JP4633462B2 - ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法 - Google Patents

３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法 Download PDF

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Publication number
JP4633462B2
JP4633462B2 JP2004524203A JP2004524203A JP4633462B2 JP 4633462 B2 JP4633462 B2 JP 4633462B2 JP 2004524203 A JP2004524203 A JP 2004524203A JP 2004524203 A JP2004524203 A JP 2004524203A JP 4633462 B2 JP4633462 B2 JP 4633462B2
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Japan
Prior art keywords
formula
alkyl
compound
halogen
dihydro
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JP2004524203A
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Japanese (ja)
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JP2005534685A (ja
JP2005534685A5 (enExample
Inventor
アニス，ゲイリー・デイビツド
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EIDP Inc
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EI Du Pont de Nemours and Co
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D231/08—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with oxygen or sulfur atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2004524203A 2002-07-31 2003-07-29 ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法 Expired - Lifetime JP4633462B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40035602P 2002-07-31 2002-07-31
US44645103P 2003-02-11 2003-02-11
PCT/US2003/023820 WO2004011453A2 (en) 2002-07-31 2003-07-29 Method for preparing 3-halo-4,5-dihydro-1h-pyrazoles

Publications (3)

Publication Number Publication Date
JP2005534685A JP2005534685A (ja) 2005-11-17
JP2005534685A5 JP2005534685A5 (enExample) 2006-09-14
JP4633462B2 true JP4633462B2 (ja) 2011-02-16

Family

ID=31191368

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004524203A Expired - Lifetime JP4633462B2 (ja) 2002-07-31 2003-07-29 ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法

Country Status (17)

Country Link
US (2) US7335780B2 (enExample)
EP (2) EP2100889B1 (enExample)
JP (1) JP4633462B2 (enExample)
KR (1) KR101071048B1 (enExample)
AT (2) ATE450523T1 (enExample)
AU (2) AU2003257027B2 (enExample)
BR (1) BRPI0313342B1 (enExample)
CA (1) CA2494047C (enExample)
DE (2) DE60336867D1 (enExample)
DK (2) DK2100889T3 (enExample)
ES (1) ES2334660T3 (enExample)
IL (2) IL165502A (enExample)
MX (2) MX277756B (enExample)
PL (1) PL216029B1 (enExample)
RU (1) RU2326877C2 (enExample)
TW (1) TWI343376B (enExample)
WO (1) WO2004011453A2 (enExample)

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* Cited by examiner, † Cited by third party
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TWI312274B (en) 2001-08-13 2009-07-21 Du Pont Method for controlling particular insect pests by applying anthranilamide compounds
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
WO2003016282A2 (en) * 2001-08-13 2003-02-27 E.I. Du Pont De Nemours And Company Substituted 1h-dihydropyrazoles, their preparation and use
CN1865258A (zh) 2001-08-15 2006-11-22 纳幕尔杜邦公司 用于控制无脊椎害虫的邻位取代的芳基酰胺化合物
EP1417176B1 (en) 2001-08-16 2008-12-17 E.I. Du Pont De Nemours And Company Substituted anthranilamides for controlling invertebrate pests
TW200724033A (en) * 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI326283B (en) 2002-07-31 2010-06-21 Du Pont Method for preparing fused oxazinones
EP1560820B1 (en) * 2002-11-15 2010-05-26 E.I. Du Pont De Nemours And Company Novel anthranilamide insecticides
TWI289708B (en) 2002-12-25 2007-11-11 Qualcomm Mems Technologies Inc Optical interference type color display
PT1599463E (pt) 2003-01-28 2013-09-03 Du Pont Insecticidas à base de ciano-antranilamida
TWI367882B (en) * 2003-03-26 2012-07-11 Du Pont Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates
WO2004111030A1 (en) * 2003-06-12 2004-12-23 E.I. Dupont De Nemours And Company Method for preparing fused oxazinones
US7342705B2 (en) 2004-02-03 2008-03-11 Idc, Llc Spatial light modulator with integrated optical compensation structure
AU2005250328A1 (en) * 2004-04-13 2005-12-15 E.I. Dupont De Nemours And Company Anthranilamide insecticides
US7561323B2 (en) * 2004-09-27 2009-07-14 Idc, Llc Optical films for directing light towards active areas of displays
KR101292486B1 (ko) * 2004-11-18 2013-08-01 이 아이 듀폰 디 네모아 앤드 캄파니 안트라닐아미드 살충제
ES2385496T3 (es) 2005-03-18 2012-07-25 E.I. Du Pont De Nemours And Company Conversión de 2-pirazolinas en pirazoles utilizando bromo
US8012499B2 (en) * 2005-08-24 2011-09-06 E.I. Du Pont De Nemours And Company Anthranilamides for controlling invertebrate pests
US9019183B2 (en) 2006-10-06 2015-04-28 Qualcomm Mems Technologies, Inc. Optical loss structure integrated in an illumination apparatus
WO2008045207A2 (en) 2006-10-06 2008-04-17 Qualcomm Mems Technologies, Inc. Light guide
CN104496901B (zh) * 2006-12-15 2016-05-25 石原产业株式会社 邻氨基苯甲酰胺系化合物的制造方法
JP2009001541A (ja) * 2006-12-15 2009-01-08 Ishihara Sangyo Kaisha Ltd 新規ピラゾール化合物を中間体として用いるアントラニルアミド系化合物の製造方法
JP5507045B2 (ja) 2006-12-15 2014-05-28 石原産業株式会社 アントラニルアミド系化合物の製造方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
US8068710B2 (en) 2007-12-07 2011-11-29 Qualcomm Mems Technologies, Inc. Decoupled holographic film and diffuser
CN101550130B (zh) * 2008-04-01 2012-11-07 中国中化股份有限公司 一种制备3-卤代-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酰卤的方法
JP5406581B2 (ja) * 2008-04-16 2014-02-05 石原産業株式会社 アントラニルアミド系化合物の製造方法
AU2012211165A1 (en) 2011-01-28 2013-07-04 E. I. Du Pont De Nemours And Company Method for preparing 2-aminobenzamide derivatives
MX2015007205A (es) 2012-12-06 2016-03-31 Quanticel Pharmaceuticals Inc Inhibidores de la desmetilasa de histona.
WO2020026259A1 (en) * 2018-07-31 2020-02-06 Sumitomo Chemical India Ltd. Ethyl 2-bromo-4-[2-(3-halopyridin-2-yl)-hydrazinyl]-4-oxobutanoate hbr salt, method of preparation and use thereof
WO2020117493A1 (en) 2018-12-03 2020-06-11 Fmc Corporation Method for preparing n-phenylpyrazole-1-carboxamides
WO2021193432A1 (ja) 2020-03-25 2021-09-30 石原産業株式会社 シクラニリプロールの製造中間体の製造方法
CN114057686A (zh) * 2020-08-05 2022-02-18 沈阳中化农药化工研发有限公司 一种溴代吡唑羧酸酯类化合物的制备方法
US20240270726A1 (en) * 2021-06-04 2024-08-15 Pi Industries Ltd. A novel process for the preparation of anthranilic diamides
TW202342443A (zh) * 2022-01-31 2023-11-01 美商富曼西公司 用於製備３－溴－１－（３－氯吡啶－２－基）－４，５－二氫－１ｈ－吡唑－５－甲酸乙酯之方法
TW202409000A (zh) 2022-08-29 2024-03-01 美商富曼西公司 用於製備３－鹵代－４，５－二氫－１ｈ－吡唑之高效新方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3577471A (en) * 1968-02-01 1971-05-04 Gulf Research Development Co Halogen interchange process
GB1410191A (en) * 1972-02-10 1975-10-15 Minnesota Mining & Mfg 3-chloro-1-aryl-2-pyrazolines
US5281571A (en) * 1990-10-18 1994-01-25 Monsanto Company Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles
MY138097A (en) * 2000-03-22 2009-04-30 Du Pont Insecticidal anthranilamides
US6838074B2 (en) * 2001-08-08 2005-01-04 Bristol-Myers Squibb Company Simultaneous imaging of cardiac perfusion and a vitronectin receptor targeted imaging agent
TWI312274B (en) 2001-08-13 2009-07-21 Du Pont Method for controlling particular insect pests by applying anthranilamide compounds
TWI327566B (en) * 2001-08-13 2010-07-21 Du Pont Novel substituted ihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
ITMI20011784A1 (it) 2001-08-13 2003-02-13 Atofina Processo per la preparazione di metacrilammide(maa)da acetoncianidrina
TW200724033A (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
TWI326283B (en) 2002-07-31 2010-06-21 Du Pont Method for preparing fused oxazinones

Also Published As

Publication number Publication date
US7705160B2 (en) 2010-04-27
MXPA05001117A (es) 2005-04-28
BRPI0313342B1 (pt) 2016-04-19
MX338829B (es) 2016-05-03
DE60336867D1 (de) 2011-06-01
DE60330357D1 (de) 2010-01-14
IL165502A (en) 2010-05-31
IL165502A0 (en) 2006-01-15
ATE450523T1 (de) 2009-12-15
AU2003257027B2 (en) 2010-09-16
EP1537097A2 (en) 2005-06-08
KR101071048B1 (ko) 2011-10-06
MX277756B (es) 2010-07-30
AU2010257241B2 (en) 2011-11-10
WO2004011453A3 (en) 2004-03-18
CA2494047A1 (en) 2004-02-05
RU2005105325A (ru) 2005-07-20
IL201407A (en) 2013-01-31
EP2100889A1 (en) 2009-09-16
EP1537097B1 (en) 2009-12-02
AU2010257241A1 (en) 2011-01-13
DK1537097T3 (da) 2010-04-12
WO2004011453A2 (en) 2004-02-05
AU2003257027A1 (en) 2004-02-16
PL216029B1 (pl) 2014-02-28
TW200406383A (en) 2004-05-01
ES2334660T3 (es) 2010-03-15
DK2100889T3 (da) 2011-08-08
CA2494047C (en) 2011-05-24
US20050215798A1 (en) 2005-09-29
JP2005534685A (ja) 2005-11-17
BR0313342A (pt) 2005-07-12
ATE506356T1 (de) 2011-05-15
EP2100889B1 (en) 2011-04-20
KR20050026043A (ko) 2005-03-14
US20080108821A1 (en) 2008-05-08
US7335780B2 (en) 2008-02-26
TWI343376B (en) 2011-06-11
RU2326877C2 (ru) 2008-06-20
PL375409A1 (en) 2005-11-28

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