JP2005534685A5 - - Google Patents
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- Publication number
- JP2005534685A5 JP2005534685A5 JP2004524203A JP2004524203A JP2005534685A5 JP 2005534685 A5 JP2005534685 A5 JP 2005534685A5 JP 2004524203 A JP2004524203 A JP 2004524203A JP 2004524203 A JP2004524203 A JP 2004524203A JP 2005534685 A5 JP2005534685 A5 JP 2005534685A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- formula
- halogen
- compound
- optionally substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 238000000034 method Methods 0.000 claims description 24
- 229910052736 halogen Inorganic materials 0.000 claims description 16
- 150000002367 halogens Chemical class 0.000 claims description 16
- 229910052801 chlorine Inorganic materials 0.000 claims description 15
- 229910052794 bromium Inorganic materials 0.000 claims description 10
- 125000000217 alkyl group Chemical group 0.000 claims description 9
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 9
- 150000001875 compounds Chemical class 0.000 claims description 8
- -1 4,5-dihydro-1H-pyrazole compound Chemical class 0.000 claims description 6
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims description 6
- 125000000590 4-methylphenyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1*)C([H])([H])[H] 0.000 claims description 5
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 4
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 4
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 4
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 4
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 claims description 4
- 125000006650 (C2-C4) alkynyl group Chemical group 0.000 claims description 4
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 4
- 125000004663 dialkyl amino group Chemical group 0.000 claims description 4
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims description 4
- 229910052731 fluorine Inorganic materials 0.000 claims description 4
- 125000001188 haloalkyl group Chemical group 0.000 claims description 4
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 4
- 239000002904 solvent Substances 0.000 claims description 4
- 125000001424 substituent group Chemical group 0.000 claims description 4
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 claims description 4
- 150000001721 carbon Chemical group 0.000 claims description 2
- 229910052799 carbon Inorganic materials 0.000 claims description 2
- 229910052740 iodine Inorganic materials 0.000 claims description 2
- WEVYAHXRMPXWCK-UHFFFAOYSA-N Acetonitrile Chemical compound CC#N WEVYAHXRMPXWCK-UHFFFAOYSA-N 0.000 description 3
- YMWUJEATGCHHMB-UHFFFAOYSA-N Dichloromethane Chemical compound ClCCl YMWUJEATGCHHMB-UHFFFAOYSA-N 0.000 description 3
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 description 3
- HQQTZCPKNZVLFF-UHFFFAOYSA-N 4h-1,2-benzoxazin-3-one Chemical class C1=CC=C2ONC(=O)CC2=C1 HQQTZCPKNZVLFF-UHFFFAOYSA-N 0.000 description 2
- HEDRZPFGACZZDS-UHFFFAOYSA-N Chloroform Chemical compound ClC(Cl)Cl HEDRZPFGACZZDS-UHFFFAOYSA-N 0.000 description 2
- WYURNTSHIVDZCO-UHFFFAOYSA-N Tetrahydrofuran Chemical compound C1CCOC1 WYURNTSHIVDZCO-UHFFFAOYSA-N 0.000 description 2
- PXBFMLJZNCDSMP-UHFFFAOYSA-N 2-Aminobenzamide Chemical class NC(=O)C1=CC=CC=C1N PXBFMLJZNCDSMP-UHFFFAOYSA-N 0.000 description 1
- 0 CC1(CN(*)N=C(*)C1)N(C)C Chemical compound CC1(CN(*)N=C(*)C1)N(C)C 0.000 description 1
- 150000001412 amines Chemical class 0.000 description 1
- 125000000623 heterocyclic group Chemical group 0.000 description 1
- 238000010992 reflux Methods 0.000 description 1
- 239000000126 substance Substances 0.000 description 1
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40035602P | 2002-07-31 | 2002-07-31 | |
| US44645103P | 2003-02-11 | 2003-02-11 | |
| PCT/US2003/023820 WO2004011453A2 (en) | 2002-07-31 | 2003-07-29 | Method for preparing 3-halo-4,5-dihydro-1h-pyrazoles |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005534685A JP2005534685A (ja) | 2005-11-17 |
| JP2005534685A5 true JP2005534685A5 (enExample) | 2006-09-14 |
| JP4633462B2 JP4633462B2 (ja) | 2011-02-16 |
Family
ID=31191368
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004524203A Expired - Lifetime JP4633462B2 (ja) | 2002-07-31 | 2003-07-29 | ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法 |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US7335780B2 (enExample) |
| EP (2) | EP2100889B1 (enExample) |
| JP (1) | JP4633462B2 (enExample) |
| KR (1) | KR101071048B1 (enExample) |
| AT (2) | ATE450523T1 (enExample) |
| AU (2) | AU2003257027B2 (enExample) |
| BR (1) | BRPI0313342B1 (enExample) |
| CA (1) | CA2494047C (enExample) |
| DE (2) | DE60330357D1 (enExample) |
| DK (2) | DK1537097T3 (enExample) |
| ES (1) | ES2334660T3 (enExample) |
| IL (2) | IL165502A (enExample) |
| MX (2) | MX277756B (enExample) |
| PL (1) | PL216029B1 (enExample) |
| RU (1) | RU2326877C2 (enExample) |
| TW (1) | TWI343376B (enExample) |
| WO (1) | WO2004011453A2 (enExample) |
Families Citing this family (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2002319814A1 (en) * | 2001-08-13 | 2003-03-03 | E.I. Du Pont De Nemours And Company | Substituted 1h-dihydropyrazoles, their preparation and use |
| MY142967A (en) * | 2001-08-13 | 2011-01-31 | Du Pont | Method for controlling particular insect pests by applying anthranilamide compounds |
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| DE60226875D1 (de) | 2001-08-15 | 2008-07-10 | Du Pont | Orthosubstituierte arylamide zur bekämpfung von wirbellosen schädlingen |
| US7199138B2 (en) | 2001-08-16 | 2007-04-03 | E. I. Du Pont De Nemours And Company | Substituted anthranilamides for controlling invertebrate pests |
| TW200724033A (en) | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| TWI326283B (en) | 2002-07-31 | 2010-06-21 | Du Pont | Method for preparing fused oxazinones |
| AU2003295491B2 (en) * | 2002-11-15 | 2009-10-08 | E.I. Du Pont De Nemours And Company | Novel anthranilamide insecticides |
| TWI289708B (en) | 2002-12-25 | 2007-11-11 | Qualcomm Mems Technologies Inc | Optical interference type color display |
| WO2004067528A1 (en) | 2003-01-28 | 2004-08-12 | E.I. Du Pont De Nemours And Company | Cyano anthranilamide insecticides |
| TWI367882B (en) * | 2003-03-26 | 2012-07-11 | Du Pont | Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates |
| KR20060008336A (ko) * | 2003-06-12 | 2006-01-26 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 융합된 옥사지논 제조 방법 |
| US7342705B2 (en) | 2004-02-03 | 2008-03-11 | Idc, Llc | Spatial light modulator with integrated optical compensation structure |
| WO2005118552A2 (en) * | 2004-04-13 | 2005-12-15 | E.I. Dupont De Nemours And Company | Anthranilamide insecticides |
| US7561323B2 (en) * | 2004-09-27 | 2009-07-14 | Idc, Llc | Optical films for directing light towards active areas of displays |
| JP5215669B2 (ja) * | 2004-11-18 | 2013-06-19 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | アントラニルアミド殺虫剤 |
| KR101337159B1 (ko) | 2005-03-18 | 2013-12-05 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 브롬을 사용한 2-피라졸린의 피라졸으로의 전환 |
| MX2008002236A (es) * | 2005-08-24 | 2008-03-27 | Du Pont | Antranilamidas para controlar plagas de invertebrados. |
| US8872085B2 (en) | 2006-10-06 | 2014-10-28 | Qualcomm Mems Technologies, Inc. | Display device having front illuminator with turning features |
| KR101460351B1 (ko) | 2006-10-06 | 2014-11-10 | 퀄컴 엠이엠에스 테크놀로지스, 인크. | 광학적 손실 구조체를 포함하는 표시장치 |
| JP2009001541A (ja) * | 2006-12-15 | 2009-01-08 | Ishihara Sangyo Kaisha Ltd | 新規ピラゾール化合物を中間体として用いるアントラニルアミド系化合物の製造方法 |
| JP5507045B2 (ja) * | 2006-12-15 | 2014-05-28 | 石原産業株式会社 | アントラニルアミド系化合物の製造方法 |
| CN104496901B (zh) * | 2006-12-15 | 2016-05-25 | 石原产业株式会社 | 邻氨基苯甲酰胺系化合物的制造方法 |
| TWI415827B (zh) | 2006-12-21 | 2013-11-21 | Du Pont | 製備２-胺基-５-氰基苯甲酸衍生物之方法 |
| US8068710B2 (en) | 2007-12-07 | 2011-11-29 | Qualcomm Mems Technologies, Inc. | Decoupled holographic film and diffuser |
| CN101550130B (zh) * | 2008-04-01 | 2012-11-07 | 中国中化股份有限公司 | 一种制备3-卤代-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酰卤的方法 |
| JP5406581B2 (ja) | 2008-04-16 | 2014-02-05 | 石原産業株式会社 | アントラニルアミド系化合物の製造方法 |
| AU2012211165A1 (en) | 2011-01-28 | 2013-07-04 | E. I. Du Pont De Nemours And Company | Method for preparing 2-aminobenzamide derivatives |
| US8987461B2 (en) | 2012-12-06 | 2015-03-24 | Quanticel Pharmaceuticals, Inc. | Histone demethylase inhibitors |
| WO2020026259A1 (en) * | 2018-07-31 | 2020-02-06 | Sumitomo Chemical India Ltd. | Ethyl 2-bromo-4-[2-(3-halopyridin-2-yl)-hydrazinyl]-4-oxobutanoate hbr salt, method of preparation and use thereof |
| EA202191554A1 (ru) | 2018-12-03 | 2021-09-02 | Фмк Корпорейшн | Способ получения n-фенилпиразол-1-карбоксамидов |
| KR20220157967A (ko) | 2020-03-25 | 2022-11-29 | 이시하라 산교 가부시끼가이샤 | 시클라닐리프롤의 제조 중간체의 제조 방법 |
| CN114057686A (zh) * | 2020-08-05 | 2022-02-18 | 沈阳中化农药化工研发有限公司 | 一种溴代吡唑羧酸酯类化合物的制备方法 |
| AR126069A1 (es) * | 2021-06-04 | 2023-09-06 | Pi Industries Ltd | Un proceso novedoso para la preparación de diamidas antranílicas |
| TW202342443A (zh) * | 2022-01-31 | 2023-11-01 | 美商富曼西公司 | 用於製備３－溴－１－（３－氯吡啶－２－基）－４，５－二氫－１ｈ－吡唑－５－甲酸乙酯之方法 |
| TW202409000A (zh) | 2022-08-29 | 2024-03-01 | 美商富曼西公司 | 用於製備３－鹵代－４，５－二氫－１ｈ－吡唑之高效新方法 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3577471A (en) * | 1968-02-01 | 1971-05-04 | Gulf Research Development Co | Halogen interchange process |
| GB1410191A (en) | 1972-02-10 | 1975-10-15 | Minnesota Mining & Mfg | 3-chloro-1-aryl-2-pyrazolines |
| US5281571A (en) * | 1990-10-18 | 1994-01-25 | Monsanto Company | Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles |
| MY138097A (en) * | 2000-03-22 | 2009-04-30 | Du Pont | Insecticidal anthranilamides |
| US6838074B2 (en) * | 2001-08-08 | 2005-01-04 | Bristol-Myers Squibb Company | Simultaneous imaging of cardiac perfusion and a vitronectin receptor targeted imaging agent |
| AR036872A1 (es) * | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| TWI371450B (en) * | 2001-08-13 | 2012-09-01 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use |
| MY142967A (en) * | 2001-08-13 | 2011-01-31 | Du Pont | Method for controlling particular insect pests by applying anthranilamide compounds |
| ITMI20011784A1 (it) | 2001-08-13 | 2003-02-13 | Atofina | Processo per la preparazione di metacrilammide(maa)da acetoncianidrina |
| TW200724033A (en) | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| TWI326283B (en) | 2002-07-31 | 2010-06-21 | Du Pont | Method for preparing fused oxazinones |
-
2003
- 2003-07-02 TW TW092118075A patent/TWI343376B/zh not_active IP Right Cessation
- 2003-07-29 RU RU2005105325/04A patent/RU2326877C2/ru active
- 2003-07-29 DE DE60330357T patent/DE60330357D1/de not_active Expired - Lifetime
- 2003-07-29 MX MXPA05001117 patent/MX277756B/es unknown
- 2003-07-29 KR KR1020057001599A patent/KR101071048B1/ko not_active Expired - Lifetime
- 2003-07-29 AU AU2003257027A patent/AU2003257027B2/en not_active Expired
- 2003-07-29 MX MX2010000157A patent/MX338829B/es active IP Right Grant
- 2003-07-29 DK DK03772096.8T patent/DK1537097T3/da active
- 2003-07-29 DK DK09008363.5T patent/DK2100889T3/da active
- 2003-07-29 AT AT03772096T patent/ATE450523T1/de active
- 2003-07-29 CA CA2494047A patent/CA2494047C/en not_active Expired - Fee Related
- 2003-07-29 BR BRPI0313342A patent/BRPI0313342B1/pt active IP Right Grant
- 2003-07-29 EP EP09008363A patent/EP2100889B1/en not_active Expired - Lifetime
- 2003-07-29 ES ES03772096T patent/ES2334660T3/es not_active Expired - Lifetime
- 2003-07-29 US US10/518,325 patent/US7335780B2/en not_active Expired - Lifetime
- 2003-07-29 JP JP2004524203A patent/JP4633462B2/ja not_active Expired - Lifetime
- 2003-07-29 PL PL375409A patent/PL216029B1/pl unknown
- 2003-07-29 AT AT09008363T patent/ATE506356T1/de active
- 2003-07-29 DE DE60336867T patent/DE60336867D1/de not_active Expired - Lifetime
- 2003-07-29 EP EP03772096A patent/EP1537097B1/en not_active Expired - Lifetime
- 2003-07-29 WO PCT/US2003/023820 patent/WO2004011453A2/en not_active Ceased
-
2004
- 2004-12-01 IL IL165502A patent/IL165502A/en active IP Right Grant
- 2004-12-01 IL IL201407A patent/IL201407A/en active IP Right Grant
-
2007
- 2007-12-21 US US12/004,902 patent/US7705160B2/en not_active Expired - Lifetime
-
2010
- 2010-12-16 AU AU2010257241A patent/AU2010257241B2/en not_active Expired
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