JP4329291B2 - 含窒素五員環化合物 - Google Patents

含窒素五員環化合物 Download PDF

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Publication number
JP4329291B2
JP4329291B2 JP2001309559A JP2001309559A JP4329291B2 JP 4329291 B2 JP4329291 B2 JP 4329291B2 JP 2001309559 A JP2001309559 A JP 2001309559A JP 2001309559 A JP2001309559 A JP 2001309559A JP 4329291 B2 JP4329291 B2 JP 4329291B2
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group
compound
trans
solvent
residue
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JP2001309559A
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English (en)
Japanese (ja)
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JP2002356472A5 (US07816364-20101019-C00114.png
JP2002356472A (ja
Inventor
公助 安田
啓氏 森本
三郎 河南
匡毅 彦田
健 松本
健司 荒川
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Mitsubishi Tanabe Pharma Corp
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Mitsubishi Tanabe Pharma Corp
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Priority to JP2001309559A priority Critical patent/JP4329291B2/ja
Publication of JP2002356472A publication Critical patent/JP2002356472A/ja
Publication of JP2002356472A5 publication Critical patent/JP2002356472A5/ja
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Publication of JP4329291B2 publication Critical patent/JP4329291B2/ja
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP2001309559A 2000-10-06 2001-10-05 含窒素五員環化合物 Expired - Fee Related JP4329291B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2001309559A JP4329291B2 (ja) 2000-10-06 2001-10-05 含窒素五員環化合物

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP2000308528 2000-10-06
JP2000-308528 2000-10-06
JP2000-312562 2000-10-12
JP2000312562 2000-10-12
JP2001099251 2001-03-30
JP2001-99251 2001-03-30
JP2001309559A JP4329291B2 (ja) 2000-10-06 2001-10-05 含窒素五員環化合物

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2005105732A Division JP2005200427A (ja) 2000-10-06 2005-04-01 含窒素五員環化合物

Publications (3)

Publication Number Publication Date
JP2002356472A JP2002356472A (ja) 2002-12-13
JP2002356472A5 JP2002356472A5 (US07816364-20101019-C00114.png) 2005-09-15
JP4329291B2 true JP4329291B2 (ja) 2009-09-09

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JP2001309559A Expired - Fee Related JP4329291B2 (ja) 2000-10-06 2001-10-05 含窒素五員環化合物

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JP (1) JP4329291B2 (US07816364-20101019-C00114.png)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050197350A1 (en) * 2003-03-31 2005-09-08 Taisho Pharmaceutical Co., Ltd. Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
KR101146849B1 (ko) * 2003-12-11 2012-05-16 미쓰비시 타나베 파마 코퍼레이션 α-아미노산 유도체 및 그 의약 용도
ATE537141T1 (de) 2004-02-05 2011-12-15 Kyorin Seiyaku Kk Bicycloesterderivat
KR20060129021A (ko) * 2004-02-18 2006-12-14 교린 세이야꾸 가부시키 가이샤 비시클로아미드 유도체
WO2005082847A1 (ja) * 2004-02-27 2005-09-09 Kyorin Pharmaceutical Co., Ltd. ビシクロ誘導体
DE102004023632A1 (de) * 2004-05-10 2005-12-08 Grünenthal GmbH Substituierte Cyclohexylcarbonsäure-Derivate
US7601714B2 (en) * 2004-07-08 2009-10-13 Boehringer Ingelheim Pharmaceuticals, Inc. Pyrimidine derivatives useful as inhibitors of PKC-theta
EP1794120B1 (en) * 2004-07-23 2012-04-11 Nuada, LLC Peptidase inhibitors
AP2007003973A0 (en) * 2004-10-12 2007-07-30 Glenmark Pharmaceuticals Sa Novel dideptidyl peptidase IV inhibitors, pharmaceutical compositions containing them, and proces for their preparation
DOP2006000008A (es) 2005-01-10 2006-08-31 Arena Pharm Inc Terapia combinada para el tratamiento de la diabetes y afecciones relacionadas y para el tratamiento de afecciones que mejoran mediante un incremento de la concentración sanguínea de glp-1
CA2645154C (en) 2006-03-08 2011-11-29 Kyorin Pharmaceutical Co., Ltd. Method for producing aminoacetylpyrrolidinecarbonitrile derivative and production intermediate thereof
DK1971862T3 (da) 2006-04-11 2011-02-14 Arena Pharm Inc Fremgangsmåder til anvendelse af GPR119-receptor til identificering af forbindelser anvendelige til øgning af knoglemasse hos en person
PE20071221A1 (es) 2006-04-11 2007-12-14 Arena Pharm Inc Agonistas del receptor gpr119 en metodos para aumentar la masa osea y para tratar la osteoporosis y otras afecciones caracterizadas por masa osea baja, y la terapia combinada relacionada a estos agonistas
JP2009190971A (ja) * 2006-06-06 2009-08-27 Mitsubishi Tanabe Pharma Corp ２−シアノピロリジン誘導体
ATE550319T1 (de) 2007-03-22 2012-04-15 Kyorin Seiyaku Kk Verfahren zur herstellung eines aminoacetylpyrrolidincarbonitrilderivats
JP2011509289A (ja) * 2008-01-10 2011-03-24 サン・ファーマ・アドバンスド・リサーチ・カンパニー・リミテッド 新規なアシルシアノピロリジン誘導体
EP2108960A1 (en) 2008-04-07 2009-10-14 Arena Pharmaceuticals, Inc. Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditons modulated by PYY
CN102119139A (zh) 2008-08-07 2011-07-06 杏林制药株式会社 二环[2.2.2]辛胺衍生物的制造方法
AR077642A1 (es) 2009-07-09 2011-09-14 Arena Pharm Inc Moduladores del metabolismo y el tratamiento de trastornos relacionados con el mismo
MX2012011631A (es) 2010-04-06 2013-01-18 Arena Pharm Inc Moduladores del receptor gpr119 y el tratamiento de trastornos relacionados con el mismo.
US10894787B2 (en) 2010-09-22 2021-01-19 Arena Pharmaceuticals, Inc. Modulators of the GPR119 receptor and the treatment of disorders related thereto
US20140018371A1 (en) 2011-04-01 2014-01-16 Arena Pharmaceuticals, Inc. Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto
US20140066369A1 (en) 2011-04-19 2014-03-06 Arena Pharmaceuticals, Inc. Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto
US20140038889A1 (en) 2011-04-22 2014-02-06 Arena Pharmaceuticals, Inc. Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto
WO2012145604A1 (en) 2011-04-22 2012-10-26 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012170702A1 (en) 2011-06-08 2012-12-13 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2013055910A1 (en) 2011-10-12 2013-04-18 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2014074668A1 (en) 2012-11-08 2014-05-15 Arena Pharmaceuticals, Inc. Modulators of gpr119 and the treatment of disorders related thereto
CN107683135A (zh) 2015-03-09 2018-02-09 因特克林医疗有限公司 用于治疗非酒精性脂肪肝疾病和/或脂肪营养不良的方法
SG11201909046XA (en) 2017-04-03 2019-10-30 Coherus Biosciences Inc PPARγ AGONIST FOR TREATMENT OF PROGRESSIVE SUPRANUCLEAR PALSY

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Publication number Publication date
JP2002356472A (ja) 2002-12-13

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