enExample)
CA (1) CA2692135C (enExample)
CL (1) CL2008001855A1 (enExample)
CO (1) CO6251209A2 (enExample)
CR (1) CR11224A (enExample)
DK (1) DK2164331T3 (enExample)
DO (1) DOP2009000281A (enExample)
EA (1) EA020530B1 (enExample)
ES (1) ES2655299T3 (enExample)
IL (1) IL202379A (enExample)
JO (1) JO3396B1 (enExample)
MA (1) MA31675B1 (enExample)
MX (1) MX347688B (enExample)
MY (1) MY162692A (enExample)
NO (1) NO2164331T3 (enExample)
NZ (1) NZ582706A (enExample)
PE (1) PE20090840A1 (enExample)
SG (1) SG182219A1 (enExample)
TW (1) TW200911822A (enExample)
UY (1) UY31171A1 (enExample)
WO (1) WO2008157726A1 (enExample)
ZA (2) ZA200909003B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
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JP2014148531A (ja) * 2007-06-20 2014-08-21 Anacor Pharmaceuticals Inc ホウ素含有小分子

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US8668911B2 (en) * 2009-05-14 2014-03-11 The Regents Of The University Of Michigan Streptococcus vaccine compositions and methods of using the same
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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2014148531A (ja) * 2007-06-20 2014-08-21 Anacor Pharmaceuticals Inc ホウ素含有小分子
JP2016040275A (ja) * 2007-06-20 2016-03-24 アナコール ファーマシューティカルズ，インコーポレイテッド ホウ素含有小分子

Also Published As

Publication number Publication date
DK2164331T3 (da) 2018-01-29
KR20100051615A (ko) 2010-05-17
BRPI0813450B1 (pt) 2019-05-07
UY31171A1 (es) 2009-04-30
WO2008157726A1 (en) 2008-12-24
BRPI0813450B8 (pt) 2021-05-25
US8895534B2 (en) 2014-11-25
EA200901617A1 (ru) 2010-06-30
CR11224A (es) 2010-06-28
EP2164331A4 (en) 2011-09-07
EA020530B1 (ru) 2014-11-28
CO6251209A2 (es) 2011-02-21
KR20160049025A (ko) 2016-05-04
US20090227541A1 (en) 2009-09-10
MY162692A (en) 2017-07-14
SG182219A1 (en) 2012-07-30
IL202379A (en) 2016-02-29
JP2016040275A (ja) 2016-03-24
KR20150100945A (ko) 2015-09-02
EP2164331A1 (en) 2010-03-24
DOP2009000281A (es) 2010-07-31
JP2014148531A (ja) 2014-08-21
BRPI0813450A2 (pt) 2014-12-30
AU2008265630B2 (en) 2013-06-20
CN104017008A (zh) 2014-09-03
ES2655299T3 (es) 2018-02-19
KR101685656B1 (ko) 2016-12-12
CA2692135C (en) 2017-01-24
CA2692135A1 (en) 2008-12-24
ZA201104573B (en) 2014-03-26
US10533021B2 (en) 2020-01-14
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US20150133402A1 (en) 2015-05-14
JP2010530881A (ja) 2010-09-16
CL2008001855A1 (es) 2009-05-29
AR067105A1 (es) 2009-09-30
MX347688B (es) 2017-05-09
ZA200909003B (en) 2022-03-30
NO2164331T3 (enExample) 2018-04-28
EP2164331B1 (en) 2017-11-29
AU2008265630A1 (en) 2008-12-24
IL202379A0 (en) 2010-06-30
MA31675B1 (fr) 2010-09-01
US20100292504A1 (en) 2010-11-18
JO3396B1 (ar) 2019-10-20
CN101772302B (zh) 2014-05-07
TW200911822A (en) 2009-03-16
US7816344B2 (en) 2010-10-19
KR101578351B1 (ko) 2015-12-17
US9796735B2 (en) 2017-10-24
CN101772302A (zh) 2010-07-07
PE20090840A1 (es) 2009-07-08
US20180016285A1 (en) 2018-01-18
JP6570391B2 (ja) 2019-09-04

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