JP4633462B2 - ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法 - Google Patents

３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法 Download PDF

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Publication number
JP4633462B2
JP4633462B2 JP2004524203A JP2004524203A JP4633462B2 JP 4633462 B2 JP4633462 B2 JP 4633462B2 JP 2004524203 A JP2004524203 A JP 2004524203A JP 2004524203 A JP2004524203 A JP 2004524203A JP 4633462 B2 JP4633462 B2 JP 4633462B2
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Japan
Prior art keywords
formula
alkyl
compound
halogen
dihydro
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Japanese (ja)
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JP2005534685A5 (enExample
JP2005534685A (ja
Inventor
アニス，ゲイリー・デイビツド
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EIDP Inc
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EI Du Pont de Nemours and Co
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D231/08—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with oxygen or sulfur atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Photoreceptors In Electrophotography (AREA)
JP2004524203A 2002-07-31 2003-07-29 ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法 Expired - Lifetime JP4633462B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40035602P 2002-07-31 2002-07-31
US44645103P 2003-02-11 2003-02-11
PCT/US2003/023820 WO2004011453A2 (en) 2002-07-31 2003-07-29 Method for preparing 3-halo-4,5-dihydro-1h-pyrazoles

Publications (3)

Publication Number Publication Date
JP2005534685A JP2005534685A (ja) 2005-11-17
JP2005534685A5 JP2005534685A5 (enExample) 2006-09-14
JP4633462B2 true JP4633462B2 (ja) 2011-02-16

Family

ID=31191368

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004524203A Expired - Lifetime JP4633462B2 (ja) 2002-07-31 2003-07-29 ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法

Country Status (17)

Country Link
US (2) US7335780B2 (enExample)
EP (2) EP2100889B1 (enExample)
JP (1) JP4633462B2 (enExample)
KR (1) KR101071048B1 (enExample)
AT (2) ATE450523T1 (enExample)
AU (2) AU2003257027B2 (enExample)
BR (1) BRPI0313342B1 (enExample)
CA (1) CA2494047C (enExample)
DE (2) DE60330357D1 (enExample)
DK (2) DK1537097T3 (enExample)
ES (1) ES2334660T3 (enExample)
IL (2) IL165502A (enExample)
MX (2) MX277756B (enExample)
PL (1) PL216029B1 (enExample)
RU (1) RU2326877C2 (enExample)
TW (1) TWI343376B (enExample)
WO (1) WO2004011453A2 (enExample)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002319814A1 (en) * 2001-08-13 2003-03-03 E.I. Du Pont De Nemours And Company Substituted 1h-dihydropyrazoles, their preparation and use
MY142967A (en) * 2001-08-13 2011-01-31 Du Pont Method for controlling particular insect pests by applying anthranilamide compounds
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
DE60226875D1 (de) 2001-08-15 2008-07-10 Du Pont Orthosubstituierte arylamide zur bekämpfung von wirbellosen schädlingen
US7199138B2 (en) 2001-08-16 2007-04-03 E. I. Du Pont De Nemours And Company Substituted anthranilamides for controlling invertebrate pests
TW200724033A (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI326283B (en) 2002-07-31 2010-06-21 Du Pont Method for preparing fused oxazinones
AU2003295491B2 (en) * 2002-11-15 2009-10-08 E.I. Du Pont De Nemours And Company Novel anthranilamide insecticides
TWI289708B (en) 2002-12-25 2007-11-11 Qualcomm Mems Technologies Inc Optical interference type color display
WO2004067528A1 (en) 2003-01-28 2004-08-12 E.I. Du Pont De Nemours And Company Cyano anthranilamide insecticides
TWI367882B (en) * 2003-03-26 2012-07-11 Du Pont Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates
KR20060008336A (ko) * 2003-06-12 2006-01-26 이 아이 듀폰 디 네모아 앤드 캄파니 융합된 옥사지논 제조 방법
US7342705B2 (en) 2004-02-03 2008-03-11 Idc, Llc Spatial light modulator with integrated optical compensation structure
WO2005118552A2 (en) * 2004-04-13 2005-12-15 E.I. Dupont De Nemours And Company Anthranilamide insecticides
US7561323B2 (en) * 2004-09-27 2009-07-14 Idc, Llc Optical films for directing light towards active areas of displays
JP5215669B2 (ja) * 2004-11-18 2013-06-19 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー アントラニルアミド殺虫剤
KR101337159B1 (ko) 2005-03-18 2013-12-05 이 아이 듀폰 디 네모아 앤드 캄파니 브롬을 사용한 2-피라졸린의 피라졸으로의 전환
MX2008002236A (es) * 2005-08-24 2008-03-27 Du Pont Antranilamidas para controlar plagas de invertebrados.
US8872085B2 (en) 2006-10-06 2014-10-28 Qualcomm Mems Technologies, Inc. Display device having front illuminator with turning features
KR101460351B1 (ko) 2006-10-06 2014-11-10 퀄컴 엠이엠에스 테크놀로지스, 인크. 광학적 손실 구조체를 포함하는 표시장치
JP2009001541A (ja) * 2006-12-15 2009-01-08 Ishihara Sangyo Kaisha Ltd 新規ピラゾール化合物を中間体として用いるアントラニルアミド系化合物の製造方法
JP5507045B2 (ja) * 2006-12-15 2014-05-28 石原産業株式会社 アントラニルアミド系化合物の製造方法
CN104496901B (zh) * 2006-12-15 2016-05-25 石原产业株式会社 邻氨基苯甲酰胺系化合物的制造方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
US8068710B2 (en) 2007-12-07 2011-11-29 Qualcomm Mems Technologies, Inc. Decoupled holographic film and diffuser
CN101550130B (zh) * 2008-04-01 2012-11-07 中国中化股份有限公司 一种制备3-卤代-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酰卤的方法
JP5406581B2 (ja) 2008-04-16 2014-02-05 石原産業株式会社 アントラニルアミド系化合物の製造方法
AU2012211165A1 (en) 2011-01-28 2013-07-04 E. I. Du Pont De Nemours And Company Method for preparing 2-aminobenzamide derivatives
US8987461B2 (en) 2012-12-06 2015-03-24 Quanticel Pharmaceuticals, Inc. Histone demethylase inhibitors
WO2020026259A1 (en) * 2018-07-31 2020-02-06 Sumitomo Chemical India Ltd. Ethyl 2-bromo-4-[2-(3-halopyridin-2-yl)-hydrazinyl]-4-oxobutanoate hbr salt, method of preparation and use thereof
EA202191554A1 (ru) 2018-12-03 2021-09-02 Фмк Корпорейшн Способ получения n-фенилпиразол-1-карбоксамидов
KR20220157967A (ko) 2020-03-25 2022-11-29 이시하라 산교 가부시끼가이샤 시클라닐리프롤의 제조 중간체의 제조 방법
CN114057686A (zh) * 2020-08-05 2022-02-18 沈阳中化农药化工研发有限公司 一种溴代吡唑羧酸酯类化合物的制备方法
AR126069A1 (es) * 2021-06-04 2023-09-06 Pi Industries Ltd Un proceso novedoso para la preparación de diamidas antranílicas
TW202342443A (zh) * 2022-01-31 2023-11-01 美商富曼西公司 用於製備３－溴－１－（３－氯吡啶－２－基）－４，５－二氫－１ｈ－吡唑－５－甲酸乙酯之方法
TW202409000A (zh) 2022-08-29 2024-03-01 美商富曼西公司 用於製備３－鹵代－４，５－二氫－１ｈ－吡唑之高效新方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3577471A (en) * 1968-02-01 1971-05-04 Gulf Research Development Co Halogen interchange process
GB1410191A (en) 1972-02-10 1975-10-15 Minnesota Mining & Mfg 3-chloro-1-aryl-2-pyrazolines
US5281571A (en) * 1990-10-18 1994-01-25 Monsanto Company Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles
MY138097A (en) * 2000-03-22 2009-04-30 Du Pont Insecticidal anthranilamides
US6838074B2 (en) * 2001-08-08 2005-01-04 Bristol-Myers Squibb Company Simultaneous imaging of cardiac perfusion and a vitronectin receptor targeted imaging agent
AR036872A1 (es) * 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
TWI371450B (en) * 2001-08-13 2012-09-01 Du Pont Novel substituted dihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use
MY142967A (en) * 2001-08-13 2011-01-31 Du Pont Method for controlling particular insect pests by applying anthranilamide compounds
ITMI20011784A1 (it) 2001-08-13 2003-02-13 Atofina Processo per la preparazione di metacrilammide(maa)da acetoncianidrina
TW200724033A (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI326283B (en) 2002-07-31 2010-06-21 Du Pont Method for preparing fused oxazinones

Also Published As

Publication number Publication date
DK1537097T3 (da) 2010-04-12
RU2005105325A (ru) 2005-07-20
IL201407A (en) 2013-01-31
AU2003257027B2 (en) 2010-09-16
US7335780B2 (en) 2008-02-26
MX338829B (es) 2016-05-03
AU2010257241B2 (en) 2011-11-10
BRPI0313342B1 (pt) 2016-04-19
BR0313342A (pt) 2005-07-12
EP1537097A2 (en) 2005-06-08
US7705160B2 (en) 2010-04-27
CA2494047A1 (en) 2004-02-05
ATE506356T1 (de) 2011-05-15
EP1537097B1 (en) 2009-12-02
ATE450523T1 (de) 2009-12-15
US20080108821A1 (en) 2008-05-08
WO2004011453A3 (en) 2004-03-18
DE60330357D1 (de) 2010-01-14
IL165502A (en) 2010-05-31
US20050215798A1 (en) 2005-09-29
KR101071048B1 (ko) 2011-10-06
AU2010257241A1 (en) 2011-01-13
KR20050026043A (ko) 2005-03-14
DK2100889T3 (da) 2011-08-08
PL375409A1 (en) 2005-11-28
DE60336867D1 (de) 2011-06-01
MXPA05001117A (es) 2005-04-28
EP2100889B1 (en) 2011-04-20
ES2334660T3 (es) 2010-03-15
CA2494047C (en) 2011-05-24
TW200406383A (en) 2004-05-01
IL165502A0 (en) 2006-01-15
JP2005534685A (ja) 2005-11-17
PL216029B1 (pl) 2014-02-28
WO2004011453A2 (en) 2004-02-05
MX277756B (es) 2010-07-30
TWI343376B (en) 2011-06-11
EP2100889A1 (en) 2009-09-16
RU2326877C2 (ru) 2008-06-20
AU2003257027A1 (en) 2004-02-16

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