JP4928949B2 - タンパク質キナーゼモジュレーターとしてのピラゾール誘導体 - Google Patents

タンパク質キナーゼモジュレーターとしてのピラゾール誘導体 Download PDF

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JP4928949B2
JP4928949B2 JP2006546339A JP2006546339A JP4928949B2 JP 4928949 B2 JP4928949 B2 JP 4928949B2 JP 2006546339 A JP2006546339 A JP 2006546339A JP 2006546339 A JP2006546339 A JP 2006546339A JP 4928949 B2 JP4928949 B2 JP 4928949B2
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Japan
Prior art keywords
phenyl
pyrazol
chloro
group
methyl
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Expired - Fee Related
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JP2006546339A
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Japanese (ja)
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JP2007516272A (ja
JP2007516272A5 (https=
Inventor
バレリオ、ベルディーニ
ゴードン、サクスティー
マリヌス、レーンデルト、フェルドンク
スティーブン、ジョン、ウッドヘッド
ポール、グラハム、ワイアット
ロバート、ジョージ、ボイル
ハンナ、フィオナ、ソアー
デイビッド、ウィンター、ウォーカー
イアン、コリンズ
ロバート、ダウンハム
ロビン、アーサー、エリス、カー
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Cancer Research Technology Ltd
Astex Therapeutics Ltd
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Cancer Research Technology Ltd
Astex Therapeutics Ltd
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Priority claimed from GB0329617A external-priority patent/GB0329617D0/en
Application filed by Cancer Research Technology Ltd, Astex Therapeutics Ltd filed Critical Cancer Research Technology Ltd
Publication of JP2007516272A publication Critical patent/JP2007516272A/ja
Publication of JP2007516272A5 publication Critical patent/JP2007516272A5/ja
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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US8691806B2 (en) 2014-04-08
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